Apelin Receptor

Apelin Receptor
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货号	产品名	CAS号	信息
CSN23653	[Pyr1]-Apelin-13	217082-60-5	[Pyr1]-Apelin-13 is a potent peptide apelin agonist with EC50 of 0.37 nM.
CSN24633	MM 54	1313027-43-8	MM 54 is a potent apelin receptor antagonist with Ki of 82 nM and IC50 of 93 nM.
CSN26194	MM 07	1876450-21-3	MM 07 is a biased apelin receptor agonist, with a KD of 300 nM in CHO-K1 cells and a KD of 172 nM in human heart. It stimulates endothelial NOS phosphorylation and expression, promotes proliferation, and attenuates apoptosis of human pulmonary arterial endothelial cells in vitro.
CSN21287	ML221	877636-42-5	ML221 is a potent apelin receptor (APJ) antagonist with IC50s of 0.70 μM and 1.75 μM in cAMP and β-arrestin assay respectively.
CSN23651	Apelin-13	217082-58-1	Apelin-13 is the endogenous ligand of the orphan G protein-coupled receptor APJ, activates APJ receptor with an EC50 value of 0.37 nM in CHO cells[1][2].