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货号 | 产品名 | CAS号 | 信息 |
---|---|---|---|
CSN23653 | [Pyr1]-Apelin-13 | 217082-60-5 | [Pyr1]-Apelin-13 is a potent peptide apelin agonist with EC50 of 0.37 nM. |
CSN24633 | MM 54 | 1313027-43-8 | MM 54 is a potent apelin receptor antagonist with Ki of 82 nM and IC50 of 93 nM. |
CSN26194 | MM 07 | 1876450-21-3 | MM 07 is a biased apelin receptor agonist, with a KD of 300 nM in CHO-K1 cells and a KD of 172 nM in human heart. It stimulates endothelial NOS phosphorylation and expression, promotes proliferation, and attenuates apoptosis of human pulmonary arterial endothelial cells in vitro. |
CSN21287 | ML221 | 877636-42-5 | ML221 is a potent apelin receptor (APJ) antagonist with IC50s of 0.70 μM and 1.75 μM in cAMP and β-arrestin assay respectively. |
CSN23651 | Apelin-13 | 217082-58-1 | Apelin-13 is the endogenous ligand of the orphan G protein-coupled receptor APJ, activates APJ receptor with an EC50 value of 0.37 nM in CHO cells[1][2]. |
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