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Bombesin Receptor

Bombesin Receptor

货号 产品名 CAS号 信息
CSN21385 PD176252 204067-01-6 PD176252 is a potent antagonist of neuromedin-B preferring (BB1) and gastrin-releasing peptide-preferring (BB2) receptor with Kis of 0.17 nM and 1 nM for human BB1 and BB2 receptors, and 0.66 nM, 16 nM for Rat BB1 and BB2 receptors, respectively; also an agonist of N-Formyl peptide receptor1/2 (FPR1/FPR2), with EC50s of 0.31 and 0.66 μM in HL-60 cells.
CSN24208 ML-18 1422269-30-4 ML-18 is a nonpeptide BRS-3 antagonist with IC50 value of 4.8μM.
CSN17401 MK-5046 1022152-70-0 MK-5046 is a BRS-3 agonist, binds to BRS-3 with high affinity (mouse Ki = 1.6 nM, human Ki = 25 nM).
CSN21526 Bombesin 31362-50-2 Bombesin, a tetradecapeptide originally isolated from frog skin, has an important role in the release of gastrin and the activation of G-protein receptors.
CSN24640 BA 1 183241-31-8 BA 1 is a specific agonist of bombesin receptor with IC50 values of 0.26, 1.55 and 2.52 nM for BB1, BB2 and BB3 respectively. It can enhance glucose transport in obese and diabetic primary myocytes.
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