优势价格
快速发货
品质保证
技术支持
400-920-2911 sales@csnpharm.cn
Adrenergic Receptor
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN24598 | WB 4101 HCl | 2170-58-3 | WB 4101 hydrochloride is a selective antagonist of α1A-adrenergic receptor. |
| CSN24706 | Tampramine fumarate | 83166-18-1 | Tampramine is a tricyclic antidepressant (TCA). It acts as a selective norepinephrine reuptake inhibitor and has negligible affinity for adrenergic, histaminergic, and muscarinic receptors. |
| CSN24608 | Talsupram HCl | 25487-28-9 | Talsupram hydrochloride is a selective noradrenalin re-uptake inhibitor. |
| CSN24592 | Amibegron hydrochloride | 121524-09-2 | SR 58611A hydrochloride is a selective β3-adrenergic receptor agonist with anxiolytic and antidepressant effects in rodent models. |
| CSN24600 | SNAP 5089 HCl | 157066-77-8 | SNAP 5089 is a selective antagonist of α1A-adrenoceptor. |
| CSN24736 | SNAP 5089 | 157066-76-7 | SNAP 5089 is a selective antagonist of the subtype α1A-adrenoceptor. It binds with high affinity to α1A-adrenoceptor with a Ki value of 0.35 nM. |
| CSN11918 | Sertindole | 106516-24-9 | Sertindole, a neuroleptic, is one of the antipsychotic medications available, with a high affinity for dopamine D2, serotonin 5-HT2A, 5-HT2C, and α1-adrenergic receptors. |
| CSN24604 | Pronethalol hydrochloride | 51-02-5 | Pronethalol hydrochloride is an antagonist of β-adrenergic antagonist for the treatment of angina pectoris and some arrhythmias. |
| CSN24602 | 2-((2,3-Dihydrobenzo[b][1,4]dioxin-2-yl)methyl)-1-ethyl-1H-imidazole hydrochloride | 81167-22-8 | Imiloxan hydrochloride is a highly selective antagonist of α2-adrenoceptor. |
| CSN26499 | Fiduxosin | 208993-54-8 | Fiduxosin is an alpha(1)-adrenoceptor antagonist with higher affinity for alpha(1A)-adrenoceptors and for alpha(1D)-adrenoceptors than for alpha(1B)-adrenoceptors. |
| CSN33116 | (S)-2-((S)-(2-Ethoxyphenoxy)(phenyl)methyl)morpholine | 98819-76-2 | Esreboxetine is a selective norepinephrine reuptake inhibitor. |
| CSN24610 | Efaroxan hydrochloride | 89197-00-2 | Efaroxan hydrochloride is an antagonist of α2 adrenoceptor and imidazoline I1 receptor ligand. The pKi values are 7.87, 7.42, 5.74, 7.28 and < 5 for α2A, α2B, α2C, I1 and I2 receptors, respectively. |
| CSN26575 | Detomidine carboxylic acid | 115664-39-6 | Detomidine carboxylic acid is the major urinary metabolite of Detomidine. Detomidine is a synthetic α2-adrenergic agonist and an animal analgesic sedative. Detomidine also has cardiac and respiratory effects and an antidiuretic action[1][2]. |
| CSN26579 | Dabuzalgron | 219311-44-1 | Dabuzalgron (previously codenamed R-450; Ro-115-1240) is a novel partial alphaA/IL receptor agonist that is administered in its hydrochloride form to control urethral smooth muscle contraction. The hemodynamic changes in the drug are very small and it is a potential drug for the treatment of stress urinary incontinence. |
| CSN26578 | Clonidine | 4205-90-7 | Clonidine (also known as Catapres, Kapvay, Nexiclon, and Clophelin) is a sympathomimetic medication used to treat high blood pressure, attention deficit hyperactivity disorder, anxiety disorders, withdrawal (from either alcohol, opioids, or smoking), migraine, menopausal flushing, diarrhea, and certain pain conditions. It is classified as a centrally acting α2 adrenergic agonist and imidazoline receptor agonist that has been in clinical use for over 40 years. |
| CSN24596 | Cirazoline hydrochloride | 40600-13-3 | Cirazoline hydrochloride is a selective agonist of alpha1-adrenoceptor. |
| CSN33167 | Bucindolol | 71119-11-4 | Bucindolol is a high-affinity, competitive beta blocker. |
| CSN24601 | Azepexole dihydrochloride | 36067-72-8 | B-HT 933 dihydrochloride is selective agonist of α2-adrenoceptor. |
| CSN26577 | Arbutamine | 128470-16-6 | Arbutamine is a cardiac stimulant. It stimulates adrenergic receptors. Arbutamine is a synthetic catecholamine with positive chronotropic and inotropic properties, used in echocardiography and diagnostic coronary angiography. Arbutamine binds to and activates beta-1 adrenergic receptors in the myocardium, thereby increasing heart rate and increasing force of myocardial contraction. Arbutamine, administered through a closed-loop, computer-controlled drug-delivery system, is indicated to elicit acute cardiovascular responses, similar to those produced by exercise, in order to aid in diagnosing the presence or absence of coronary artery disease in patients who cannot exercise adequately. |
| CSN32920 | 4-(2-((2,4,6-Trifluorophenoxy)methyl)phenyl)piperidine | 1227056-84-9 | Ampreloxetine is a norepinephrine reuptake inhibitor. |
| CSN32921 | 4-(2-((2,4,6-Trifluorophenoxy)methyl)phenyl)piperidine hydrochloride | 1227056-87-2 | Ampreloxetine is a norepinephrine reuptake inhibitor. |
| CSN24599 | A-61603 | 107756-30-9 | A 61603 hydrobromide is a selective α1A-adrenergic receptor agonist. |
| CSN24609 | 3-MPPI | 133399-65-2 | 3-MPPI is a very potent ligand for α1 sites and regulates smooth muscle contraction. The pKi values for α1B, α1D, α1A adrenoceptors are 8.74, 9.44, 9.57 respectively. It also binds to 5-HT1A sites (Ki = 50 nM). |
| CSN24595 | 2-PMDQ | 139047-55-5 | 2-PMDQ is a selective α1-adrenoceptor antagonist with antihypertensive effect. |
| CSN24597 | 2-((4-(2-Methoxyphenyl)piperazin-1-yl)methyl)-6-methyl-2,3-dihydroimidazo[1,2-c]quinazolin-5(6H)-one | 149847-77-8 | 2-MPMDQ is a selective antagonist of α1-AR adrenoceptor and can act as a hypotensive. |
| CSN41014 | Iprindole | 5560-72-5 | |
| CSN40605 | Jatrorrhizine hydroxide | 483-43-2 | |
| CSN39211 | ADRA1D receptor antagonist 1 | 1191908-14-1 | |
| CSN42110 | Spiperone hydrochloride | 2022-29-9 | |
| CSN34474 | QF0301B | 149247-12-1 | |
| CSN36657 | L-745870 hydrochloride | 1173023-36-3 | |
| CSN37126 | L-745870 trihydrochloride | 866021-03-6 | |
| CSN42437 | Dextromilnacipran | 96847-55-1 | |
| CSN42968 | Tedatioxetine hydrobromide | 960151-65-9 | |
| CSN63870 | Paliperidone-d4 | 1020719-55-4 | |
| CSN62845 | Melitracen-d6 hydrochloride | 1189648-08-5 | |
| CSN66549 | Tesofensine | 195875-84-4 | |
| CSN83984 | (-)-Penbutolol | 38363-40-5 | |
| CSN83992 | Melitracen | 5118-29-6 | |
| CSN90871 | 1-[4-(4-fluorophenyl)-4-oxobutyl][1,4-bipiperidine]-4-carboxamidedihydrochloride | 2448-68-2 | |
| CSN107472 | 3-(3-(4-Phenylpiperazin-1-yl)propyl)quinazoline-2,4(1H,3H)-dione | 2208-51-7 | |
| CSN103803 | Butanserin | 87051-46-5 | |
| CSN107372 | 4-[2-(4-Methylphenyl)sulfanylphenyl]piperidine | 508233-95-2 |
