ATP-binding Cassette Sub-family G member 2 | Membrane Transporter/Ion Channel| CSNpharm

BCRP

BCRP
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货号	产品名	CAS号	信息
CSN17725	YHO-13351	1346753-00-1	YHO-13351 is the water-soluble prodrug of YHO-13177, which is a potent and specific inhibitor of BCRP.
CSN18565	YHO-13351 free base	912288-64-3	YHO-13351 free base is the water-soluble prodrug of YHO-13177, which is a potent and specific inhibitor of BCRP.
CSN18564	YHO-13177	912287-56-0	YHO-13177 is a selective and potent inhibitor of BCRP, it potentiates the cytotoxicity of SN-38 in cancer cells and has no effect on P-glycoprotein–mediated paclitaxel resistance in MDR1-transduced human leukemia K562 cells.
CSN20009	ML753286	1699720-89-2	ML753286 is a potent inhibitor for BCRP, but not for P-glycoprotein (P-gp), organic anion-transporting polypeptide (OATP), or major cytochrome P450s (CYPs).
CSN17368	KS176	1253452-78-6	KS176 is a potent and selective inhibitor for the breast cancer resistance protein (BCRP) multidrug transporter with IC50s of 0.59 and 1.39 μM in Pheo A and Hoechst 33342 assays respectively.
CSN13172	Ko 143	461054-93-3	Ko 143 is a practical breast cancer resistance protein multidrug transporter inhibitor BCRP, with the EC90 value of 26 nM.
CSN21978	Glafenine hydrochloride	65513-72-6	Glafenine hydrochloride is a non-narcotic analgesic and non-steroidal anti-inflammatory drug and an ABCG2 inhibitor with an IC50 of 3.2 μM.