400-920-2911 sales@csnpharm.cn
Adenosine Receptor
货号 | 产品名 | CAS号 | 信息 |
---|---|---|---|
CSN19381 | Xanthine | 69-89-6 | Xanthine is a natural occuring purine-base adenosine receptor antagonist, from which a number of stimulants such as caffeine and theobromine are derived. |
CSN24475 | XAC 3HCl | 1783977-95-6 | XAC is an adenosine receptor antagonist with IC50 value of 16μM for Adenosine Receptor A2. |
CSN21258 | Tecadenoson | 204512-90-3 | Tecadenoson is a selective A1 adenosine receptor agonist. |
CSN23108 | SCH 442416 | 316173-57-6 | SCH-442416 is a selective adenosine A2A receptor antagonist. SCH-442416 binds to human and rat A2A receptors with high affinity (Ki values are 0.048 and 0.5 nM respectively). It displays > 23000-fold selectivity for hA2A over hA1 in vitro with minimal affinity for hA2B and hA3 receptors (IC50 > 10 μM). |
CSN21946 | Proxyphylline | 603-00-9 | Proxyphylline is a xanthine-derivatived antagonists of A1 and A2 adenosine receptors, which relaxe smooth muscles, particularly bronchial muscles. |
CSN23113 | SDZ WAG 994 | 130714-47-5 | Potent, selective A1 agonist |
CSN21751 | NECA | 35920-39-9 | NECA, an analog of adenosine, is agonist of adenosine receptors with Kis of 1880, 6660, and 3.5 nM for A1, A2A, and A3, respectively. |
CSN22994 | N6-Cyclopentyladenosine | 41552-82-3 | N6-Cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist with Ki of 2.3 nM for human A1 receptor. |
CSN18631 | N-[(4-Aminophenyl)methyl]adenosine | 95523-13-0 | N-[(4-Aminophenyl)methyl]adenosine is an adenosine receptor inhibitor, with Ki of 29 nM for rat ecto-5′-nucleotidase. |
CSN25517 | N-(2-Hydroxyethyl)adenosine | 4338-48-1 | N-(2-Hydroxyethyl)adenosine has been studied as an anticonvulsant through the activation of adenosine A1 receptor (AA1R). It attenuates cell death induced by H2O2 through antioxidant action. |
CSN24570 | MRS 1220 | 183721-15-5 | MRS1220 is a potent and highly selective antagonist at the human A3 adenosine receptor. Ki values are 0.65, 305, and 52 nM at hA3, rA1 and rA2A respectively. MRS1220 displays an IC50 > 1 μM for inhibition of binding to rat A3 receptors. |
CSN22988 | MRS 1754 | 264622-58-4 | MRS 1754 is a selective adenosine A2B receptor antagonist with Ki of 1.97 nM for hA2B. |
CSN22987 | MRS 1706 | 264622-53-9 | MRS 1706 is a potent and selective adenosine A2B receptor inverse agonist with Ki of 1.39 nM. |
CSN22873 | KW 3902 | 136199-02-5 | KW 3902 is a Selective adenosine A1 receptor antagonist with Ki of 0.19 nM. |
CSN23107 | SCH 202676 Hydrobromide | 265980-25-4 | Inhibitor of ligand binding to G-protein-coupled receptors |
CSN22792 | DPCPX | 102146-07-6 | DPCPX is a potent and selective A1 adenosine receptor antagonist, both in vitro and in vivo, with Ki of 3.9 nM for human A1. |
CSN23120 | SLV 320 | 251945-92-3 | Derenofylline (SLV 320) is a potent, selective and orally active adenosine A1 receptor antagonist, with Ki values of 1 nM, 200 nM and 398 nM for human A1, A3 and A2A receptors respectively. Derenofylline suppresses cardiac fibrosis and attenuates albuminuria without affecting blood pressure in rats[1]. |
CSN18682 | CGS 21680 HCl | 124431-80-7 | CGS 21680 HCl is A2A adenosine receptor agonist with Ki value of 27 nM, which can be used to distinguish A2A- and A2B-mediated effect and shows affinity for both A1 and A3 adenosine receptors. |
CSN24568 | CGS 15943 | 104615-18-1 | CGS 15943 is a potent adenosine receptor antagonist with Ki values of 3.5, 4.2, 16 and 51 nM for human A1, A2A, A2B and A3 receptors respectively. |
CSN22708 | BAY 60-6583 | 910487-58-0 | BAY 60-6583 is a potent adenosine A2B receptor agonist with EC50 of 2.83 nM for murine A2B receptor. |
CSN21468 | Alloxazine | 490-59-5 | Alloxazine is a selective antagonist of A2B adenosine receptor. |
CSN23524 | Adenosine | 58-61-7 | Adenosine is a nucleoside that is composed of adenine and d-ribose and plays many important biological roles in addition to being components of DNA and RNA. |
CSN25244 | Adenosine amine congener | 96760-69-9 | Adenosine amine congener hydrate is a potent aqueous-soluble A1 adenosine receptor agonist with Ki value of 0.85nM for binding against [3H]N6-cyclohexyladenosine in rat cerebral cortex membranes. |
CSN24565 | 8-Cyclopentyl-1,3-dimethylxanthine | 35873-49-5 | 8-Cyclopentyl-1,3-dimethylxanthine is a selective antagonist of adenosine A1 receptor with pKi of 7.5-8. |
CSN24575 | 8-(3-Chlorostyryl)caffeine | 147700-11-6 | 8-(3-Chlorostyryl)caffeine is a selective adenosine A2A receptor antagonist (Ki = 54 nM at rat A2) and monoamine oxidase B (MAO-B) inhibitor (Ki = 100 nM). |
CSN22645 | 2-Chloro-N6-cyclopentyladenosine | 37739-05-2 | 2-Chloro-N6-cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist with Ki of 0.8 nM for human A1. |
CSN22617 | (±)-5'-Chloro-5'-deoxy-ENBA | 103626-26-2 | (±)-5'-Chloro-5'-deoxy-ENBA is a highly selective adenosine A1 receptor agonist with Ki of 0.51 nM. |
CSN32734 | KI-74 | 1489263-00-4 |