Adenosine Receptor

Adenosine Receptor
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货号	产品名	CAS号	信息
CSN19381	Xanthine	69-89-6	Xanthine is a natural occuring purine-base adenosine receptor antagonist, from which a number of stimulants such as caffeine and theobromine are derived.
CSN24475	XAC 3HCl	1783977-95-6	XAC is an adenosine receptor antagonist with IC50 value of 16μM for Adenosine Receptor A2.
CSN21258	Tecadenoson	204512-90-3	Tecadenoson is a selective A1 adenosine receptor agonist.
CSN23108	SCH 442416	316173-57-6	SCH-442416 is a selective adenosine A2A receptor antagonist. SCH-442416 binds to human and rat A2A receptors with high affinity (Ki values are 0.048 and 0.5 nM respectively). It displays > 23000-fold selectivity for hA2A over hA1 in vitro with minimal affinity for hA2B and hA3 receptors (IC50 > 10 μM).
CSN21946	Proxyphylline	603-00-9	Proxyphylline is a xanthine-derivatived antagonists of A1 and A2 adenosine receptors, which relaxe smooth muscles, particularly bronchial muscles.
CSN23113	SDZ WAG 994	130714-47-5	Potent, selective A1 agonist
CSN21751	NECA	35920-39-9	NECA, an analog of adenosine, is agonist of adenosine receptors with Kis of 1880, 6660, and 3.5 nM for A1, A2A, and A3, respectively.
CSN22994	N6-Cyclopentyladenosine	41552-82-3	N6-Cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist with Ki of 2.3 nM for human A1 receptor.
CSN18631	N-[(4-Aminophenyl)methyl]adenosine	95523-13-0	N-[(4-Aminophenyl)methyl]adenosine is an adenosine receptor inhibitor, with Ki of 29 nM for rat ecto-5′-nucleotidase.
CSN25517	N-(2-Hydroxyethyl)adenosine	4338-48-1	N-(2-Hydroxyethyl)adenosine has been studied as an anticonvulsant through the activation of adenosine A1 receptor (AA1R). It attenuates cell death induced by H2O2 through antioxidant action.
CSN24570	MRS 1220	183721-15-5	MRS1220 is a potent and highly selective antagonist at the human A3 adenosine receptor. Ki values are 0.65, 305, and 52 nM at hA3, rA1 and rA2A respectively. MRS1220 displays an IC50 > 1 μM for inhibition of binding to rat A3 receptors.
CSN22988	MRS 1754	264622-58-4	MRS 1754 is a selective adenosine A2B receptor antagonist with Ki of 1.97 nM for hA2B.
CSN22987	MRS 1706	264622-53-9	MRS 1706 is a potent and selective adenosine A2B receptor inverse agonist with Ki of 1.39 nM.
CSN22873	KW 3902	136199-02-5	KW 3902 is a Selective adenosine A1 receptor antagonist with Ki of 0.19 nM.
CSN23107	SCH 202676 Hydrobromide	265980-25-4	Inhibitor of ligand binding to G-protein-coupled receptors
CSN22792	DPCPX	102146-07-6	DPCPX is a potent and selective A1 adenosine receptor antagonist, both in vitro and in vivo, with Ki of 3.9 nM for human A1.
CSN23120	SLV 320	251945-92-3	Derenofylline (SLV 320) is a potent, selective and orally active adenosine A1 receptor antagonist, with Ki values of 1 nM, 200 nM and 398 nM for human A1, A3 and A2A receptors respectively. Derenofylline suppresses cardiac fibrosis and attenuates albuminuria without affecting blood pressure in rats[1].
CSN18682	CGS 21680 HCl	124431-80-7	CGS 21680 HCl is A2A adenosine receptor agonist with Ki value of 27 nM, which can be used to distinguish A2A- and A2B-mediated effect and shows affinity for both A1 and A3 adenosine receptors.
CSN24568	CGS 15943	104615-18-1	CGS 15943 is a potent adenosine receptor antagonist with Ki values of 3.5, 4.2, 16 and 51 nM for human A1, A2A, A2B and A3 receptors respectively.
CSN22708	BAY 60-6583	910487-58-0	BAY 60-6583 is a potent adenosine A2B receptor agonist with EC50 of 2.83 nM for murine A2B receptor.
CSN21468	Alloxazine	490-59-5	Alloxazine is a selective antagonist of A2B adenosine receptor.
CSN23524	Adenosine	58-61-7	Adenosine is a nucleoside that is composed of adenine and d-ribose and plays many important biological roles in addition to being components of DNA and RNA.
CSN25244	Adenosine amine congener	96760-69-9	Adenosine amine congener hydrate is a potent aqueous-soluble A1 adenosine receptor agonist with Ki value of 0.85nM for binding against [3H]N6-cyclohexyladenosine in rat cerebral cortex membranes.
CSN24565	8-Cyclopentyl-1,3-dimethylxanthine	35873-49-5	8-Cyclopentyl-1,3-dimethylxanthine is a selective antagonist of adenosine A1 receptor with pKi of 7.5-8.
CSN24575	8-(3-Chlorostyryl)caffeine	147700-11-6	8-(3-Chlorostyryl)caffeine is a selective adenosine A2A receptor antagonist (Ki = 54 nM at rat A2) and monoamine oxidase B (MAO-B) inhibitor (Ki = 100 nM).
CSN22645	2-Chloro-N6-cyclopentyladenosine	37739-05-2	2-Chloro-N6-cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist with Ki of 0.8 nM for human A1.
CSN22617	(±)-5'-Chloro-5'-deoxy-ENBA	103626-26-2	(±)-5'-Chloro-5'-deoxy-ENBA is a highly selective adenosine A1 receptor agonist with Ki of 0.51 nM.
CSN32734	KI-74	1489263-00-4

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Adenosine Receptor
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