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5-HT Receptor
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN12245 | (S)-4-((3-(2-(Dimethylamino)ethyl)-1H-indol-5-yl)methyl)oxazolidin-2-one | 139264-17-8 | Zolmitriptan is an agonist of 5-HT1B/5-HT1D receptors with anti-migraine properties. |
| CSN12542 | Ziprasidone | 146939-27-7 | Ziprasidone is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity. |
| CSN12748 | Ziprasidone HCl | 122883-93-6 | Ziprasidone HCl is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity, and is used in the treatment of schizophrenia and bipolar disorder. |
| CSN12812 | Ziprasidone HCl monohydrate | 138982-67-9 | Ziprasidone HCl H2O is a full antagonist of D2 receptors and of 5-HT2A receptors and is a partial agonist of 5-HT1A receptors, of 5-HT2C receptors and 5-HT1D receptors, used as an atypical antipsychoticfor the treatment of schizophrenia as well as acute mania and mixed states associated with bipolar disorder. |
| CSN12928 | Vortioxetine | 508233-74-7 | Vortioxetine is a 5-HT3, 5-HT1D, and 5-HT7 antagonist, a 5-HT1A agonist, and a 5-HT1B partial agonist. |
| CSN12929 | Vortioxetine HBr | 960203-27-4 | Vortioxetine HCl, a multimodal serotonergic agent, inhibits 5-HT1A, 5-HT1B, 5-HT3A, 5-HT7 receptor and SERT with IC50 of 15 nM, 33 nM, 3.7 nM, 19 nM and 1.6 nM, respectively. |
| CSN12174 | Urapidil | 34661-75-1 | Urapidil is a sympatholytic antihypertensive drug. |
| CSN13073 | Tropisetron | 89565-68-4 | Tropisetron is a selective 5-HT3 receptor antagonist and α7-nicotinic receptor agonist with an IC50 of 70.1 ± 0.9 nM for 5-HT3 receptor. |
| CSN12150 | Trimipramine maleate | 521-78-8 | Trimipramine maleate is a serotonin transport and norepinephrine uptake blocker, is a tricyclic antidepressant (TCA) with antipsychotic and sedative properties. |
| CSN12786 | Trazodone | 19794-93-5 | Trazodone is an antidepressant of the serotonin antagonist and reuptake inhibitor (SARI) class. |
| CSN12597 | Trazodone HCl | 25332-39-2 | Trazodone HCl is a selective serotonin reuptake inhibitor and 5HT2 receptor antagonist, used as an antidepressant medication. |
| CSN12475 | Sumatriptan succinate | 103628-48-4 | Sumatriptan Succinate can selectively bind to and activate 5-HT1 receptors. |
| CSN11920 | Setiptiline | 57262-94-9 | Setiptiline is a serotonin receptor antagonist. |
| CSN13121 | SB-269970 HCl | 261901-57-9 | SB-269970 HCl is a HCl salt form of SB-269970, which is a 5-HT7 receptor antagonist with pKi of 8.3 and exhibits > 50-fold selectivity against other receptors. |
| CSN13111 | SB 242084 2HCl | 1049747-87-6 | SB-242084 2HCl is a selective and brain-penetrant antagonist for the 5HT2C receptor. |
| CSN11875 | Rupatadine | 158876-82-5 | Rupatadine is a potent dual PAF/H1 antagonist with Ki of 0.55/0.1 μM (rabbit platelet membranes/guinea pig cerebellum membranes). |
| CSN12847 | RS-127445 HCl | 199864-86-3 | RS-127445 is a selective, high affinity and orally bioavailable serotonin 5-HT2B receptor antagonist. RS-127445 is found to have nanomolar affinity for the 5-HT2B receptor (pKi=9.5) and 1,000 fold selectivity for this receptor as compared to numerous other receptor and ion channel binding sites. |
| CSN11853 | 2-(5-((1H-1,2,4-Triazol-1-yl)methyl)-1H-indol-3-yl)-N,N-dimethylethanamine | 144034-80-0 | Rizatriptan a selective 5-HT1 receptor agonist used for the treatment of migraine headaches. |
| CSN11849 | Ritanserin | 87051-43-2 | Ritanserin is a serotonin receptor antagonist which was never marketed for clinical use but has been used in scientific research. |
| CSN12479 | Risperidone | 106266-06-2 | Risperidone is a multiple-target antipsychotic with high affinity for 5-HT2A and D2 receptors, alpha 1, alpha 2 and H1 receptors. |
| CSN11813 | Quetiapine | 111974-69-7 | Quetiapine is an atypical antipsychotic used in the treatment of schizophrenia, bipolar I mania, bipolar II depression, bipolar I depression. |
| CSN11812 | Quetiapine hemifumarate | 111974-72-2 | Quetiapine Fumarate is a second-generation antipsychotic with affinity for D2, 5-HT2A, H1, alpha 1 and 5-HT1A receptors, used as an atypical antipsychotic for the treatment of schizophrenia, bipolar disorder, and major depressive disorder. |
| CSN11795 | Prucalopride | 179474-81-8 | Prucalopride is a high-affinity 5-HT4 receptor agonist。 |
| CSN13137 | Ondansetron | 99614-02-5 | Ondansetron is a serotonin 5-HT3 receptor antagonist used mainly as anantiemetic (to treat nausea and vomiting), often following chemotherapy. |
| CSN13092 | 1-(3-(4-(3-Chlorophenyl)piperazin-1-yl)propyl)-3-ethyl-4-(2-phenoxyethyl)-1H-1,2,4-triazol-5(4H)-one hydrochloride | 82752-99-6 | Nefazodone HCl is a 5-HT2A receptor antagonist with Ki of 5.8 nM and an inhibitor of serotonin and noradrenalin uptake with IC50s of 290 and 300 nM respectively, it is an antidepressant drug. |
| CSN12511 | Naratriptan | 121679-13-8 | Naratriptan is a selective 5-HT1 receptor subtype agonist and is a triptan drug that is used for the treatment of migraine headaches. |
| CSN12745 | Naratriptan HCl | 143388-64-1 | Naratriptan HCl is a selective sulfonamide 5-HT1D and 5-HT1B receptor agonist with anti-migraine property . |
| CSN11510 | Naftidrofuryl | 31329-57-4 | Naftidrofuryl is a vasodilator used in the management of peripheral and cerebral vascular disorders. |
| CSN11473 | Mosapride Citrate | 112885-42-4 | Mosapride Citrate is both a selective 5HT4 agonist and a 5HT3 antagonist, use as a gastroprokinetic agent. |
| CSN12491 | Mosapride | 112885-41-3 | Mosapride a selective 5HT4 agonist used as a gastroprokinetic agent. |
| CSN11451 | Mirtazapine | 85650-52-8 | Mirtazapine is a potent tetracyclic antidepressant. |
| CSN13120 | LY 344864 | 186544-26-3 | LY344864 is a selective receptor agonist with an affinity of 6 nM (Ki) at the recently cloned 5-HT1F receptor. |
| CSN12876 | LY310762 | 192927-92-7 | LY310762 is a potent and selective antagonist for the 5-HT1D serotonin receptor with EC50 value of 31 nM. |
| CSN12364 | Lurasidone HCl | 367514-88-3 | Lurasidone HCl is a multiple-target antagonist of dopamine D2 receptor, 5-HT2 receptor, 5-HT7 receptor, adrenergic α2A and α2C receptors, also works as a partial 5-HT1A receptor agonist. It used as an atypical antipsychotic medication for the treatment of several mental disorders. |
| CSN11336 | Loxapine succinate | 27833-64-3 | Loxapine succinate salt is an multiple-target antagonist of both D2/D4 dopamine receptor and 5-HT2A/2B, 5-H7 serotonin receptor, used as an antipsychotic agent. |
| CSN12407 | Loxapine | 1977-10-2 | Loxapine succinate is a D2DR and D4DR inhibitor, serotonergic receptor antagonist and also a dibenzoxazepine anti-psychotic agent. |
| CSN11251 | 3-(2-(4-(4-Fluorobenzoyl)piperidin-1-yl)ethyl)quinazoline-2,4(1H,3H)-dione (2R,3R)-2,3-dihydroxysuccinate | 83846-83-7 | Ketanserin Tartrate is a water soluble selective 5-HT2A and 5-HT1D antagonist. |
| CSN11471 | Indeloxazine hydrochloride | 65043-22-3 | Indeloxazine HCl is an antidepressant and cerebral activator. |
| CSN11195 | 3-(10,11-Dihydro-5H-dibenzo[b,f]azepin-5-yl)-N,N-dimethylpropan-1-amine hydrochloride | 113-52-0 | Imipramine HCl is a tricyclic inhibitor of both serotonin and norepinephrine transporters with Ki values of 7.7 nM and 67 nM, respectively. |
| CSN11188 | Iloperidone | 133454-47-4 | Iloperidone is a D2/5-HT2 receptor antagonist, which is an atypical antipsychotic for the treatment of schizophrenia symptoms. |
| CSN11019 | Flibanserin | 167933-07-5 | Flibanserin is a serotonergic antidepressant used to treat hypoactive sexual desire disorder. It is also a P-Glycoprotein Inhibitor. |
| CSN12986 | Buspirone | 36505-84-7 | Buspirone is an anxiolytic drug that is primarily used to treat generalized anxiety disorder (GAD). |
| CSN12514 | 6-Chloro-4-methyl-3-oxo-N-(quinuclidin-3-yl)-3,4-dihydro-2H-benzo[b][1,4]oxazine-8-carboxamide hydrochloride | 123040-16-4 | Azasetron HCl is a potent, selective and competitive 5-HT3 receptor antagonist with pKi value of 9.27. |
| CSN12652 | trans-5-Chloro-2-methyl-2,3,3a,12b-tetrahydro-1H-dibenzo[2,3:6,7]oxepino[4,5-c]pyrrole maleate | 85650-56-2 | Asenapine Maleate is a 5-HT and dopamine D2 receptor antagonist used to treat schizophrenia and bipolar mania. |
| CSN12124 | Asenapine | 65576-45-6 | Asenapine inhibits adrenergic receptor (α1, α2A, α2B, α2C) with Ki of 0.25-1.2 nM and also inhibits 5-HT receptor(1A, 1B, 2A, 2B, 2C, 5A, 6, 7) with Ki of 0.03-4.0 nM. |
| CSN12463 | 7-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one | 129722-12-9 | Aripiprazole is a multiple-target agent used to treat schizophrenia and bipolar disorder, working as both a silent antagonist and a high-efficacy partial agonist of D2 receptor, as well as works as a partial agonist of 5-HT1A/5-HT2A, 5-HT2 receptor,a potent inverse agonist of 5-HT2B receptor, a functional antagonist of 5-HT7 receptor. |
