Adenosine Receptor

Adenosine Receptor
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货号	产品名	CAS号	信息
CSN24475	Xanthine amine congener hydrochloride	1783977-95-6	XAC is an adenosine receptor antagonist with IC50 value of 16μM for Adenosine Receptor A2.
CSN19829	Trabodenoson	871108-05-3	Trabodenoson is a potent and highly selective adenosine A1 receptor agonist.
CSN16416	Theophylline	58-55-9	Theophylline is a natural product present in tea and cocoa, working as a phosphodiesterase inhibitor, adenosine receptor blocker, and histone deacetylase activator.
CSN21258	Tecadenoson	204512-90-3	Tecadenoson is a selective A1 adenosine receptor agonist.
CSN27356	Taminadenant	1337962-47-6	Taminadenant is an antagonist of adenosine receptor.
CSN23108	SCH442416	316173-57-6	SCH-442416 is a selective adenosine A2A receptor antagonist. SCH-442416 binds to human and rat A2A receptors with high affinity (Ki values are 0.048 and 0.5 nM respectively). It displays > 23000-fold selectivity for hA2A over hA1 in vitro with minimal affinity for hA2B and hA3 receptors (IC50 > 10 μM).
CSN23057	PSB-603	1092351-10-4	PSB 603 is a adenosine A2B receptor antagonist with Ki of 0.553 nM.
CSN23056	PSB36	524944-72-7	PSB 36 is a potent and selective A1 adenosine receptor antagonist that displays binding affinity of 0.12 nM for rA1.
CSN23054	PSB-0788	1027513-54-7	PSB 0788 is a potent and selective adenosine A2B receptor antagonist with IC50 of 3.64 nM at human A2B receptor.
CSN21946	Proxyphylline	603-00-9	Proxyphylline is a xanthine-derivatived antagonists of A1 and A2 adenosine receptors, which relaxe smooth muscles, particularly bronchial muscles.
CSN23050	PQ-69	910045-32-8	PQ 69 is a potent and selective A1 receptor inverse agonist taht exhibits high binding affinity at A1 receptor with Kis of 0.07 and 0.96 nM for rat and human receptors respectively.
CSN23113	(2R,3R,4R,5R)-5-(6-(Cyclohexylamino)-9H-purin-9-yl)-2-(hydroxymethyl)-4-methoxytetrahydrofuran-3-ol	130714-47-5	Potent, selective A1 agonist
CSN23153	TC-G 1004	1061747-72-5	Potent and selective A2A antagonist
CSN20000	Neladenoson dalanate	1239309-58-0	Neladenoson dalanate is a potent and selective adenosine A1 receptor agonist, and potentially useful for treatment of cardiovascular diseases.
CSN21751	5'-N-Ethylcarboxamidoadenosine	35920-39-9	NECA, an analog of adenosine, is agonist of adenosine receptors with Kis of 1880, 6660, and 3.5 nM for A1, A2A, and A3, respectively.
CSN22994	N6-Cyclopentyladenosine	41552-82-3	N6-Cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist with Ki of 2.3 nM for human A1 receptor.
CSN25517	N-(2-Hydroxyethyl)adenosine	4338-48-1	N-(2-Hydroxyethyl)adenosine has been studied as an anticonvulsant through the activation of adenosine A1 receptor (AA1R). It attenuates cell death induced by H2O2 through antioxidant action.
CSN24570	MRS1220	183721-15-5	MRS1220 is a potent and highly selective antagonist at the human A3 adenosine receptor. Ki values are 0.65, 305, and 52 nM at hA3, rA1 and rA2A respectively. MRS1220 displays an IC50 > 1 μM for inhibition of binding to rat A3 receptors.
CSN22990	MRS5698	1377273-00-1	MRS 5698 is a high affinity and selective A3 adenosine receptor agonist with Ki ~ 3 nM.
CSN22989	MRS-3777 hemioxalate	1186195-57-2	MRS 3777 Hemioxalate is a high affinity adenosine A3 receptor antagonist with Ki of 47 nM.
CSN22988	MRS 1754	264622-58-4	MRS 1754 is a selective adenosine A2B receptor antagonist with Ki of 1.97 nM for hA2B.
CSN22987	MRS-1706	264622-53-9	MRS 1706 is a potent and selective adenosine A2B receptor inverse agonist with Ki of 1.39 nM.
CSN22873	Rolofylline	136199-02-5	KW 3902 is a Selective adenosine A1 receptor antagonist with Ki of 0.19 nM.
CSN22860	ISAM-140	932191-62-3	ISAM 140 is a high affinity A2B receptor antagonist with Ki of 3.49 nM.
CSN23107	SCH 202676 Hydrobromide	265980-25-4	Inhibitor of ligand binding to G-protein-coupled receptors
CSN22848	HEMADO	403842-38-6	HEMADO is a high affinity and selective adenosine A3 receptor agonist with Ki of 1.1 nM for human A3.
CSN22792	DPCPX	102146-07-6	DPCPX is a potent and selective A1 adenosine receptor antagonist, both in vitro and in vivo, with Ki of 3.9 nM for human A1.
CSN23120	Derenofylline	251945-92-3	Derenofylline (SLV 320) is a potent, selective and orally active adenosine A1 receptor antagonist, with Ki values of 1 nM, 200 nM and 398 nM for human A1, A3 and A2A receptors respectively. Derenofylline suppresses cardiac fibrosis and attenuates albuminuria without affecting blood pressure in rats[1].
CSN22838	GS-6201	752222-83-6	CVT-6883 is a selective antagonist of adenosine A2B receptors with Ki of 22 nM for human A2B.
CSN21199	Ciforadenant(CPI-444)	1202402-40-1	CPI-444 is an orally administered antagonist of the adenosine A2A receptor. Upon oral administration, CPI-444 binds to adenosine A2A receptors expressed on the surface of immune cells, including T-lymphocytes, natural killer (NK) cells, macrophages and dendritic cells (DCs).
CSN24568	CGS 15943	104615-18-1	CGS 15943 is a potent adenosine receptor antagonist with Ki values of 3.5, 4.2, 16 and 51 nM for human A1, A2A, A2B and A3 receptors respectively.
CSN23897	BAY-545	1699717-32-2	BAY-545 is a structure-optimizd adenosine receptor A2B antagonist with IC50 value of of 59 nM.
CSN24164	BAY-218	2162982-11-6	BAY-218 is an AHR antagonist.
CSN22708	BAY 60-6583	910487-58-0	BAY 60-6583 is a potent adenosine A2B receptor agonist with EC50 of 2.83 nM for murine A2B receptor.
CSN27286	BAY 2416964	2242464-44-2	BAY 2416964 is an antagonist of aryl hydrocarbon receptor (AhR) with IC50 of 341 nM.
CSN21201	Imaradenant (AZD4635)	1321514-06-0	AZD4635 is an A2AR antagonist which can reverse adenosine mediated T cell suppression.
CSN21468	Alloxazine	490-59-5	Alloxazine is a selective antagonist of A2B adenosine receptor.
CSN23524	Adenosine	58-61-7	Adenosine is a nucleoside that is composed of adenine and d-ribose and plays many important biological roles in addition to being components of DNA and RNA.
CSN21333	Adenosine antagonist-1	431040-19-6	Adenosine antagonist-1 is an adenosine A3 receptor (AA3R) antagonist.
CSN25244	Adenosine amine congener	96760-69-9	Adenosine amine congener hydrate is a potent aqueous-soluble A1 adenosine receptor agonist with Ki value of 0.85nM for binding against [3H]N6-cyclohexyladenosine in rat cerebral cortex membranes.
CSN24753	AB928	2239273-34-6	AB928 is a dual A2aR/A2bR antagonist that inhibits A2aR and A2bR with an equilibrium binding constant of 1.4 and 2 nM, respectively.
CSN18264	A2AR-agonist-1	41552-95-8	A2AR-agonist-1 is a potent A2AR and ENT1 agonist with Ki of 4.39 and 3.47 for A2AR and ENT1.
CSN24565	8-Cyclopentyl-1,3-dimethylxanthine	35873-49-5	8-Cyclopentyl-1,3-dimethylxanthine is a selective antagonist of adenosine A1 receptor with pKi of 7.5-8.
CSN24575	(E)-8-(3-Chlorostyryl)caffeine	147700-11-6	8-(3-Chlorostyryl)caffeine is a selective adenosine A2A receptor antagonist (Ki = 54 nM at rat A2) and monoamine oxidase B (MAO-B) inhibitor (Ki = 100 nM).
CSN22645	(2R,3R,4S,5R)-2-(2-Chloro-6-(cyclopentylamino)-9H-purin-9-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol	37739-05-2	2-Chloro-N6-cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist with Ki of 0.8 nM for human A1.
CSN22617	(±)-5'-Chloro-5'-deoxy-ENBA	103626-26-2	(±)-5'-Chloro-5'-deoxy-ENBA is a highly selective adenosine A1 receptor agonist with Ki of 0.51 nM.
CSN32734	KI-7	1489263-00-4
CSN106584	2-Butyl-9-methyl-8-(2H-1,2,3-triazol-2-yl)-9H-purin-6-amine	496955-42-1
CSN107412	(2-Amino-4,5-dimethylthiophen-3-yl)(3-(trifluoromethyl)phenyl)methanone	132861-87-1
CSN51551	4-Nitrophenyl hydrogen phenylphosphonate	57072-35-2

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Adenosine Receptor
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