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Adrenergic Receptor

Adrenergic Receptor

货号 产品名 CAS号 信息
CSN18767 Tolazoline HCl 59-97-2 Tolazoline HCl is a competitive non-selective α-adrenergic receptor antagonist, used as a a vasodilator directly acting on blood vessels and also increasing cardiac output.
CSN12086 Tiamenidine 31428-61-2 Thioridazine is an antipsychotic drug, used in the treatment of schizophrenia and psychosis, shows D4 selectivity or serotonin antagonism.
CSN19307 Tetrahydrozoline HCl 522-48-5 Tetrahydrozoline HCl is an imidazole-derived alpha-adrenergic receptor agonist which can result vasoconstriction and decreased nasal and ophthalmic congestion.
CSN25553 SR59230A 174689-39-5 SR59230A is a potent and selective Adrenergic Receptor β3 antagonist with IC50 values of 40, 408, and 648nM for Adrenergic Receptor β3, β1 and β2, respectively. It shows blood-brain barrier penetrability.
CSN21822 Rauwolscine HCl 6211-32-1 Rauwolscine hydrochloride is an antagonist of alpha2-adrenergic and partial agonist of 5-HT1A receptor.
CSN18749 Piribedil 3605-01-4 Piribedil is an antiparkinsonian agent and piperazine derivative which acts as a D2 and D3 receptor agonist.
CSN18980 Piperoxan HCl 135-87-5 Piperoxan HCl is an α2 adrenoceptor antagonist.
CSN18661 Naphazoline 835-31-4 Naphazoline is the common name for 2-(1-naphthylmethyl)-2-imidazoline HCl, it is a sympathomimetic agent with marked alpha adrenergic activity.
CSN22198 LY377604 204592-94-9 LY377604 is a human β3-adrenergic receptor agonist with an EC50 of 2.4 nM and also a β1- and β2-adrenergic receptor antagonist. Ly377604 has been used in trials studying the treatment of Obesity.
CSN23830 Lofexidine 31036-80-3 Lofexidine is a selective α2-receptor agonist, commonly used to alleviate the physical symptoms of heroin and other types of opioid withdrawal[1][2].
CSN18745 Lofexidine HCl 21498-08-8 Lofexidine HCl is an α2A-adrenergic receptor agonist, commonly used to alleviate the physical symptoms of heroin and other types of opioid withdrawal.
CSN21997 Labetalone HCl 96441-14-4 Labetalone hydrochloride is hydrochloride form of labetalone, a blocker of both alpha- and beta-adrenergic receptors that is used as an antihypertensive.
CSN22444 L-765314 189349-50-6 L-765314 is a potent and selective α1b adrenergic receptor antagonist with Kis of 5.4±0.6 nM and 2.0±0.66 nM for rat and human α1b adrenergic receptor, respectively.
CSN18526 L-(-)-α-Methyldopa HCl 884-39-9 L-(-)-α-Methyldopa HCl is an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive drug used as a sympatholytic or antihypertensive.
CSN19723 Isoxsuprine HCl 579-56-6 Isoxsuprine is a modulator of β2 adrenoreceptor and has agonist or antagonist effects.
CSN19742 Idazoxan HCl 79944-56-2 Idazoxan is an alpha2-adrenoceptor antagonist potentially for the treatment of schizophrenia.
CSN20255 ICI-118551 72795-19-8 ICI-118551 is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors, respectively.
CSN23785 GUANABENZ 5051-62-7 Guanabenz is an agonist of α2-adrenergic receptor with antihypertensive effect and is enerally used in combination with diuretics.
CSN19298 Fenspiride HCl 5053-08-7 Fenspiride HCl is an antagonist of α-adrenergic receptors and H1 histamine receptors and also inhibits phosphodiesterase 4 and phosphodiesterase 3 activities with logIC50 values of 4.16 and 3.44, respectively.
CSN19404 Detomidine 76631-46-4 Detomidine produce dose-dependent sedative and analgesic effects, is a nonnarcotic, synthetic α2-adrenergic agonist.
CSN20033 CL316243 Disodium Salt 138908-40-4 CL-316243 is a potent and highly selective β3-adrenoceptor agonist (EC50 = 3 nM) and > 10000-fold selective over β1 and β2 receptors. CL-316243 restores the expression of down-regulated fatty acid oxidation genes in type 2 diabetic mice.
CSN20252 CGP-20712 137888-49-4 CGP 20712 is a highly selective and potent β1-adrenoceptor antagonist (IC50 = 0.7 nM). Displays 10,000-fold selectivity over β2-adrenoceptors.
CSN19303 Bopindolol 62658-63-3 Bopindolol is a beta blocker. It is an ester which acts as a prodrug for its active metabolite 4-(3-t-butylamino-2-hydroxypropoxy)-2-methylindole.
CSN18702 Apraclonidine HCl 73218-79-8 Apraclonidine HCl is a clonidine-derived selective agonist of alpha2-adrenergic receptor.
CSN21296 AGN 192836 171102-29-7 AGN 192836 is a potent and selective α2 adrenergic agonist with EC50s of 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor, respectively.
CSN27295 (S)-Viloxazine Hydrochloride 56287-61-7 (S)-Viloxazine Hydrochloride is the S-isomer of Viloxazine, a selective norepinephrine reuptake inhibitor (NRI) that can be used as an antidepressant.
CSN27296 (R)-Viloxazine Hydrochloride 56287-63-9 (R)-Viloxazine Hydrochloride is the R-isomer of Viloxazine, a selective norepinephrine reuptake inhibitor (NRI) that can be used as an antidepressant.
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