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Adenosine Receptor
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN19381 | Xanthine | 69-89-6 | Xanthine is a natural occuring purine-base adenosine receptor antagonist, from which a number of stimulants such as caffeine and theobromine are derived. |
| CSN16416 | Theophylline | 58-55-9 | Theophylline is a natural product present in tea and cocoa, working as a phosphodiesterase inhibitor, adenosine receptor blocker, and histone deacetylase activator. |
| CSN21258 | Tecadenoson | 204512-90-3 | Tecadenoson is a selective A1 adenosine receptor agonist. |
| CSN23108 | SCH 442416 | 316173-57-6 | SCH-442416 is a selective adenosine A2A receptor antagonist. SCH-442416 binds to human and rat A2A receptors with high affinity (Ki values are 0.048 and 0.5 nM respectively). It displays > 23000-fold selectivity for hA2A over hA1 in vitro with minimal affinity for hA2B and hA3 receptors (IC50 > 10 μM). |
| CSN21946 | Proxyphylline | 603-00-9 | Proxyphylline is a xanthine-derivatived antagonists of A1 and A2 adenosine receptors, which relaxe smooth muscles, particularly bronchial muscles. |
| CSN16615 | Norisoboldine | 23599-69-1 | Norisoboldine is an isoquinoline alkaloid isolated and purfied from the roots of Lindera aggregata, which acts as an AhR agonist, and enhances the function of the adenosine A1 receptor. |
| CSN18541 | N6-[2-(4-Aminophenyl)ethyl]adenosine | 89705-21-5 | N6-[2-(4-Aminophenyl)ethyl]adenosine is a potent, non-selective A3 adenosine receptor agonist. |
| CSN22994 | N6-Cyclopentyladenosine | 41552-82-3 | N6-Cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist with Ki of 2.3 nM for human A1 receptor. |
| CSN18631 | N-[(4-Aminophenyl)methyl]adenosine | 95523-13-0 | N-[(4-Aminophenyl)methyl]adenosine is an adenosine receptor inhibitor, with Ki of 29 nM for rat ecto-5′-nucleotidase. |
| CSN25517 | N-(2-Hydroxyethyl)adenosine | 4338-48-1 | N-(2-Hydroxyethyl)adenosine has been studied as an anticonvulsant through the activation of adenosine A1 receptor (AA1R). It attenuates cell death induced by H2O2 through antioxidant action. |
| CSN22988 | MRS 1754 | 264622-58-4 | MRS 1754 is a selective adenosine A2B receptor antagonist with Ki of 1.97 nM for hA2B. |
| CSN22987 | MRS 1706 | 264622-53-9 | MRS 1706 is a potent and selective adenosine A2B receptor inverse agonist with Ki of 1.39 nM. |
| CSN22873 | KW 3902 | 136199-02-5 | KW 3902 is a Selective adenosine A1 receptor antagonist with Ki of 0.19 nM. |
| CSN16958 | IB-MECA | 152918-18-8 | IB-MECA is an agonist of the adenosine A3 receptor with EC50 values of 0.11 μM. IB-MECA is a potent and selective A3 adenosine receptor agonist with Ki value of 1.1, 54 and 56 nM for A3, A1 and A2A receptors, respectively, which possessing cardioprotective effect and reduces infarct size upon reperfusion in rats. |
| CSN17618 | GR79236 | 124555-18-6 | GR79236 is a highly potent and selective adenosine A1 receptor agonist (Ki = 3.1 nM) that has analgesic and anti-inflammatory actions in humans and animals. |
| CSN23120 | SLV 320 | 251945-92-3 | Derenofylline (SLV 320) is a potent, selective and orally active adenosine A1 receptor antagonist, with Ki values of 1 nM, 200 nM and 398 nM for human A1, A3 and A2A receptors respectively. Derenofylline suppresses cardiac fibrosis and attenuates albuminuria without affecting blood pressure in rats[1]. |
| CSN18682 | CGS 21680 HCl | 124431-80-7 | CGS 21680 HCl is A2A adenosine receptor agonist with Ki value of 27 nM, which can be used to distinguish A2A- and A2B-mediated effect and shows affinity for both A1 and A3 adenosine receptors. |
| CSN22708 | BAY 60-6583 | 910487-58-0 | BAY 60-6583 is a potent adenosine A2B receptor agonist with EC50 of 2.83 nM for murine A2B receptor. |
| CSN21468 | Alloxazine | 490-59-5 | Alloxazine is a selective antagonist of A2B adenosine receptor. |
| CSN23524 | Adenosine | 58-61-7 | Adenosine is a nucleoside that is composed of adenine and d-ribose and plays many important biological roles in addition to being components of DNA and RNA. |
| CSN25244 | Adenosine amine congener | 96760-69-9 | Adenosine amine congener hydrate is a potent aqueous-soluble A1 adenosine receptor agonist with Ki value of 0.85nM for binding against [3H]N6-cyclohexyladenosine in rat cerebral cortex membranes. |
| CSN17107 | 2-Cl-IB-MECA | 163042-96-4 | 2-Cl-IB-MECA is a highly selective A3 adenosine receptor agonist with Ki value of 0.33nM, displaying 2500- and 1400-fold selectivity over A1 and A2A receptors, respectively. |
| CSN22645 | 2-Chloro-N6-cyclopentyladenosine | 37739-05-2 | 2-Chloro-N6-cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist with Ki of 0.8 nM for human A1. |