Adenosine Receptor

Adenosine Receptor
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货号	产品名	CAS号	信息
CSN24475	Xanthine amine congener hydrochloride	1783977-95-6	XAC is an adenosine receptor antagonist with IC50 value of 16μM for Adenosine Receptor A2.
CSN19829	Trabodenoson	871108-05-3	Trabodenoson is a potent and highly selective adenosine A1 receptor agonist.
CSN16416	Theophylline	58-55-9	Theophylline is a natural product present in tea and cocoa, working as a phosphodiesterase inhibitor, adenosine receptor blocker, and histone deacetylase activator.
CSN21258	Tecadenoson	204512-90-3	Tecadenoson is a selective A1 adenosine receptor agonist.
CSN27356	Taminadenant	1337962-47-6	Taminadenant is an antagonist of adenosine receptor.
CSN23108	SCH442416	316173-57-6	SCH-442416 is a selective adenosine A2A receptor antagonist. SCH-442416 binds to human and rat A2A receptors with high affinity (Ki values are 0.048 and 0.5 nM respectively). It displays > 23000-fold selectivity for hA2A over hA1 in vitro with minimal affinity for hA2B and hA3 receptors (IC50 > 10 μM).
CSN23057	PSB-603	1092351-10-4	PSB 603 is a adenosine A2B receptor antagonist with Ki of 0.553 nM.
CSN23056	PSB36	524944-72-7	PSB 36 is a potent and selective A1 adenosine receptor antagonist that displays binding affinity of 0.12 nM for rA1.
CSN23054	PSB-0788	1027513-54-7	PSB 0788 is a potent and selective adenosine A2B receptor antagonist with IC50 of 3.64 nM at human A2B receptor.
CSN21946	Proxyphylline	603-00-9	Proxyphylline is a xanthine-derivatived antagonists of A1 and A2 adenosine receptors, which relaxe smooth muscles, particularly bronchial muscles.
CSN23050	PQ-69	910045-32-8	PQ 69 is a potent and selective A1 receptor inverse agonist taht exhibits high binding affinity at A1 receptor with Kis of 0.07 and 0.96 nM for rat and human receptors respectively.
CSN23113	SDZ WAG 994	130714-47-5	Potent, selective A1 agonist
CSN23153	TC-G 1004	1061747-72-5	Potent and selective A2A antagonist
CSN20000	Neladenoson dalanate	1239309-58-0	Neladenoson dalanate is a potent and selective adenosine A1 receptor agonist, and potentially useful for treatment of cardiovascular diseases.
CSN21751	5'-N-Ethylcarboxamidoadenosine	35920-39-9	NECA, an analog of adenosine, is agonist of adenosine receptors with Kis of 1880, 6660, and 3.5 nM for A1, A2A, and A3, respectively.
CSN22994	N6-Cyclopentyladenosine	41552-82-3	N6-Cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist with Ki of 2.3 nM for human A1 receptor.
CSN25517	N-(2-Hydroxyethyl)adenosine	4338-48-1	N-(2-Hydroxyethyl)adenosine has been studied as an anticonvulsant through the activation of adenosine A1 receptor (AA1R). It attenuates cell death induced by H2O2 through antioxidant action.
CSN24570	MRS1220	183721-15-5	MRS1220 is a potent and highly selective antagonist at the human A3 adenosine receptor. Ki values are 0.65, 305, and 52 nM at hA3, rA1 and rA2A respectively. MRS1220 displays an IC50 > 1 μM for inhibition of binding to rat A3 receptors.
CSN22990	MRS5698	1377273-00-1	MRS 5698 is a high affinity and selective A3 adenosine receptor agonist with Ki ~ 3 nM.
CSN22989	MRS-3777 hemioxalate	1186195-57-2	MRS 3777 Hemioxalate is a high affinity adenosine A3 receptor antagonist with Ki of 47 nM.
CSN22988	MRS 1754	264622-58-4	MRS 1754 is a selective adenosine A2B receptor antagonist with Ki of 1.97 nM for hA2B.
CSN22987	MRS-1706	264622-53-9	MRS 1706 is a potent and selective adenosine A2B receptor inverse agonist with Ki of 1.39 nM.
CSN22873	Rolofylline	136199-02-5	KW 3902 is a Selective adenosine A1 receptor antagonist with Ki of 0.19 nM.
CSN22860	ISAM-140	932191-62-3	ISAM 140 is a high affinity A2B receptor antagonist with Ki of 3.49 nM.
CSN23107	SCH 202676 Hydrobromide	265980-25-4	Inhibitor of ligand binding to G-protein-coupled receptors
CSN22848	HEMADO	403842-38-6	HEMADO is a high affinity and selective adenosine A3 receptor agonist with Ki of 1.1 nM for human A3.
CSN22792	DPCPX	102146-07-6	DPCPX is a potent and selective A1 adenosine receptor antagonist, both in vitro and in vivo, with Ki of 3.9 nM for human A1.
CSN23120	Derenofylline	251945-92-3	Derenofylline (SLV 320) is a potent, selective and orally active adenosine A1 receptor antagonist, with Ki values of 1 nM, 200 nM and 398 nM for human A1, A3 and A2A receptors respectively. Derenofylline suppresses cardiac fibrosis and attenuates albuminuria without affecting blood pressure in rats[1].
CSN22838	GS-6201	752222-83-6	CVT-6883 is a selective antagonist of adenosine A2B receptors with Ki of 22 nM for human A2B.
CSN21199	Ciforadenant(CPI-444)	1202402-40-1	CPI-444 is an orally administered antagonist of the adenosine A2A receptor. Upon oral administration, CPI-444 binds to adenosine A2A receptors expressed on the surface of immune cells, including T-lymphocytes, natural killer (NK) cells, macrophages and dendritic cells (DCs).
CSN24568	CGS 15943	104615-18-1	CGS 15943 is a potent adenosine receptor antagonist with Ki values of 3.5, 4.2, 16 and 51 nM for human A1, A2A, A2B and A3 receptors respectively.
CSN23897	BAY-545	1699717-32-2	BAY-545 is a structure-optimizd adenosine receptor A2B antagonist with IC50 value of of 59 nM.
CSN24164	BAY-218	2162982-11-6	BAY-218 is an AHR antagonist.
CSN22708	BAY 60-6583	910487-58-0	BAY 60-6583 is a potent adenosine A2B receptor agonist with EC50 of 2.83 nM for murine A2B receptor.
CSN27286	BAY 2416964	2242464-44-2	BAY 2416964 is an antagonist of aryl hydrocarbon receptor (AhR) with IC50 of 341 nM.
CSN21201	Imaradenant (AZD4635)	1321514-06-0	AZD4635 is an A2AR antagonist which can reverse adenosine mediated T cell suppression.
CSN21468	Alloxazine	490-59-5	Alloxazine is a selective antagonist of A2B adenosine receptor.
CSN23524	Adenosine	58-61-7	Adenosine is a nucleoside that is composed of adenine and d-ribose and plays many important biological roles in addition to being components of DNA and RNA.
CSN21333	Adenosine antagonist-1	431040-19-6	Adenosine antagonist-1 is an adenosine A3 receptor (AA3R) antagonist.
CSN25244	Adenosine amine congener	96760-69-9	Adenosine amine congener hydrate is a potent aqueous-soluble A1 adenosine receptor agonist with Ki value of 0.85nM for binding against [3H]N6-cyclohexyladenosine in rat cerebral cortex membranes.
CSN24753	AB928	2239273-34-6	AB928 is a dual A2aR/A2bR antagonist that inhibits A2aR and A2bR with an equilibrium binding constant of 1.4 and 2 nM, respectively.
CSN18264	A2AR-agonist-1	41552-95-8	A2AR-agonist-1 is a potent A2AR and ENT1 agonist with Ki of 4.39 and 3.47 for A2AR and ENT1.
CSN24565	8-Cyclopentyl-1,3-dimethylxanthine	35873-49-5	8-Cyclopentyl-1,3-dimethylxanthine is a selective antagonist of adenosine A1 receptor with pKi of 7.5-8.
CSN24575	(E)-8-(3-Chlorostyryl)caffeine	147700-11-6	8-(3-Chlorostyryl)caffeine is a selective adenosine A2A receptor antagonist (Ki = 54 nM at rat A2) and monoamine oxidase B (MAO-B) inhibitor (Ki = 100 nM).
CSN22645	(2R,3R,4S,5R)-2-(2-Chloro-6-(cyclopentylamino)-9H-purin-9-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol	37739-05-2	2-Chloro-N6-cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist with Ki of 0.8 nM for human A1.
CSN22617	(±)-5'-Chloro-5'-deoxy-ENBA	103626-26-2	(±)-5'-Chloro-5'-deoxy-ENBA is a highly selective adenosine A1 receptor agonist with Ki of 0.51 nM.
CSN32734	KI-7	1489263-00-4
CSN106584	2-Butyl-9-methyl-8-(2H-1,2,3-triazol-2-yl)-9H-purin-6-amine	496955-42-1
CSN107412	(2-Amino-4,5-dimethylthiophen-3-yl)(3-(trifluoromethyl)phenyl)methanone	132861-87-1
CSN51551	4-Nitrophenyl hydrogen phenylphosphonate	57072-35-2

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Adenosine Receptor
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