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Adenosine Receptor

Adenosine Receptor

货号 产品名 CAS号 信息
CSN24475 Xanthine amine congener HCl 1783977-95-6 XAC is an adenosine receptor antagonist with IC50 value of 16μM for Adenosine Receptor A2.
CSN19829 Trabodenoson 871108-05-3 Trabodenoson is a potent and highly selective adenosine A1 receptor agonist.
CSN16416 1,3-Dimethyl-1H-purine-2,6(3H,9H)-dione 58-55-9 Theophylline is a natural product present in tea and cocoa, working as a phosphodiesterase inhibitor, adenosine receptor blocker, and histone deacetylase activator.
CSN21258 Tecadenoson 204512-90-3 Tecadenoson is a selective A1 adenosine receptor agonist.
CSN27356 Taminadenant 1337962-47-6 Taminadenant is an antagonist of adenosine receptor.
CSN23108 SCH442416 316173-57-6 SCH-442416 is a selective adenosine A2A receptor antagonist. SCH-442416 binds to human and rat A2A receptors with high affinity (Ki values are 0.048 and 0.5 nM respectively). It displays > 23000-fold selectivity for hA2A over hA1 in vitro with minimal affinity for hA2B and hA3 receptors (IC50 > 10 μM).
CSN23057 PSB-603 1092351-10-4 PSB 603 is a adenosine A2B receptor antagonist with Ki of 0.553 nM.
CSN23056 PSB36 524944-72-7 PSB 36 is a potent and selective A1 adenosine receptor antagonist that displays binding affinity of 0.12 nM for rA1.
CSN23054 PSB-0788 1027513-54-7 PSB 0788 is a potent and selective adenosine A2B receptor antagonist with IC50 of 3.64 nM at human A2B receptor.
CSN21946 Proxyphylline 603-00-9 Proxyphylline is a xanthine-derivatived antagonists of A1 and A2 adenosine receptors, which relaxe smooth muscles, particularly bronchial muscles.
CSN23050 PQ-69 910045-32-8 PQ 69 is a potent and selective A1 receptor inverse agonist taht exhibits high binding affinity at A1 receptor with Kis of 0.07 and 0.96 nM for rat and human receptors respectively.
CSN23113 SDZ-WAG994 130714-47-5 Potent, selective A1 agonist
CSN23153 TC-G 1004 1061747-72-5 Potent and selective A2A antagonist
CSN20000 Neladenoson dalanate 1239309-58-0 Neladenoson dalanate is a potent and selective adenosine A1 receptor agonist, and potentially useful for treatment of cardiovascular diseases.
CSN21751 5'-N-Ethylcarboxamidoadenosine 35920-39-9 NECA, an analog of adenosine, is agonist of adenosine receptors with Kis of 1880, 6660, and 3.5 nM for A1, A2A, and A3, respectively.
CSN22994 N6-Cyclopentyladenosine 41552-82-3 N6-Cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist with Ki of 2.3 nM for human A1 receptor.
CSN25517 (2R,3R,4S,5R)-2-(6-((2-Hydroxyethyl)amino)-9H-purin-9-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol 4338-48-1 N-(2-Hydroxyethyl)adenosine has been studied as an anticonvulsant through the activation of adenosine A1 receptor (AA1R). It attenuates cell death induced by H2O2 through antioxidant action.
CSN24570 MRS1220 183721-15-5 MRS1220 is a potent and highly selective antagonist at the human A3 adenosine receptor. Ki values are 0.65, 305, and 52 nM at hA3, rA1 and rA2A respectively. MRS1220 displays an IC50 > 1 μM for inhibition of binding to rat A3 receptors.
CSN22990 MRS5698 1377273-00-1 MRS 5698 is a high affinity and selective A3 adenosine receptor agonist with Ki ~ 3 nM.
CSN22989 MRS-3777 hemioxalate 1186195-57-2 MRS 3777 Hemioxalate is a high affinity adenosine A3 receptor antagonist with Ki of 47 nM.
CSN22988 MRS 1754 264622-58-4 MRS 1754 is a selective adenosine A2B receptor antagonist with Ki of 1.97 nM for hA2B.
CSN22987 MRS-1706 264622-53-9 MRS 1706 is a potent and selective adenosine A2B receptor inverse agonist with Ki of 1.39 nM.
CSN22873 Rolofylline 136199-02-5 KW 3902 is a Selective adenosine A1 receptor antagonist with Ki of 0.19 nM.
CSN22860 ISAM-140 932191-62-3 ISAM 140 is a high affinity A2B receptor antagonist with Ki of 3.49 nM.
CSN23107 SCH-202676 hydrobromide 265980-25-4 Inhibitor of ligand binding to G-protein-coupled receptors
CSN22848 HEMADO 403842-38-6 HEMADO is a high affinity and selective adenosine A3 receptor agonist with Ki of 1.1 nM for human A3.
CSN22792 DPCPX 102146-07-6 DPCPX is a potent and selective A1 adenosine receptor antagonist, both in vitro and in vivo, with Ki of 3.9 nM for human A1.
CSN23120 Derenofylline 251945-92-3 Derenofylline (SLV 320) is a potent, selective and orally active adenosine A1 receptor antagonist, with Ki values of 1 nM, 200 nM and 398 nM for human A1, A3 and A2A receptors respectively. Derenofylline suppresses cardiac fibrosis and attenuates albuminuria without affecting blood pressure in rats[1].
CSN22838 GS-6201 752222-83-6 CVT-6883 is a selective antagonist of adenosine A2B receptors with Ki of 22 nM for human A2B.
CSN21199 (S)-7-(5-Methylfuran-2-yl)-3-((6-(((tetrahydrofuran-3-yl)oxy)methyl)pyridin-2-yl)methyl)-3H-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine 1202402-40-1 CPI-444 is an orally administered antagonist of the adenosine A2A receptor. Upon oral administration, CPI-444 binds to adenosine A2A receptors expressed on the surface of immune cells, including T-lymphocytes, natural killer (NK) cells, macrophages and dendritic cells (DCs).
CSN24568 CGS 15943 104615-18-1 CGS 15943 is a potent adenosine receptor antagonist with Ki values of 3.5, 4.2, 16 and 51 nM for human A1, A2A, A2B and A3 receptors respectively.
CSN23897 BAY-545 1699717-32-2 BAY-545 is a structure-optimizd adenosine receptor A2B antagonist with IC50 value of of 59 nM.
CSN24164 BAY-218 2162982-11-6 BAY-218 is an AHR antagonist.
CSN22708 BAY 60-6583 910487-58-0 BAY 60-6583 is a potent adenosine A2B receptor agonist with EC50 of 2.83 nM for murine A2B receptor.
CSN27286 BAY 2416964 2242464-44-2 BAY 2416964 is an antagonist of aryl hydrocarbon receptor (AhR) with IC50 of 341 nM.
CSN21201 6-(2-Chloro-6-methylpyridin-4-yl)-5-(4-fluorophenyl)-1,2,4-triazin-3-amine 1321514-06-0 AZD4635 is an A2AR antagonist which can reverse adenosine mediated T cell suppression.
CSN21468 Alloxazine 490-59-5 Alloxazine is a selective antagonist of A2B adenosine receptor.
CSN23524 (2R,3R,4S,5R)-2-(6-Amino-9H-purin-9-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol 58-61-7 Adenosine is a nucleoside that is composed of adenine and d-ribose and plays many important biological roles in addition to being components of DNA and RNA.
CSN21333 Adenosine antagonist-1 431040-19-6 Adenosine antagonist-1 is an adenosine A3 receptor (AA3R) antagonist.
CSN25244 Adenosine amine congener   96760-69-9 Adenosine amine congener hydrate is a potent aqueous-soluble A1 adenosine receptor agonist with Ki value of 0.85nM for binding against [3H]N6-cyclohexyladenosine in rat cerebral cortex membranes.
CSN24753 3-(2-Amino-6-(1-((6-(2-hydroxypropan-2-yl)pyridin-2-yl)methyl)-1H-1,2,3-triazol-4-yl)pyrimidin-4-yl)-2-methylbenzonitrile   2239273-34-6 AB928 is a dual A2aR/A2bR antagonist that inhibits A2aR and A2bR with an equilibrium binding constant of 1.4 and 2 nM, respectively.
CSN18264 A2AR-agonist-1 41552-95-8 A2AR-agonist-1 is a potent A2AR and ENT1 agonist with Ki of 4.39 and 3.47 for A2AR and ENT1.
CSN24565 8-Cyclopentyl-1,3-dimethylxanthine 35873-49-5 8-Cyclopentyl-1,3-dimethylxanthine is a selective antagonist of adenosine A1 receptor with pKi of 7.5-8.
CSN24575 (E)-8-(3-Chlorostyryl)caffeine 147700-11-6 8-(3-Chlorostyryl)caffeine is a selective adenosine A2A receptor antagonist (Ki = 54 nM at rat A2) and monoamine oxidase B (MAO-B) inhibitor (Ki = 100 nM).
CSN22645 CCPA 37739-05-2 2-Chloro-N6-cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist with Ki of 0.8 nM for human A1.
CSN22617 (±)-5'-Chloro-5'-deoxy-ENBA 103626-26-2 (±)-5'-Chloro-5'-deoxy-ENBA is a highly selective adenosine A1 receptor agonist with Ki of 0.51 nM.
CSN32734 KI-7 1489263-00-4
CSN106584 ST 1535 496955-42-1
CSN107412 PD 81723 132861-87-1
CSN51551 4-Nitrophenyl Phenylphosphonate 57072-35-2
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