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货号 | 产品名称 | CAS号 | 简介 |
---|---|---|---|
CSN20392 | MDL28170 | 88191-84-8 | MDL28170 is a potent, selective inhibitor of calpain and cathepsin B (Ki values are 10 and 25 nM respectively) that does not inhibit trypsin-like seri |
CSN26140 | TRULI | 1424635-83-5 | TRULI is an ATP-competitive inhibitor of Lats kinases. It is a potent, non-toxic, and reversible inhibitor of Hippo signaling which causes Yap-depende |
CSN26180 | PU-02 | 313984-77-9 | PU-02 is an antagonist of serotonin (5-HT) receptor subtype 5-HT3. |
CSN27205 | ILK-IN-3 | 6975-75-3 | ILK-IN-3 is an integrin linked kinase inhibitor. |
CSN27206 | CIL62 | 117593-36-9 | CIL56 is a inducer of regulated, non-apoptotic cell death. It is a lead compound of FIN56, |
CSN27211 | JX06 | 729-46-4 | JX06 is a selective covalent PDK1 inhibitor with IC50 values of 49, 101 and 313nM for PDK-1, PDK-2 and PDK-3, respectively. |
CSN27238 | Nafenopin | 3771-19-5 | Nafenopin is a peroxisome proliferator that is used to promote liver tumors. It has been used as an antihyperlipoproteinemic agent. |
CSN27244 | 2′,5′-Dideoxyadenosine | 6698-26-6 | 2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site with an IC50 of 3 µM . 2',5'-Dideoxyadenosine |
CSN27600 | TD-198946 | 364762-86-7 | TD-198946, a thienoindazole derivative, is a potent chondrogenic agent. |
CSN26189 | Afimoxifene | 68392-35-8 | Afimoxifene is the active metabolite of tamoxifen and a selective estrogen receptor (ER) modulator that is widely used in the therapeutic and chemopre |
CSN27723 | MID-1 | 312608-54-1 | MID-1 is a MG53-IRS-1 interaction disruptor. It abolished MG53-mediated IRS-1 ubiquitination and degradation, as well as sensitized insulin signaling |
CSN27743 | GW806742X | 579515-63-2 | GW806742X is an ATP mimetic MLKL inhibitor with Kd value of 9.3μM, and a VEGFR2 inhibitor with IC50 value of 2nM. |
CSN27773 | mTOR inhibitor-1 | 468747-17-3 | mTOR inhibitor-1 is an ATP-competitive inhibitor of mTOR. It suppressed A549 cell proliferation and induced autophagy. |
CSN27768 | AT-56 | 162640-98-4 | AT 56 is an orally active L-PGDS inhibitor with IC50 value of 95μM. It inhibits the production of PGD2 from PGH2 in vitro, with no effect on PG |
CSN27841 | PFM01 | 1558598-41-6 | PFM 01 is a MRE11 endonuclease inhibitor which can prevent double-stranded break resection. It enhances NHEJ and reduces homologous recombination. |
CSN27839 | NSD2-PWWP1 antagonist 3f | 1210906-48-1 | NSD2-PWWP1 antagonist 3f can bind to the NSD2-PWWP1 domain with Kd value of 3.4μM and abrogates histone H3K36me2 binding to the PWWP1 domain in cells. |
CSN27842 | IT-603 | 292168-90-2 | IT-603 is a c-Rel inhibitor with IC50 value of 3μM. |
CSN27837 | Rhodamine 123 | 62669-70-9 | |
CSN27843 | Sulforhodamine 101 | 60311-02-6 | Sulforhodamine 101, a fluorescent dye (Ex ~586nm, Em ~606nm), is a selective astrocyte marker. |
CSN27848 | GW604714X | 853953-65-8 | GW604714X is a highly specific MPC (mitochondrial pyruvate carrier) inhibitor with Ki value<0.1nM. |
CSN27868 | 16-(S)-ML188 | 1417700-12-9 | 16-(S)-ML188 is a non-covalent SARS-CoV 3CLpro inhibitor with good enzyme and antiviral inhibitory activity. |
CSN27872 | Melatonin Biotin | 2193462-87-0 | Melatonin Biotin is compound conjuncted melatonin with biotin. |
CSN27873 | ChX710 | 2438721-44-7 | ChX710 can boost cellular response to cytosolic DNA via STING. It efficiently primed cellular response to transfected plasmid DNA as assessed by poten |
CSN28337 | Pseudouridine | 1445-07-4 | Pseudouridine is a modified nucleoside. |
CSN27986 | 1,2-DOPC | 4235-95-4 | 1,2-DOPC is a phospholipid utilized for liposome production. |
CSN28422 | MK2-IN-3 | 724711-21-1 | MK2 Inhibitor III is a potent and selective MK-2 inhibitor with IC50 value of 8.5nM. |
CSN28421 | MDK6620 | 304456-62-0 | MDK6620 is a potent and selective IMP1 inhibitor by inhibiting IMP1 binding to c-Myc mRNA with IC50 value of 5μM. It downregulates several mRNA transc |
CSN28430 | GSK2837808A | 1445879-21-9 | GSK2837808A is a potent and selective LDHA and LDHB inhibitor with IC50 values of 2.6nM and 43nM for LDHA and LDHB, respectively. It reduces glucose u |
CSN26245 | TAO Kinase inhibitor 1 | 850467-66-2 | TAO Kinase inhibitor 1 is a selective, ATP-competitive thousand-and-one amino acid kinases (TAOK) inhibitor with IC50s of 11 to 15 nM for TAOK1 and 2, |
CSN28763 | LY293111 | 161172-51-6 | LY293111 is a potent LTB4 receptor antagonist with IC50 values of 17.6nM and 6.3nM for inhibition of the specific binding of radiolabeled-LTB4 to isol |
CSN28765 | MYLS22 | 306959-01-3 | MYLS22 is a first-in-class small molecule-specific OPA1 inhibitor which inhibits tumor angiogenesis, impacts tumor growth and metastatization dependen |
CSN28769 | TKN87180 | 756487-18-0 | TKN8718 is a hydrolyzable ADC linker. |
CSN28768 | Fmoc-Phe-Lys(Boc)-PAB | 206133-42-8 | Fmoc-Phe-Lys(Boc)-PAB is a hydrolyzable ADC linker. |
CSN28771 | 8-Azaadenosine | 10299-44-2 | 8-Azaadenosine is an ADAR1inhibitor. |
CSN28783 | NSC 617145 | 203115-63-3 | NSC 617145 is a WRN helicase inhibitor with IC50 value of 250nM. |
CSN28785 | EGFR-IN-5 | 2225887-26-1 | EGFR-IN-5 is an inhibitor of EGFR with IC50 values of 10.4 nM, 1.1 nM, 34 nM and 7.2 nM for EGFR, EGFRL858R, EGFRL858R/T790M, and EGFRL858R/T790M/C797 |
CSN29557 | CLT-003 | 100823-03-8 | TC11 is a potent inhibitor of tumor cell proliferation and an inducer of apoptosis via activation of caspase-3, 8 and 9. |
CSN29564 | DUN99845 | 727699-84-5 | DUN99845 was reported as a STING inhbiitor, which inhibited the activation of the STING signal pathway and to prevent or treat a STING-mediated disea |
CSN29561 | VU0071063 | 333415-38-6 | VU0071063 can activate native Kir6.2/SUR1 channels, thereby inhibiting glucose-stimulated calcium entry in isolated mouse pancreatic β cells. |