AMPAR
货号 | 产品名 | CAS号 | 信息 |
---|---|---|---|
CSN13605 | β-ODAP | 5302-45-4 | β-ODAP is an analog of glutamic acid present in Lathyrus sativus (grass pea) that activates AMPA receptors. |
CSN17953 | ZK200775 | 161605-73-8 | ZK200775 is a highly selective AMPA/kainate antagonist with little activity against NMDA with Ki values of 3.2 nM, 100 nM, and 8.5 μM against quisqualate, kainate, and NMDA, respectively. |
CSN13591 | Talampanel | 161832-65-1 | Talampanel, a potent and selective AMPA-receptor antagonist, is a potential antiepileptic drug (AED). |
CSN13810 | Piracetam | 7491-74-9 | Piracetam is a cyclic derivative of GABA which works as a positive allosteric modulator of the AMPA receptor. |
CSN24155 | Philanthotoxin 74 2HCl | 1227301-51-0 | Philanthotoxin 74 dihydrochloride (PhTx 74) is an AMPAR antagonist; inhibits GluR3 and GluR1 with IC50s of 263 and 296 nM, respectively. |
CSN17813 | PEPA | 141286-78-4 | PEPA is an allosteric modulator of AMPA receptors and binds to the GluA2o and GluA3o LBDs and can be utilized as an indicator of AMPA receptor heterogeneity. |
CSN13580 | Noopept | 157115-85-0 | Noopept is a potent nootropic that improves cognitive ability. |
CSN22241 | NBQX | 118876-58-7 | NBQX is a potent, selective and competitive AMPAR antagonist, which shows activity of neuroprotective and anticonvulsant. |
CSN17585 | Naspm | 122306-11-0 | Naspm is a potent and selective Ca2+ permeable AMPA receptor (Ca-perm AMPAR) blocker. |
CSN17275 | Naspm 3HCl | 1049731-36-3 | Naspm 3HCl is a potent and selective Ca2+ permeable AMPA receptor (Ca-perm AMPAR) blocker. |
CSN22957 | LY 404187 | 211311-95-4 | LY 404187 is a selective positive allosteric modulator of AMPA receptors with IC50s of 0.15, 0.21, 1.66 and 5.65 μM for GluA2i, GluA4i, GluA3i and GluA1i respectively. |
CSN11282 | Lentinan | 37339-90-5 | Lentinan, a natural product isolated and purified from shiitake mushroom (Lentinus edodes), is an intravenous anti-tumor polysaccharide isolated from the fruit body of shiitake. |
CSN25435 | Lentinan | 37339-90-5 | Lentinan, a natural product isolated and purified from shiitake mushroom (Lentinus edodes), is an intravenous anti-tumor polysaccharide isolated from the fruit body of shiitake. |
CSN16600 | L-Theanine | 3081-61-6 | L-theanine is an amino acid found most commonly in tea leaves and binds to ionotropic glutamate receptors in the micromolar range, including the AMPA and kainate receptors and, to a lesser extent, the NMDA receptor. |
CSN25362 | IDRA 21 | 22503-72-6 | IDRA-21 is a positive AMPA receptor modulator. IDRA-21 inhibits synaptic and extrasynaptic NMDA receptor mediated events in cultured cerebellar granule cells. IDRA 21 enhances ischemic hippocampal neuron injury. |
CSN21401 | L-Quisqualic Acid | 52809-07-1 | Glutamate receptor agonist acting at AMPA receptors and metabotropic glutamate receptors positively linked to phosphoinositide hydrolysis. Sensitizes neurons in hippocampus to depolarization by L-AP6 (the so called 'quis' effect). |
CSN27523 | Farampator | 211735-76-1 | Farampator (CX-691;Org24448) is an AMPA receptor positive modulator. |
CSN22784 | CX 614 | 191744-13-5 | CX 614 is a positive allosteric modulator of AMPA receptors. |
CSN22766 | CNQX | 115066-14-3 | CNQX is a potent and selective non-NMDA iGluR antagonist. |
CSN24616 | ATPA | 140158-50-5 | ATPA is a selective and potent GluK1 kainate receptor agonist with Ki of 4.3 nM. |
CSN25263 | 1-BCP | 34023-62-6 | 1-BCP is can modulate AMPA receptor gated currents and enhence memory. |
CSN11876 | (S)-Willardiine | 21416-43-3 | (S)-Willardiine is a potent agonist of AMPA/kainate receptors with EC50 of 44.8 μM. |
CSN23429 | L-Glutamic Acid | 56-86-0 | (S)-Glutamic acid acts as an excitatory neurotransmitter in the central nervous system. |
CSN22635 | (S)-AMPA | 83643-88-3 | (S)-AMPA is a selective AMPA agonist. |
CSN22631 | (RS)-AMPA | 77521-29-0 |