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Apelin Receptor

货号 产品名 CAS号 信息
CSN23653 (Glp1)-Apelin-13 217082-60-5 [Pyr1]-Apelin-13 is a potent peptide apelin agonist with EC50 of 0.37 nM.
CSN24633 MM 54 1313027-43-8 MM 54 is a potent apelin receptor antagonist with Ki of 82 nM and IC50 of 93 nM.
CSN26194 MM 07 1876450-21-3 MM 07 is a biased apelin receptor agonist, with a KD of 300 nM in CHO-K1 cells and a KD of 172 nM in human heart. It stimulates endothelial NOS phosphorylation and expression, promotes proliferation, and attenuates apoptosis of human pulmonary arterial endothelial cells in vitro.
CSN21287 ML221 877636-42-5 ML221 is a potent apelin receptor (APJ) antagonist with IC50s of 0.70 μM and 1.75 μM in cAMP and β-arrestin assay respectively.
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