Adenosine Receptor

Adenosine Receptor
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货号	产品名	CAS号	信息
CSN19381	Xanthine	69-89-6	Xanthine is a natural occuring purine-base adenosine receptor antagonist, from which a number of stimulants such as caffeine and theobromine are derived.
CSN16416	Theophylline	58-55-9	Theophylline is a natural product present in tea and cocoa, working as a phosphodiesterase inhibitor, adenosine receptor blocker, and histone deacetylase activator.
CSN21258	Tecadenoson	204512-90-3	Tecadenoson is a selective A1 adenosine receptor agonist.
CSN23108	SCH 442416	316173-57-6	SCH-442416 is a selective adenosine A2A receptor antagonist. SCH-442416 binds to human and rat A2A receptors with high affinity (Ki values are 0.048 and 0.5 nM respectively). It displays > 23000-fold selectivity for hA2A over hA1 in vitro with minimal affinity for hA2B and hA3 receptors (IC50 > 10 μM).
CSN21946	Proxyphylline	603-00-9	Proxyphylline is a xanthine-derivatived antagonists of A1 and A2 adenosine receptors, which relaxe smooth muscles, particularly bronchial muscles.
CSN23113	SDZ WAG 994	130714-47-5	Potent, selective A1 agonist
CSN16615	Norisoboldine	23599-69-1	Norisoboldine is an isoquinoline alkaloid isolated and purfied from the roots of Lindera aggregata, which acts as an AhR agonist, and enhances the function of the adenosine A1 receptor.
CSN18541	N6-[2-(4-Aminophenyl)ethyl]adenosine	89705-21-5	N6-[2-(4-Aminophenyl)ethyl]adenosine is a potent, non-selective A3 adenosine receptor agonist.
CSN22994	N6-Cyclopentyladenosine	41552-82-3	N6-Cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist with Ki of 2.3 nM for human A1 receptor.
CSN18631	N-[(4-Aminophenyl)methyl]adenosine	95523-13-0	N-[(4-Aminophenyl)methyl]adenosine is an adenosine receptor inhibitor, with Ki of 29 nM for rat ecto-5′-nucleotidase.
CSN25517	N-(2-Hydroxyethyl)adenosine	4338-48-1	N-(2-Hydroxyethyl)adenosine has been studied as an anticonvulsant through the activation of adenosine A1 receptor (AA1R). It attenuates cell death induced by H2O2 through antioxidant action.
CSN22988	MRS 1754	264622-58-4	MRS 1754 is a selective adenosine A2B receptor antagonist with Ki of 1.97 nM for hA2B.
CSN22987	MRS 1706	264622-53-9	MRS 1706 is a potent and selective adenosine A2B receptor inverse agonist with Ki of 1.39 nM.
CSN22873	KW 3902	136199-02-5	KW 3902 is a Selective adenosine A1 receptor antagonist with Ki of 0.19 nM.
CSN23107	SCH 202676 Hydrobromide	265980-25-4	Inhibitor of ligand binding to G-protein-coupled receptors
CSN16958	IB-MECA	152918-18-8	IB-MECA is an agonist of the adenosine A3 receptor with EC50 values of 0.11 μM. IB-MECA is a potent and selective A3 adenosine receptor agonist with Ki value of 1.1, 54 and 56 nM for A3, A1 and A2A receptors, respectively, which possessing cardioprotective effect and reduces infarct size upon reperfusion in rats.
CSN17618	GR79236	124555-18-6	GR79236 is a highly potent and selective adenosine A1 receptor agonist (Ki = 3.1 nM) that has analgesic and anti-inflammatory actions in humans and animals.
CSN22792	DPCPX	102146-07-6	DPCPX is a potent and selective A1 adenosine receptor antagonist, both in vitro and in vivo, with Ki of 3.9 nM for human A1.
CSN23120	SLV 320	251945-92-3	Derenofylline (SLV 320) is a potent, selective and orally active adenosine A1 receptor antagonist, with Ki values of 1 nM, 200 nM and 398 nM for human A1, A3 and A2A receptors respectively. Derenofylline suppresses cardiac fibrosis and attenuates albuminuria without affecting blood pressure in rats[1].
CSN18682	CGS 21680 HCl	124431-80-7	CGS 21680 HCl is A2A adenosine receptor agonist with Ki value of 27 nM, which can be used to distinguish A2A- and A2B-mediated effect and shows affinity for both A1 and A3 adenosine receptors.
CSN22708	BAY 60-6583	910487-58-0	BAY 60-6583 is a potent adenosine A2B receptor agonist with EC50 of 2.83 nM for murine A2B receptor.
CSN21468	Alloxazine	490-59-5	Alloxazine is a selective antagonist of A2B adenosine receptor.
CSN23524	Adenosine	58-61-7	Adenosine is a nucleoside that is composed of adenine and d-ribose and plays many important biological roles in addition to being components of DNA and RNA.
CSN25244	Adenosine amine congener	96760-69-9	Adenosine amine congener hydrate is a potent aqueous-soluble A1 adenosine receptor agonist with Ki value of 0.85nM for binding against [3H]N6-cyclohexyladenosine in rat cerebral cortex membranes.
CSN17909	AB-MECA	152918-26-8	AB-MECA is a high affinity A3 adenosine receptor agonist, has high affinity for recombinant A1 and A3 receptors.
CSN17107	2-Cl-IB-MECA	163042-96-4	2-Cl-IB-MECA is a highly selective A3 adenosine receptor agonist with Ki value of 0.33nM, displaying 2500- and 1400-fold selectivity over A1 and A2A receptors, respectively.
CSN22645	2-Chloro-N6-cyclopentyladenosine	37739-05-2	2-Chloro-N6-cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist with Ki of 0.8 nM for human A1.
CSN22617	(±)-5'-Chloro-5'-deoxy-ENBA	103626-26-2	(±)-5'-Chloro-5'-deoxy-ENBA is a highly selective adenosine A1 receptor agonist with Ki of 0.51 nM.

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Adenosine Receptor
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