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Adenosine Receptor

Adenosine Receptor

货号 产品名 CAS号 信息
CSN24475 Xanthine amine congener hydrochloride 1783977-95-6 XAC is an adenosine receptor antagonist with IC50 value of 16μM for Adenosine Receptor A2.
CSN19829 Trabodenoson 871108-05-3 Trabodenoson is a potent and highly selective adenosine A1 receptor agonist.
CSN16416 Theophylline 58-55-9 Theophylline is a natural product present in tea and cocoa, working as a phosphodiesterase inhibitor, adenosine receptor blocker, and histone deacetylase activator.
CSN21258 Tecadenoson 204512-90-3 Tecadenoson is a selective A1 adenosine receptor agonist.
CSN27356 Taminadenant 1337962-47-6 Taminadenant is an antagonist of adenosine receptor.
CSN23108 SCH442416 316173-57-6 SCH-442416 is a selective adenosine A2A receptor antagonist. SCH-442416 binds to human and rat A2A receptors with high affinity (Ki values are 0.048 and 0.5 nM respectively). It displays > 23000-fold selectivity for hA2A over hA1 in vitro with minimal affinity for hA2B and hA3 receptors (IC50 > 10 μM).
CSN23057 PSB-603 1092351-10-4 PSB 603 is a adenosine A2B receptor antagonist with Ki of 0.553 nM.
CSN23056 PSB36 524944-72-7 PSB 36 is a potent and selective A1 adenosine receptor antagonist that displays binding affinity of 0.12 nM for rA1.
CSN23054 PSB-0788 1027513-54-7 PSB 0788 is a potent and selective adenosine A2B receptor antagonist with IC50 of 3.64 nM at human A2B receptor.
CSN21946 Proxyphylline 603-00-9 Proxyphylline is a xanthine-derivatived antagonists of A1 and A2 adenosine receptors, which relaxe smooth muscles, particularly bronchial muscles.
CSN23050 PQ-69 910045-32-8 PQ 69 is a potent and selective A1 receptor inverse agonist taht exhibits high binding affinity at A1 receptor with Kis of 0.07 and 0.96 nM for rat and human receptors respectively.
CSN23113 SDZ WAG 994 130714-47-5 Potent, selective A1 agonist
CSN23153 TC-G 1004 1061747-72-5 Potent and selective A2A antagonist
CSN20000 Neladenoson dalanate 1239309-58-0 Neladenoson dalanate is a potent and selective adenosine A1 receptor agonist, and potentially useful for treatment of cardiovascular diseases.
CSN21751 5'-N-Ethylcarboxamidoadenosine 35920-39-9 NECA, an analog of adenosine, is agonist of adenosine receptors with Kis of 1880, 6660, and 3.5 nM for A1, A2A, and A3, respectively.
CSN22994 N6-Cyclopentyladenosine 41552-82-3 N6-Cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist with Ki of 2.3 nM for human A1 receptor.
CSN25517 N-(2-Hydroxyethyl)adenosine 4338-48-1 N-(2-Hydroxyethyl)adenosine has been studied as an anticonvulsant through the activation of adenosine A1 receptor (AA1R). It attenuates cell death induced by H2O2 through antioxidant action.
CSN24570 MRS1220 183721-15-5 MRS1220 is a potent and highly selective antagonist at the human A3 adenosine receptor. Ki values are 0.65, 305, and 52 nM at hA3, rA1 and rA2A respectively. MRS1220 displays an IC50 > 1 μM for inhibition of binding to rat A3 receptors.
CSN22990 MRS5698 1377273-00-1 MRS 5698 is a high affinity and selective A3 adenosine receptor agonist with Ki ~ 3 nM.
CSN22989 MRS-3777 hemioxalate 1186195-57-2 MRS 3777 Hemioxalate is a high affinity adenosine A3 receptor antagonist with Ki of 47 nM.
CSN22988 MRS 1754 264622-58-4 MRS 1754 is a selective adenosine A2B receptor antagonist with Ki of 1.97 nM for hA2B.
CSN22987 MRS-1706 264622-53-9 MRS 1706 is a potent and selective adenosine A2B receptor inverse agonist with Ki of 1.39 nM.
CSN22873 Rolofylline 136199-02-5 KW 3902 is a Selective adenosine A1 receptor antagonist with Ki of 0.19 nM.
CSN22860 ISAM-140 932191-62-3 ISAM 140 is a high affinity A2B receptor antagonist with Ki of 3.49 nM.
CSN23107 SCH 202676 Hydrobromide 265980-25-4 Inhibitor of ligand binding to G-protein-coupled receptors
CSN22848 HEMADO 403842-38-6 HEMADO is a high affinity and selective adenosine A3 receptor agonist with Ki of 1.1 nM for human A3.
CSN22792 DPCPX 102146-07-6 DPCPX is a potent and selective A1 adenosine receptor antagonist, both in vitro and in vivo, with Ki of 3.9 nM for human A1.
CSN23120 Derenofylline 251945-92-3 Derenofylline (SLV 320) is a potent, selective and orally active adenosine A1 receptor antagonist, with Ki values of 1 nM, 200 nM and 398 nM for human A1, A3 and A2A receptors respectively. Derenofylline suppresses cardiac fibrosis and attenuates albuminuria without affecting blood pressure in rats[1].
CSN22838 GS-6201 752222-83-6 CVT-6883 is a selective antagonist of adenosine A2B receptors with Ki of 22 nM for human A2B.
CSN21199 Ciforadenant(CPI-444) 1202402-40-1 CPI-444 is an orally administered antagonist of the adenosine A2A receptor. Upon oral administration, CPI-444 binds to adenosine A2A receptors expressed on the surface of immune cells, including T-lymphocytes, natural killer (NK) cells, macrophages and dendritic cells (DCs).
CSN24568 CGS 15943 104615-18-1 CGS 15943 is a potent adenosine receptor antagonist with Ki values of 3.5, 4.2, 16 and 51 nM for human A1, A2A, A2B and A3 receptors respectively.
CSN23897 BAY-545 1699717-32-2 BAY-545 is a structure-optimizd adenosine receptor A2B antagonist with IC50 value of of 59 nM.
CSN24164 BAY-218 2162982-11-6 BAY-218 is an AHR antagonist.
CSN22708 BAY 60-6583 910487-58-0 BAY 60-6583 is a potent adenosine A2B receptor agonist with EC50 of 2.83 nM for murine A2B receptor.
CSN27286 BAY 2416964 2242464-44-2 BAY 2416964 is an antagonist of aryl hydrocarbon receptor (AhR) with IC50 of 341 nM.
CSN21201 Imaradenant (AZD4635) 1321514-06-0 AZD4635 is an A2AR antagonist which can reverse adenosine mediated T cell suppression.
CSN21468 Alloxazine 490-59-5 Alloxazine is a selective antagonist of A2B adenosine receptor.
CSN23524 Adenosine 58-61-7 Adenosine is a nucleoside that is composed of adenine and d-ribose and plays many important biological roles in addition to being components of DNA and RNA.
CSN21333 Adenosine antagonist-1 431040-19-6 Adenosine antagonist-1 is an adenosine A3 receptor (AA3R) antagonist.
CSN25244 Adenosine amine congener   96760-69-9 Adenosine amine congener hydrate is a potent aqueous-soluble A1 adenosine receptor agonist with Ki value of 0.85nM for binding against [3H]N6-cyclohexyladenosine in rat cerebral cortex membranes.
CSN24753 AB928   2239273-34-6 AB928 is a dual A2aR/A2bR antagonist that inhibits A2aR and A2bR with an equilibrium binding constant of 1.4 and 2 nM, respectively.
CSN18264 A2AR-agonist-1 41552-95-8 A2AR-agonist-1 is a potent A2AR and ENT1 agonist with Ki of 4.39 and 3.47 for A2AR and ENT1.
CSN24565 8-Cyclopentyl-1,3-dimethylxanthine 35873-49-5 8-Cyclopentyl-1,3-dimethylxanthine is a selective antagonist of adenosine A1 receptor with pKi of 7.5-8.
CSN24575 (E)-8-(3-Chlorostyryl)caffeine 147700-11-6 8-(3-Chlorostyryl)caffeine is a selective adenosine A2A receptor antagonist (Ki = 54 nM at rat A2) and monoamine oxidase B (MAO-B) inhibitor (Ki = 100 nM).
CSN22645 (2R,3R,4S,5R)-2-(2-Chloro-6-(cyclopentylamino)-9H-purin-9-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol 37739-05-2 2-Chloro-N6-cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist with Ki of 0.8 nM for human A1.
CSN22617 (±)-5'-Chloro-5'-deoxy-ENBA 103626-26-2 (±)-5'-Chloro-5'-deoxy-ENBA is a highly selective adenosine A1 receptor agonist with Ki of 0.51 nM.
CSN32734 KI-7 1489263-00-4
CSN106584 2-Butyl-9-methyl-8-(2H-1,2,3-triazol-2-yl)-9H-purin-6-amine 496955-42-1
CSN107412 (2-Amino-4,5-dimethylthiophen-3-yl)(3-(trifluoromethyl)phenyl)methanone 132861-87-1
CSN51551 4-Nitrophenyl hydrogen phenylphosphonate 57072-35-2
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