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Adrenergic Receptor
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN24046 | Xamoterol | 81801-12-9 | Xamoterol hemifumarate is a selective partial agonist of β1-adrenoceptor. |
| CSN12102 | Todralazine | 14679-73-3 | Todralazine is capable of reducing blood pressure preferentially in hypertension. |
| CSN21863 | Tiodazosin | 66969-81-1 | Tiodazosin is a potent competitive postsynaptic alpha adrenergic receptor antagonist. |
| CSN12086 | Tiamenidine | 31428-61-2 | Thioridazine is an antipsychotic drug, used in the treatment of schizophrenia and psychosis, shows D4 selectivity or serotonin antagonism. |
| CSN21856 | Tertatolol | 83688-84-0 | Tertatolol is a potent antagonist of beta-adrenoceptor and 5-HT receptor, with unique renal vasodilatatory effects. |
| CSN25553 | SR59230A | 174689-39-5 | SR59230A is a potent and selective Adrenergic Receptor β3 antagonist with IC50 values of 40, 408, and 648nM for Adrenergic Receptor β3, β1 and β2, respectively. It shows blood-brain barrier penetrability. |
| CSN24580 | Benalfocin hydrochloride | 86129-54-6 | SKF 86466 hydrochloride is selective antagonist of pre- (Ki= 13 nM) and post-junctional (Ki= 17 nM) α2-adrenoceptors with antihypertensive activity in rat model. |
| CSN24586 | 2-Methoxyidazoxan HCl | 109544-45-8 | RX 821002 hydrochloride is a selective antagonist of α2-adrenoceptor with low affinity for imidazoline sites. The pKd values for α2D and α2A subtypes are 9.7 and 8.2 respectively. |
| CSN24576 | RS 17053 HCl | 169505-93-5 | RS 17053 hydrochloride is a selective antagonist of α1A-adrenoceptor with pKi and pA2 estimate of 9.1 - 9.9. |
| CSN24703 | Rec 15/2615 dihydrochloride | 173059-17-1 | REC-2615 (HCl) is a α1B-adrenoceptor antagonist potentially for the treatment of female sexual dysfunction. |
| CSN21822 | Rauwolscine HCl | 6211-32-1 | Rauwolscine hydrochloride is an antagonist of alpha2-adrenergic and partial agonist of 5-HT1A receptor. |
| CSN21781 | Pamatolol | 59110-35-9 | Pamatolol is a selective cardioselective antagonist of beta adrenergic receptor without sympathomimetic activity. |
| CSN19390 | Moxisylyte HCl | 964-52-3 | Moxisylyte HCl is an alpha 1-blocker antagonist, it can vasodilates cerebral vessels without reducing blood pressure. |
| CSN11443 | Midodrine | 42794-76-3 | Midodrine is an α1-receptor agonist, for the treatment of dysautonomia and orthostatic hypotension. |
| CSN18273 | Midodrine HCl | 43218-56-0 | Midodrine HCl is an α1-receptor agonist, for the treatment of dysautonomia and orthostatic hypotension. |
| CSN22198 | LY377604 | 204592-94-9 | LY377604 is a human β3-adrenergic receptor agonist with an EC50 of 2.4 nM and also a β1- and β2-adrenergic receptor antagonist. Ly377604 has been used in trials studying the treatment of Obesity. |
| CSN23830 | Lofexidine | 31036-80-3 | Lofexidine is a selective α2-receptor agonist, commonly used to alleviate the physical symptoms of heroin and other types of opioid withdrawal[1][2]. |
| CSN21712 | Lintopride | 107429-63-0 | Lintopride is an antagonist of 5HT4 receptor and moderate antagonist of 5HT3. |
| CSN21711 | Lidanserin | 73725-85-6 | Lidanserin is antagonist of 5-HT2A and α1-adrenergic receptor. |
| CSN23826 | Landiolol HCl | 144481-98-1 | Landiolol hydrochloride (ONO1101 hydrochloride) is a highly beta1 selective ultra-short acting beta-blocker (β1/β2 selectivity = 255:1, a half-life of 4 min)， acts as an adrenoceptor antagonist[1]. |
| CSN21997 | Labetalone HCl | 96441-14-4 | Labetalone hydrochloride is hydrochloride form of labetalone, a blocker of both alpha- and beta-adrenergic receptors that is used as an antihypertensive. |
| CSN22444 | L-765314 | 189349-50-6 | L-765314 is a potent and selective α1b adrenergic receptor antagonist with Kis of 5.4±0.6 nM and 2.0±0.66 nM for rat and human α1b adrenergic receptor, respectively. |
| CSN24584 | JP1302 2HCl | 1259314-65-2 | JP 1302 dihydrochloride is an antagonist of α2C-adrenoceptor with Ki value of 28 nM. |
| CSN21687 | Indanidine | 85392-79-6 | Indanidine is an agonist of alpha-adrenergic receptor. |
| CSN21958 | Indanazoline | 40507-78-6 | Indanazoline is a sympathomimetic imidazoline derivative and shows vasoconstrictive action . |
| CSN23785 | Guanabenz | 5051-62-7 | Guanabenz is an agonist of α2-adrenergic receptor with antihypertensive effect and is enerally used in combination with diuretics. |
| CSN22034 | GP2-114 | 130783-39-0 | GP2-114 is an activator of adrenergic receptor β, and produces current-dependent cardiovascular action when administered by transdermal iontophoresis. |
| CSN21621 | Ecastolol | 77695-52-4 | Ecastolol is an antagonist of beta adrenergic receptor with antianginal activities. |
| CSN21614 | Dopexamine HCl | 86484-91-5 | Dopexamine hydrochloride is an agonist of β2 adrenergic receptor. |
| CSN21435 | Benzquinamide | 63-12-7 | Benzquinamid, an antiemetic, can bind to the α2A, α2B, and α2C adrenergic receptors with Ki values of 1365, 691, and 545 nM, respectively. |
| CSN21511 | (±)-Befunolol | 39552-01-7 | Befunolol is a blocker of β-adrenoceptor. |
| CSN24583 | ARC 239 2HCl | 55974-42-0 | ARC 239 dihydrochloride is a selective antagonist of α2B adrenoceptor with pKD values of 8.8, 6.7 and 6.4 for α2B, α2A, and α2D receptors respectively. |
| CSN27295 | (S)-2-((2-Ethoxyphenoxy)methyl)morpholine hydrochloride | 56287-61-7 | (S)-Viloxazine Hydrochloride is the S-isomer of Viloxazine, a selective norepinephrine reuptake inhibitor (NRI) that can be used as an antidepressant. |
| CSN27296 | (R)-Viloxazine HCl | 56287-63-9 | (R)-Viloxazine Hydrochloride is the R-isomer of Viloxazine, a selective norepinephrine reuptake inhibitor (NRI) that can be used as an antidepressant. |
