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Adrenergic Receptor
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN18767 | Tolazoline HCl | 59-97-2 | Tolazoline HCl is a competitive non-selective α-adrenergic receptor antagonist, used as a a vasodilator directly acting on blood vessels and also increasing cardiac output. |
| CSN12086 | Tiamenidine | 31428-61-2 | Thioridazine is an antipsychotic drug, used in the treatment of schizophrenia and psychosis, shows D4 selectivity or serotonin antagonism. |
| CSN19307 | Tetrahydrozoline HCl | 522-48-5 | Tetrahydrozoline HCl is an imidazole-derived alpha-adrenergic receptor agonist which can result vasoconstriction and decreased nasal and ophthalmic congestion. |
| CSN25553 | SR59230A | 174689-39-5 | SR59230A is a potent and selective Adrenergic Receptor β3 antagonist with IC50 values of 40, 408, and 648nM for Adrenergic Receptor β3, β1 and β2, respectively. It shows blood-brain barrier penetrability. |
| CSN18749 | Piribedil | 3605-01-4 | Piribedil is an antiparkinsonian agent and piperazine derivative which acts as a D2 and D3 receptor agonist. |
| CSN18661 | Naphazoline | 835-31-4 | Naphazoline is the common name for 2-(1-naphthylmethyl)-2-imidazoline HCl, it is a sympathomimetic agent with marked alpha adrenergic activity. |
| CSN23830 | Lofexidine | 31036-80-3 | Lofexidine is a selective α2-receptor agonist, commonly used to alleviate the physical symptoms of heroin and other types of opioid withdrawal[1][2]. |
| CSN18745 | Lofexidine HCl | 21498-08-8 | Lofexidine HCl is an α2A-adrenergic receptor agonist, commonly used to alleviate the physical symptoms of heroin and other types of opioid withdrawal. |
| CSN21997 | Labetalone HCl | 96441-14-4 | Labetalone hydrochloride is hydrochloride form of labetalone, a blocker of both alpha- and beta-adrenergic receptors that is used as an antihypertensive. |
| CSN22444 | L-765314 | 189349-50-6 | L-765314 is a potent and selective α1b adrenergic receptor antagonist with Kis of 5.4±0.6 nM and 2.0±0.66 nM for rat and human α1b adrenergic receptor, respectively. |
| CSN18526 | L-(-)-α-Methyldopa HCl | 884-39-9 | L-(-)-α-Methyldopa HCl is an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive drug used as a sympatholytic or antihypertensive. |
| CSN19723 | Isoxsuprine HCl | 579-56-6 | Isoxsuprine is a modulator of β2 adrenoreceptor and has agonist or antagonist effects. |
| CSN19742 | Idazoxan HCl | 79944-56-2 | Idazoxan is an alpha2-adrenoceptor antagonist potentially for the treatment of schizophrenia. |
| CSN20255 | ICI-118551 | 72795-19-8 | ICI-118551 is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors, respectively. |
| CSN23785 | GUANABENZ | 5051-62-7 | Guanabenz is an agonist of α2-adrenergic receptor with antihypertensive effect and is enerally used in combination with diuretics. |
| CSN19298 | Fenspiride HCl | 5053-08-7 | Fenspiride HCl is an antagonist of α-adrenergic receptors and H1 histamine receptors and also inhibits phosphodiesterase 4 and phosphodiesterase 3 activities with logIC50 values of 4.16 and 3.44, respectively. |
| CSN19404 | Detomidine | 76631-46-4 | Detomidine produce dose-dependent sedative and analgesic effects, is a nonnarcotic, synthetic α2-adrenergic agonist. |
| CSN20252 | CGP-20712 | 137888-49-4 | CGP 20712 is a highly selective and potent β1-adrenoceptor antagonist (IC50 = 0.7 nM). Displays 10,000-fold selectivity over β2-adrenoceptors. |
| CSN18702 | Apraclonidine HCl | 73218-79-8 | Apraclonidine HCl is a clonidine-derived selective agonist of alpha2-adrenergic receptor. |
| CSN21296 | AGN 192836 | 171102-29-7 | AGN 192836 is a potent and selective α2 adrenergic agonist with EC50s of 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor, respectively. |
| CSN27295 | (S)-Viloxazine Hydrochloride | 56287-61-7 | (S)-Viloxazine Hydrochloride is the S-isomer of Viloxazine, a selective norepinephrine reuptake inhibitor (NRI) that can be used as an antidepressant. |
| CSN27296 | (R)-Viloxazine Hydrochloride | 56287-63-9 | (R)-Viloxazine Hydrochloride is the R-isomer of Viloxazine, a selective norepinephrine reuptake inhibitor (NRI) that can be used as an antidepressant. |