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| Cat. No. | Product Name | CAS No. | Information |
|---|---|---|---|
| CSN10004 | Cladribine | 4291-63-8 | Cladribine is an adenosine deaminase inhibitor used to treat hairy cell leukemia and multiple sclerosis. For U266, RPMI8226, and MM1.S cells, its IC50 |
| CSN10240 | Aliskiren | 173334-57-1 | Aliskiren is a renin inhibitor with IC50 of 1.5 nM. |
| CSN10349 | Atazanavir | 198904-31-3 | Atazanavir is a protease inhibitor used as an antiretroviral medication to treat and prevent HIV/AIDS. |
| CSN10369 | Azilsartan | 147403-03-0 | Azilsartan is an orally available angiotensin II type 1 (AT1) receptor antagonist with IC50 value of 2.6 nM. |
| CSN10496 | Ambrisentan | 177036-94-1 | Ambrisentan is an oral, once-daily endothelin receptor antagonist that is selective for the endothelin type A receptor (IC50s = 0.251, 0.316, 0.398, 2 |
| CSN10538 | Caffeic Acid Phenethyl Ester | 104594-70-9 | Caffeic acid phenethyl ester, a natural product isolated and purified from the barks of Cinnamomum cassia Presl, is a potent and specific inhibitor of |
| CSN10852 | DMXAA | 117570-53-3 | DMXAA is an apoptosis inducer with anti-vascular activity. It is mSTING agonist, selective for mouse STING over human STING. It Induces IFN-β and cyto |
| CSN10931 | Erlotinib | 183321-74-6 | Erlotinib is an EGFR inhibitor with IC50 of 2 nM, > 1000-fold more sensitive for EGFR than human c-Src or v-Abl. |
| CSN11084 | Gefitinib | 184475-35-2 | Gefitinibis an EGFR inhibitor for Tyr1173, Tyr992, Tyr1173 and Tyr992 in the NR6wtEGFR and NR6W cells with IC50 of 37 nM, 37nM, 26 nM and 57 nM, respe |
| CSN11131 | GW9662 | 22978-25-2 | GW9662 selectively antagonizes PPARγ with IC50 of 3.3 nM. It can inhibit the growth of mammary cancer cells. |
| CSN11187 | GM6001 | 142880-36-2 | GM6001 is a broad spectrum MMPs inhibitor for MMP-1, MMP-2, MMP-3, MMP-7, MMP-8, MMP-9, MMP-12, MMP-14, and MMP-26 with Ki of 0.4 nM, 0.5 nM, 27 nM, 3 |
| CSN11190 | Imatinib | 152459-95-5 | Imatinib is a multi-target inhibitor of v-Abl, c-Kit and PDGFR with IC50 of 0.6 μM, 0.1 μM and 0.1 μM in cell-free or cell-based assays, respectively. |
| CSN11280 | Lenalidomide | 191732-72-6 | Lenalidomide, a analog of thalidomide, is TNF-α secretion inhibitor with IC50 of 13 nM. |
| CSN11339 | Lubiprostone | 136790-76-6 | Lubiprostone is an ClC-2 chloride channel activator used in the treatment of idiopathic chronic constipation. |
| CSN11455 | Montelukast Sodium | 151767-02-1 | Montelukast Sodium is a potent, selective and competitive LTR1 antagonist with IC50 value < 5 nM, possesssing anti-inflammatory and bronchodilating ac |
| CSN11667 | Pemetrexed | 137281-23-3 | Pemetrexed is an antifolate and antimetabolite for TS(thymidylate synthase), DHFR(dihydrofolate reductase) and GARFT(glycinamide ribonucleotide formyl |
| CSN11857 | Roflumilast | 162401-32-3 | Roflumilast is a selective and long-acting inhibitor of PDE-4 with IC50 of 0.8 nM. |
| CSN11862 | Roscovitine | 186692-46-6 | Roscovitine is a potent and selective CDK inhibitor for Cdc2, CDK2 and CDK5 with IC50 of 0.65 μM, 0.7 μM and 0.16 μM and shows little effect on CDK4/6 |
| CSN11899 | SB-203580 | 152121-47-6 | SB-203580 is a p38 MAPK inhibitor with IC50 of 0.3-0.5 μM. |
| CSN12170 | Tyrphostin AG 879 | 148741-30-4 | Tyrphostin AG 879 potently inhibits HER2/ErbB2 with IC50 of 1 μM, 100- and 500-fold higher selective to ErbB2 than PDGFR and EGFR. |
| CSN12304 | BSI-201 | 160003-66-7 | BSI-201 is a PARP1 inhibitor with demonstrated effectiveness in triple-negative breast cancer (TNBC). |
| CSN12327 | Pixantrone Dimaleate | 144675-97-8 | Pixantrone dimaleate is a topoisomerase II inhibitor and DNA intercalator, with anti-tumor activity. Pixantrone dimaleate is an experimental antineopl |
| CSN12330 | Piceatannol | 10083-24-6 | Piceatannol, a natural stilbene, is selective Syk inhibitor extracted from the rhizomes of Polygonum cuspidatum Sieb. et Zucc.. |
| CSN12357 | PD153035 | 153436-54-5 | PD153035 is EGFR inhibitor with Ki and IC50 of 5.2 pM and 29 pM and could rapidly suppress autophosphorylation of EGFR. |
| CSN12358 | AG-1478 | 153436-53-4 | AG-1478 selectively inhibits EGFR with IC50 of 3 nM in cell-free assay. |
| CSN12447 | Fondaparinux Sodium | 114870-03-0 | Fondaparinux sodium is a pentasaccharide inhibitor of antithrombin-dependent factor Xa (IC50 = 40 nM). It can bind to antithrombin III. |
| CSN12489 | Pioglitazone HCl | 112529-15-4 | Pioglitazone HCl is a selective agonist of PPARγ with EC50 of 0.93 μM which is used to treat diabetes. |
| CSN12500 | Combretastatin A4 | 117048-59-6 | Combretastatin A4 is a tubulin polymerization inhibitor with Kd value of 0.4 μM for binding to β-tubulin. |
| CSN12559 | Tenofovir | 147127-20-6 | Tenofovir is an antiretroviral drug known as nucleotide analogue reverse transcriptase inhibitors (NRTIs), which block reverse transcriptase, a crucia |
| CSN12570 | Rosiglitazone Maleate | 155141-29-0 | Rosiglitazone maleate is the maleate form of rosiglitazone which is a high-affinity selective agonist of the peroxisome proliferator-activated recepto |
| CSN12700 | PD153035 HCl | 183322-45-4 | PD153035 HCl is an reversible inhibitor of EGFR with Ki and IC50 of 5.2 pM and 29 pM. |
| CSN12964 | Cabazitaxel | 183133-96-2 | Cabazitaxel is a semi-synthetic derivative of the natural taxoid 10-deacetylbaccatin III with potential antineoplastic activity. Cabazitaxel exerts it |
| CSN13185 | Pomalidomide | 19171-19-8 | Pomalidomide can inhibit LPS-induced TNF-α release with IC50 of 13 nM in PBMCs. |
| CSN13562 | Triapine | 143621-35-6 | Triapine is a ribonucleotide reductase inhibitor and a CDK inhibtor. |
| CSN16276 | PF-06840003 | 198474-05-4 | PF-06840003 is a highly selective orally bioavailable IDO-1 inhibitor with IC50 of 0.41 μM. |
| CSN16424 | Licochalcone A | 58749-22-7 | Licochalcone A, an estrogenic flavanoid, can be an inhibitor of p-glycoprotein and has anti-inflammatory actions. |
| CSN16694 | Metformin HCl | 1115-70-4 | Metformin HCl, a widely used anti-diabetic drug has potential efficacy as an anti-cancer drug, decreasing hyperglycemia in hepatocytes primarily by su |
| CSN16698 | Alendronate Sodium Trihydrate | 121268-17-5 | Alendronate Sodium Trihydrate is an inhibitor of farnesyl diphosphate synthase with IC50 of 460 nM. It is used to treat osteoporosis. |
| CSN16708 | Calcifediol | 19356-17-3 | Calcifediol is an active metabolite of vitamin D. It can inhibit the secretion of parathyroid hormone with 2 nM and commonly used as an indicator of b |
| CSN16716 | Everolimus | 159351-69-6 | Everolimus is a mTOR inhibitor of FKBP12 with IC50 of 1.6-2.4 nM. |
| CSN16720 | Fingolimod HCl | 162359-56-0 | Fingolimod HCl is a S1P antagonist with IC50 of 0.033 nM. |
| CSN16725 | Erlotinib HCl | 183319-69-9 | Erlotinib HCl is a directly acting inhibitor of human EGFR tyrosine kinase with an IC50 of 2 nM. |
| CSN19413 | Polydatin | 27208-80-6 | Polydatin, extracted from the roots ofPolygonum cuspidatumSieb, a widely used traditional Chinese remedies, possesses anti-inflammatory activity in se |
| CSN19473 | Bexarotene | 153559-49-0 | Bexarotene is a selective agonist of RXRβ (IC50 = 24 nM), RXRγ (IC50 = 25 nM) and RXRα (IC50 = 33 nM) with antineoplastic activity. |
| CSN19160 | H 89 2HCl | 130964-39-5 | H 89 2HCl is a potent and selective inhibitor of cyclic AMP-dependent protein kinase (protein kinase A) with IC50 of 48 nM. It also shows weak inhibit |
| CSN16987 | ABT-751 | 141430-65-1 | ABT-751 can inhibit microtubule polymerization through binding to β-tubulin on the colchine site. |
| CSN12943 | Marimastat | 154039-60-8 | Marimastat is a competitive and broad-spectrum MMP inhibitor with IC50 values of 3, 5, 6, 9 and 13 nM for MMP-9, MMP-1, MMP-2, MMP-14 and MMP-7, respe |
| CSN11329 | Lopinavir | 192725-17-0 | Lopinavir is an antiretroviral of the protease inhibitor class, as well as an inhibitor of P-Glycoprotein, Cytochrome P450 3A and Organic Anion Transp |
| CSN13587 | Ritonavir | 155213-67-5 | Ritonavir is both an HIV protease inhibitor and a Cytochrome P450 3A inhibitor. |
| CSN26140 | TRULI | 1424635-83-5 | TRULI is an ATP-competitive inhibitor of Lats kinases. It is a potent, non-toxic, and reversible inhibitor of Hippo signaling which causes Yap-depende |
