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Adrenergic Receptor

Adrenergic Receptor

货号 产品名 CAS号 信息
CSN24589 Zinterol 37000-20-7 Zinterol Hydrochloride is a selective agonist of β2-adrenoceptor with pKB values are 8.3 and < 5.7 for β2 and β1 receptors respectively in human artery.
CSN24046 Xamoterol 81801-12-9 Xamoterol hemifumarate is a selective partial agonist of β1-adrenoceptor.
CSN24598 WB 4101 HCl 2170-58-3 WB 4101 hydrochloride is a selective antagonist of α1A-adrenergic receptor.
CSN21863 Tiodazosin 66969-81-1 Tiodazosin is a potent competitive postsynaptic alpha adrenergic receptor antagonist.
CSN21856 Tertatolol 83688-84-0 Tertatolol is a potent antagonist of beta-adrenoceptor and 5-HT receptor, with unique renal vasodilatatory effects.
CSN24706 Tampramine fumarate 83166-18-1 Tampramine is a tricyclic antidepressant (TCA). It acts as a selective norepinephrine reuptake inhibitor and has negligible affinity for adrenergic, histaminergic, and muscarinic receptors.
CSN24608 Talsupram HCl 25487-28-9 Talsupram hydrochloride is a selective noradrenalin re-uptake inhibitor.
CSN24592 AMibegron hydrochloride 121524-09-2 SR 58611A hydrochloride is a selective β3-adrenergic receptor agonist with anxiolytic and antidepressant effects in rodent models.
CSN24600 SNAP 5089 HCl 157066-77-8 SNAP 5089 is a selective antagonist of α1A-adrenoceptor.
CSN24736 SNAP 5089 157066-76-7 SNAP 5089 is a selective antagonist of the subtype α1A-adrenoceptor. It binds with high affinity to α1A-adrenoceptor with a Ki value of 0.35 nM.
CSN11918 Sertindole 106516-24-9 Sertindole, a neuroleptic, is one of the antipsychotic medications available, with a high affinity for dopamine D2, serotonin 5-HT2A, 5-HT2C, and α1-adrenergic receptors.
CSN24586 RX 821002 HCl 109544-45-8 RX 821002 hydrochloride is a selective antagonist of α2-adrenoceptor with low affinity for imidazoline sites. The pKd values for α2D and α2A subtypes are 9.7 and 8.2 respectively.
CSN24576 RS 17053 HCl 169505-93-5 RS 17053 hydrochloride is a selective antagonist of α1A-adrenoceptor with pKi and pA2 estimate of 9.1 - 9.9.
CSN24604 Pronethalol HCl 51-02-5 Pronethalol hydrochloride is an antagonist of β-adrenergic antagonist for the treatment of angina pectoris and some arrhythmias.
CSN21781 Pamatolol 59110-35-9 Pamatolol is a selective cardioselective antagonist of beta adrenergic receptor without sympathomimetic activity.
CSN24584 JP 1302 2HCl 1259314-65-2 JP 1302 dihydrochloride is an antagonist of α2C-adrenoceptor with Ki value of 28 nM.
CSN21958 Indanazoline 40507-78-6 Indanazoline is a sympathomimetic imidazoline derivative and shows vasoconstrictive action .
CSN24602 Imiloxan HCl 81167-22-8 Imiloxan hydrochloride is a highly selective antagonist of α2-adrenoceptor.
CSN22034 GP2-114 130783-39-0 GP2-114 is an activator of adrenergic receptor β, and produces current-dependent cardiovascular action when administered by transdermal iontophoresis.
CSN26499 Fiduxosin free base 208993-54-8 Fiduxosin is an alpha(1)-adrenoceptor antagonist with higher affinity for alpha(1A)-adrenoceptors and for alpha(1D)-adrenoceptors than for alpha(1B)-adrenoceptors.
CSN33116 Esreboxetine 98819-76-2 Esreboxetine is a selective norepinephrine reuptake inhibitor.
CSN24610 Efaroxan HCl 89197-00-2 Efaroxan hydrochloride is an antagonist of α2 adrenoceptor and imidazoline I1 receptor ligand. The pKi values are 7.87, 7.42, 5.74, 7.28 and < 5 for α2A, α2B, α2C, I1 and I2 receptors, respectively.
CSN26575 Detomidine carboxylic acid 115664-39-6 Detomidine carboxylic acid is the major urinary metabolite of Detomidine. Detomidine is a synthetic α2-adrenergic agonist and an animal analgesic sedative. Detomidine also has cardiac and respiratory effects and an antidiuretic action[1][2].
CSN26579 Dabuzalgron 219311-44-1 Dabuzalgron (previously codenamed R-450; Ro-115-1240) is a novel partial alphaA/IL receptor agonist that is administered in its hydrochloride form to control urethral smooth muscle contraction. The hemodynamic changes in the drug are very small and it is a potential drug for the treatment of stress urinary incontinence.
CSN26578 Clonidine(200mg) 4205-90-7 Clonidine (also known as Catapres, Kapvay, Nexiclon, and Clophelin) is a sympathomimetic medication used to treat high blood pressure, attention deficit hyperactivity disorder, anxiety disorders, withdrawal (from either alcohol, opioids, or smoking), migraine, menopausal flushing, diarrhea, and certain pain conditions. It is classified as a centrally acting α2 adrenergic agonist and imidazoline receptor agonist that has been in clinical use for over 40 years.
CSN24596 Cirazoline HCl 40600-13-3 Cirazoline hydrochloride is a selective agonist of alpha1-adrenoceptor.
CSN33167 Bucindolol 71119-11-4 Bucindolol is a high-affinity, competitive beta blocker.
CSN24601 B-HT 933 2HCl 36067-72-8 B-HT 933 dihydrochloride is selective agonist of α2-adrenoceptor.
CSN24583 ARC 239 2HCl 55974-42-0 ARC 239 dihydrochloride is a selective antagonist of α2B adrenoceptor with pKD values of 8.8, 6.7 and 6.4 for α2B, α2A, and α2D receptors respectively.
CSN26577 Arbutamine 128470-16-6 Arbutamine is a cardiac stimulant. It stimulates adrenergic receptors. Arbutamine is a synthetic catecholamine with positive chronotropic and inotropic properties, used in echocardiography and diagnostic coronary angiography. Arbutamine binds to and activates beta-1 adrenergic receptors in the myocardium, thereby increasing heart rate and increasing force of myocardial contraction. Arbutamine, administered through a closed-loop, computer-controlled drug-delivery system, is indicated to elicit acute cardiovascular responses, similar to those produced by exercise, in order to aid in diagnosing the presence or absence of coronary artery disease in patients who cannot exercise adequately.
CSN32920 Ampreloxetine 1227056-84-9 Ampreloxetine is a norepinephrine reuptake inhibitor.
CSN32921 Ampreloxetine HCl 1227056-87-2 Ampreloxetine is a norepinephrine reuptake inhibitor.
CSN24599 A 61603 hydrobromide 107756-30-9 A 61603 hydrobromide is a selective α1A-adrenergic receptor agonist.
CSN24609 3-MPPI 133399-65-2 3-MPPI is a very potent ligand for α1 sites and regulates smooth muscle contraction. The pKi values for α1B, α1D, α1A adrenoceptors are 8.74, 9.44, 9.57 respectively. It also binds to 5-HT1A sites (Ki = 50 nM).
CSN24595 2-PMDQ 139047-55-5 2-PMDQ is a selective α1-adrenoceptor antagonist with antihypertensive effect.
CSN24597 2-MPMDQ 149847-77-8 2-MPMDQ is a selective antagonist of α1-AR adrenoceptor and can act as a hypotensive.
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