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Angiotensin Receptor
货号 | 产品名 | CAS号 | 信息 |
---|---|---|---|
CSN25363 | ZD 7155(hydrochloride) | 146709-78-6 | ZD 7155 hydrochloride is selective competitive antagonist of the angiotensin II type 1 (AT1) receptor. |
CSN12536 | Valsartan | 137862-53-4 | Valsartan is a selective angiotensin II AT1 receptor antagonist with elimination half-life of 6 hours. |
CSN16012 | trans-Tranilast | 70806-55-2 | trans-Tranilast is an antiallergic drug, used to treat bronchial asthma, allergic rhinitis and atopic dermatitis. |
CSN17430 | Tranilast sodium | 104931-56-8 | Tranilast is an antiallergic agent. |
CSN12122 | Tranilast | 53902-12-8 | Tranilast can antagonize angiotensin II and also work as an antiallergic agent. It showed inhibitory effect for NLRP3 inflammasome but not for NLRC4 or AIM2 inflammasome. Tranilast impaired the endogenous NLRP3-ASC interaction but did not affect the NLRP3-NEK7 interaction, raising the possibility that it targets NLRP3 directly. |
CSN12552 | Telmisartan | 144701-48-4 | Telmisartan is an angiotensin II receptor antagonist with Ki value of 3.7nM, used in the management of hypertension with elimination half-life of 24 hours. |
CSN12037 | Tasosartan | 145733-36-4 | Tasosartan is a long-acting angiotensin II receptor blocker. |
CSN21304 | SL910102 | 144756-71-8 | SL910102 is a nonpeptide angiotensin AT1 receptor antagonist. |
CSN16875 | PD 123319 ditrifluoroacetate | 136676-91-0 | PD123319 Ditrifluoroacetate is a potent, selective and non-peptide angiotensin AT2 receptor antagonist. |
CSN11662 | PD 123319 | 130663-39-7 | PD 123319 is a potent, selective AT2 angiotensin II receptor antagonist with IC50 of 34 nM. |
CSN12551 | Olmesartan medoxomil | 144689-63-4 | Olmesartan Medoxomil is a synthetic imidazole-derived angiotensin II receptor antagonist, acting as a prodrug with an antihypertensive property. |
CSN11603 | Olmesartan | 144689-24-7 | Olmesartan is an antagonist of angiotensin II receptor, working as an antihypertensive agent. |
CSN12515 | Losartan potassium | 124750-99-8 | Losartan Potassium is the potassium salt form of Losartan, which is a compeitive AT1 receptor inhibitor with IC50 value of 20 nM. |
CSN11333 | Losartan | 114798-26-4 | Losartan is a compeitive AT1 receptor inhibitor with IC50 value of 20 nM. |
CSN17407 | Losartan D4 | 1030937-27-9 | Losartan D4 is deuterium labeled Losartan, which is an angiotensin II receptor antagonist. |
CSN16211 | Sacubitril/Valsartan | 936623-90-4 | LCZ 696 is a mixture of neprilysin inhibitor sacubitril and the angiotensin receptor blocker valsartan in a ratio of 1:1. |
CSN22035 | L-159282 | 157263-00-8 | L-159282 is a highly potent, orally active, nonpeptide angiotensin II receptor antagonist, with anti-hypertensive activity. |
CSN12537 | Irbesartan | 138402-11-6 | Irbesartan is a selective and competitive nonpeptide angiotensin II antagonist with antihypertensive activity. |
CSN13567 | Fimasartan | 247257-48-3 | Fimasartan is an improved non-peptide angiotensin II receptor blocker used for the treatment of hypertension and heart failure, which enables higher potency and longer duration than losartan. |
CSN24625 | Losartan Carboxylic Acid | 124750-92-1 | EXP 3174 is a selective and noncompetitive antagonist of AT1 receptor with IC50 of 37 nM. |
CSN10923 | Eprosartan mesylate | 144143-96-4 | Eprosartan Mesylate is a reversible and competitive angiotensin II receptor inhibitor. |
CSN10922 | Eprosartan | 133040-01-4 | Eprosartan is an angiotensin II receptor antagonist used for the treatment of high blood pressure. |
CSN18823 | Olodanrigan | 1316755-16-4 | EMA401, a highly selective AT2R antagonist, inhibition of augmented AngII/AT2R induced p38 and p42/p44 MAPK activation, and hence inhibition of DRG neuron hyperexcitability and sprouting of DRG neurons. |
CSN17650 | CGP-42112 | 127060-75-7 | CGP-42112 is a potent Angiotensin-II subtype 2 receptor (AT2 R) agonist. |
CSN12544 | Candesartan | 139481-59-7 | Candesartan is a benzimidazole-derived and competitive AT1 inhibitor with IC50 value of 0.26 nM. |
CSN12553 | Candesartan Cilexetil | 145040-37-5 | Candesartan Cilexetil is a benzimidazole-derived and competitive AT1 inhibitor with IC50 value of 0.26 nM. |
CSN17695 | BIBS 39 | 133085-33-3 | BIBS 39 is a nonpeptide angiotensin II (AII) receptor antagonist. |
CSN12705 | Azilsartan medoxomil | 863031-21-4 | Azilsartan Medoxomil is an orally available angiotensin II type 1 (AT1) receptor antagonist with IC50 value of 2.6 nM. |
CSN13633 | Azilsartan medoxomil monopotassium | 863031-24-7 | Azilsartan medoxomil is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension. |
CSN10369 | Azilsartan | 147403-03-0 | Azilsartan is an orally available angiotensin II type 1 (AT1) receptor antagonist with IC50 value of 2.6 nM. |
CSN16922 | AVE 0991 sodium salt | 306288-04-0 | AVE 0991 sodium is a nonpeptide Ang-(1-7) receptor Mas agonist, represents an important step for exploration of the effects of Ang-(1-7) and testing of its potential as a cardiovascular drug. |
CSN16917 | AVE 0991 | 304462-19-9 | AVE 0991 is a nonpeptide Ang-(1-7) receptor Mas agonist. |
CSN20314 | AT2 receptor agonist C21 | 477775-14-7 | AT2R agonist C21 is a small-molecule ATR receptor (AT2R) agonist. |
CSN10313 | Angiotensin II human | 4474-91-3 | Angiotensin II human is a peptide hormone that causes vasoconstriction and a subsequent increase in blood pressure. |
CSN10119 | Angiotensin II 5-valine | 58-49-1 | Angiotensin II 5-valine is an angiotensin II analog which is an agonist at angiotensin receptors. |
CSN21490 | Angiotensin II (3-8), human | 12676-15-2 | Angiotensin II (3-8), human is an agonist of angiotensin AT1 receptor. Its activation is relatively weak. |
CSN13483 | Sacubitril | 149709-62-6 | AHU-377 and valsartan can compose LCZ696 in a 1:1 molar ratio. It also works as an inhibitor of neprilysin with IC50 value of 5 nM. |
CSN22012 | A81988 | 141887-34-5 | A81988 is a potent, competitive, non-peptidic antagonist of angiotensin AT1 receptors. |
CSN21995 | (2S,4S)-Sacubitril | 149709-63-7 | 2S,4S-Sacubitril is the impurity of Sacubitril and Sacubitril is approved by the Food and Drug Administration for use in combination with valsartan for the treatment of patients with heart failure. |
CSN21996 | 2R,4S-Sacubitril | 761373-05-1 | 2R,4S-Sacubitril is the impurity of Sacubitril and Sacubitril is approved by the Food and Drug Administration for use in combination with valsartan for the treatment of patients with heart failure. |
CSN28996 | Sparsentan | 254740-64-2 |