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Adrenergic Receptor
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN24589 | Zinterol | 37000-20-7 | Zinterol Hydrochloride is a selective agonist of β2-adrenoceptor with pKB values are 8.3 and < 5.7 for β2 and β1 receptors respectively in human artery. |
| CSN24046 | Xamoterol | 81801-12-9 | Xamoterol hemifumarate is a selective partial agonist of β1-adrenoceptor. |
| CSN24598 | WB 4101 HCl | 2170-58-3 | WB 4101 hydrochloride is a selective antagonist of α1A-adrenergic receptor. |
| CSN21863 | Tiodazosin | 66969-81-1 | Tiodazosin is a potent competitive postsynaptic alpha adrenergic receptor antagonist. |
| CSN21856 | Tertatolol | 83688-84-0 | Tertatolol is a potent antagonist of beta-adrenoceptor and 5-HT receptor, with unique renal vasodilatatory effects. |
| CSN24706 | Tampramine fumarate | 83166-18-1 | Tampramine is a tricyclic antidepressant (TCA). It acts as a selective norepinephrine reuptake inhibitor and has negligible affinity for adrenergic, histaminergic, and muscarinic receptors. |
| CSN24608 | Talsupram HCl | 25487-28-9 | Talsupram hydrochloride is a selective noradrenalin re-uptake inhibitor. |
| CSN24592 | AMibegron hydrochloride | 121524-09-2 | SR 58611A hydrochloride is a selective β3-adrenergic receptor agonist with anxiolytic and antidepressant effects in rodent models. |
| CSN24600 | SNAP 5089 HCl | 157066-77-8 | SNAP 5089 is a selective antagonist of α1A-adrenoceptor. |
| CSN24736 | SNAP 5089 | 157066-76-7 | SNAP 5089 is a selective antagonist of the subtype α1A-adrenoceptor. It binds with high affinity to α1A-adrenoceptor with a Ki value of 0.35 nM. |
| CSN24586 | RX 821002 HCl | 109544-45-8 | RX 821002 hydrochloride is a selective antagonist of α2-adrenoceptor with low affinity for imidazoline sites. The pKd values for α2D and α2A subtypes are 9.7 and 8.2 respectively. |
| CSN24576 | RS 17053 HCl | 169505-93-5 | RS 17053 hydrochloride is a selective antagonist of α1A-adrenoceptor with pKi and pA2 estimate of 9.1 - 9.9. |
| CSN24604 | Pronethalol HCl | 51-02-5 | Pronethalol hydrochloride is an antagonist of β-adrenergic antagonist for the treatment of angina pectoris and some arrhythmias. |
| CSN21781 | Pamatolol | 59110-35-9 | Pamatolol is a selective cardioselective antagonist of beta adrenergic receptor without sympathomimetic activity. |
| CSN21712 | Lintopride | 107429-63-0 | Lintopride is an antagonist of 5HT4 receptor and moderate antagonist of 5HT3. |
| CSN24584 | JP 1302 2HCl | 1259314-65-2 | JP 1302 dihydrochloride is an antagonist of α2C-adrenoceptor with Ki value of 28 nM. |
| CSN21958 | Indanazoline | 40507-78-6 | Indanazoline is a sympathomimetic imidazoline derivative and shows vasoconstrictive action . |
| CSN24602 | Imiloxan HCl | 81167-22-8 | Imiloxan hydrochloride is a highly selective antagonist of α2-adrenoceptor. |
| CSN22034 | GP2-114 | 130783-39-0 | GP2-114 is an activator of adrenergic receptor β, and produces current-dependent cardiovascular action when administered by transdermal iontophoresis. |
| CSN26499 | Fiduxosin free base | 208993-54-8 | Fiduxosin is an alpha(1)-adrenoceptor antagonist with higher affinity for alpha(1A)-adrenoceptors and for alpha(1D)-adrenoceptors than for alpha(1B)-adrenoceptors. |
| CSN33116 | Esreboxetine | 98819-76-2 | Esreboxetine is a selective norepinephrine reuptake inhibitor. |
| CSN24610 | Efaroxan HCl | 89197-00-2 | Efaroxan hydrochloride is an antagonist of α2 adrenoceptor and imidazoline I1 receptor ligand. The pKi values are 7.87, 7.42, 5.74, 7.28 and < 5 for α2A, α2B, α2C, I1 and I2 receptors, respectively. |
| CSN26575 | Detomidine carboxylic acid | 115664-39-6 | Detomidine carboxylic acid is the major urinary metabolite of Detomidine. Detomidine is a synthetic α2-adrenergic agonist and an animal analgesic sedative. Detomidine also has cardiac and respiratory effects and an antidiuretic action[1][2]. |
| CSN26579 | Dabuzalgron | 219311-44-1 | Dabuzalgron (previously codenamed R-450; Ro-115-1240) is a novel partial alphaA/IL receptor agonist that is administered in its hydrochloride form to control urethral smooth muscle contraction. The hemodynamic changes in the drug are very small and it is a potential drug for the treatment of stress urinary incontinence. |
| CSN26578 | Clonidine(200mg) | 4205-90-7 | Clonidine (also known as Catapres, Kapvay, Nexiclon, and Clophelin) is a sympathomimetic medication used to treat high blood pressure, attention deficit hyperactivity disorder, anxiety disorders, withdrawal (from either alcohol, opioids, or smoking), migraine, menopausal flushing, diarrhea, and certain pain conditions. It is classified as a centrally acting α2 adrenergic agonist and imidazoline receptor agonist that has been in clinical use for over 40 years. |
| CSN24596 | Cirazoline HCl | 40600-13-3 | Cirazoline hydrochloride is a selective agonist of alpha1-adrenoceptor. |
| CSN33167 | Bucindolol | 71119-11-4 | Bucindolol is a high-affinity, competitive beta blocker. |
| CSN24601 | B-HT 933 2HCl | 36067-72-8 | B-HT 933 dihydrochloride is selective agonist of α2-adrenoceptor. |
| CSN24583 | ARC 239 2HCl | 55974-42-0 | ARC 239 dihydrochloride is a selective antagonist of α2B adrenoceptor with pKD values of 8.8, 6.7 and 6.4 for α2B, α2A, and α2D receptors respectively. |
| CSN26577 | Arbutamine | 128470-16-6 | Arbutamine is a cardiac stimulant. It stimulates adrenergic receptors. Arbutamine is a synthetic catecholamine with positive chronotropic and inotropic properties, used in echocardiography and diagnostic coronary angiography. Arbutamine binds to and activates beta-1 adrenergic receptors in the myocardium, thereby increasing heart rate and increasing force of myocardial contraction. Arbutamine, administered through a closed-loop, computer-controlled drug-delivery system, is indicated to elicit acute cardiovascular responses, similar to those produced by exercise, in order to aid in diagnosing the presence or absence of coronary artery disease in patients who cannot exercise adequately. |
| CSN24599 | A 61603 hydrobromide | 107756-30-9 | A 61603 hydrobromide is a selective α1A-adrenergic receptor agonist. |
| CSN24609 | 3-MPPI | 133399-65-2 | 3-MPPI is a very potent ligand for α1 sites and regulates smooth muscle contraction. The pKi values for α1B, α1D, α1A adrenoceptors are 8.74, 9.44, 9.57 respectively. It also binds to 5-HT1A sites (Ki = 50 nM). |
| CSN24595 | 2-PMDQ | 139047-55-5 | 2-PMDQ is a selective α1-adrenoceptor antagonist with antihypertensive effect. |
| CSN24597 | 2-MPMDQ | 149847-77-8 | 2-MPMDQ is a selective antagonist of α1-AR adrenoceptor and can act as a hypotensive. |
