优势价格
快速发货
品质保证
技术支持
400-920-2911 sales@csnpharm.cn
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN19878 | 20(R)-Ginsenoside Rh2 | 112246-15-8 | 20(R)-Ginsenoside Rh2 has anticancer effects and can increase inchoate apoptotic rate, reduce apoptotic rate significantly, enhance the activity of caspase-3 and induces apoptosis in human lung adenocarcinoma A549 cells. It is a natural product isolated and purified from the roots of Panax ginseng C. A. Mey.. |
| CSN19872 | 3-Hydroxy-2,9,10-trimethoxy-5,6-dihydroisoquinolino[3,2-a]isoquinolin-7-ium chloride | 6681-15-8 | Jatrorrhizine HCl is a protoberberine alkaloid isolated from some plant species like Enantia chlorantha. It can inhibit MAO-A and MAO-B noncompetitively with IC50 value of 4μM and 62μM, respectively. Also, it has antiinflammatory, antimicrobial and antifungal activity. |
| CSN19926 | Irigenin | 548-76-5 | Irigenin is a naturally occuring O-methylated isoflavone. |
| CSN19860 | 5-Hydroxy-2-methylnaphthalene-1,4-dione | 481-42-5 | Plumbagin is an anticancer agent, induces G2/M cell cycle arrest and apoptosis in A549 cells through JNK-dependent p53 Ser15 phosphorylation and inhibits A549 and MDA-MD-231 tumour xenograft growth in nude mice. |
| CSN20001 | Thiolutin | 87-11-6 | Thiolutin is an antibiotic which inhibits bacterial RNA polymerase. Inhibits adhesion of HUVEC cells to vitronectin (IC50 = 0.83 mM) and subsequently reduces paxillin levels. Thiolutin also suppresses tumor cell-induced angiogenesis. |
| CSN19954 | Cyasterone | 17086-76-9 | Cyasterone is an inhibitor of EGFR that maybe a promising anti-cancer agent espcially in skin carcinoma. |
| CSN19857 | KB SRC 4 | 1380088-03-8 | KB SRC 4 is a potent and selective c-Src inhibitor (Ki = 44 nM) and does not inhibit c-Abl at concentrations up to 125 μM. |
| CSN19822 | RSM-932A | 850807-63-5 | RSM-932A is an anticancer drug targeting the human choline kinase alpha, an enzyme involved in increased lipid metabolism of cancer cells. |
| CSN19821 | Maytansine | 35846-53-8 | Maitansine is a cytotoxic agent. It inhibits the assembly of microtubules by binding to tubulin at the rhizoxin binding site. |
| CSN20037 | SGD-1882 | 1222490-34-7 | Pyrrolobenzodiazepine dimer (PDB dimer) is a DNA crosslinking agent that inhibits DNA synthesis. |
| CSN20168 | (±)-Zanubrutinib | 1633350-06-7 | BGB-3111 is a potent, selective and orally available Bruton's tyrosine kinase (Btk) inhibitor. |
| CSN20017 | NVS-PAK1-1 | 1783816-74-9 | NVS-PAK1-1 is a potent allosteric inhibitor of p21-activated kinase PAK1, a serine-threonine kinase that is upregulated in many cancers. NVS-PAK1-1 has an IC50 value of 5 nM for dephoshorylated PAK1 and 6 nM for phosphorylated PAK1 in an in vitro dephosphorylation assay. |
| CSN20042 | DM4 | 796073-69-3 | Maytansinoid DM4 is a tubulin inhibitor, inhibits the assemblyof microtubules by binding to tubulin, with a linker structure can create an antibody-drug conjugate (ADC). |
| CSN20156 | Pyrotinib dimaleate | 1397922-61-0 | Pyrotinib maleate is an irreversible pan-ErbB receptor tyrosine kinase inhibitor, in patients with HER2-Positive metastatic breast cancer. |
| CSN20035 | Tubulysin B | 205304-87-6 | Tubulysin B is a myxobacterial product that can function as an antiangiogenic agent in many in vitro assays with anti-microtubule, anti-mitotic, an apoptosis inducer, anticancer, anti-angiogenic, and antiproliferative activity. |
| CSN20045 | Duocarmycin A | 118292-34-5 | Duocarmycin A is a DNA alkylator agent belonging to duocarmycins family that inhibits DNA synthesis. |
| CSN20036 | (-)-Irofulven | 158440-71-2 | Irofulven is a DNA alkylator agent that inhibits DNA synthesis. |
| CSN20048 | Rachelmycin | 69866-21-3 | CC-1065 is a DNA alkylator agent belonging to duocarmycins family that inhibits DNA synthesis. |
| CSN19868 | Chelerythrine | 34316-15-9 | Chelerythrine, a natural product isolated and purified from the herbs of Chelidonium majus with potent antimanic, antiproliferatvie and antitumor effect, can inhibit telomerase activity, and is a well-known protein kinase C inhibitor. |
| CSN20016 | Coralyne | 6872-73-7 | Coralyne is a cytotoxic agent trageting topoisoerase I, used in combinational chemotherapy to improve the effectiveness in combating proliferation of cancer cells. |
| CSN20180 | PD184161 | 212631-67-9 | PD184161 is an orally-active MEK inhibitor with antitumor effects in HCC in vitro and in vivo that appear to correlate with suppression of MEK activity. |
| CSN20011 | Theliatinib | 1353644-70-8 | Theliatinib, is a small molecule, epidermal growth factor receptor tyrosine kinase inhibitor with potential antineoplastic and anti-angiogenesis activities. |
| CSN20012 | FGFR4 Inhibitor C(-)-11 | 2020395-38-2 | FGFR4 inhibitor C(-)-11 is a highly potent FGFR4 inhibitor with selectivity over FGFR1 with good stability and CYP inhibition. |
| CSN20027 | Sirtuin Inhibitor C18 | 1392810-44-4 | Sirtuin inhibitor C18 is a histone deacetylase class III inhibitor of sirtuin 1 and 2 exerting antiproliferative activity against cancer cell lines. |
| CSN20000 | Neladenoson dalanate | 1239309-58-0 | Neladenoson dalanate is a potent and selective adenosine A1 receptor agonist, and potentially useful for treatment of cardiovascular diseases. |
| CSN20054 | DM1-SMe | 138148-68-2 | DM1-SMe is a tubulin inhibitor, inhibits the assemblyof microtubules by binding to tubulin, with a linker structure can create an antibody-drug conjugate (ADC). |
| CSN20040 | Esperamicin A1 | 99674-26-7 | Esperamicin A1 is a DNA crosslinking agent that inhibits DNA synthesis. |
| CSN20041 | DM3 | 796073-54-6 | DM3 is a tubulin inhibitor, inhibits the assemblyof microtubules by binding to tubulin, with a linker structure can create an antibody-drug conjugate (ADC). |
| CSN20043 | DM3-SMe | 796073-70-6 | DM3-SMe is a tubulin inhibitor, inhibits the assemblyof microtubules by binding to tubulin, with a linker structure can create an antibody-drug conjugate (ADC). |
| CSN20053 | Sabarubicin | 211100-13-9 | Sabarubicin is a Top II inhibitor with anticancer activity. |
| CSN20038 | Thailanstatin A | 1426953-21-0 | Thailanstatin A is a spliceosome inhibitor that disrupts cancer by inhibiting DNA-editing machinery. |
| CSN20044 | DM4-SMe | 796073-68-2 | DM4-Me is a tubulin inhibitor, inhibits the assemblyof microtubules by binding to tubulin, with a linker structure can create an antibody-drug conjugate (ADC). |
| CSN20039 | Tubulysin M | 936691-46-2 | Tubulysin M is a myxobacterial product that can function as an antiangiogenic agent in many in vitro assays with anti-microtubule, anti-mitotic, an apoptosis inducer, anticancer, anti-angiogenic, and antiproliferative activity. |
| CSN20155 | XIAP/cIAP1 antagonist-1 | 1403898-55-4 | AT-IAP is a potent, orally bioavailable, dual antagonist of XIAP and cIAP1 which is functioning in anti-apoptotic and pro-survival signaling pathways. |
| CSN20046 | Duocarmycin MA | 1613286-57-9 | Seco-duocarmycin MA is a DNA alkylator agent belonging to duocarmycins family that inhibits DNA synthesis. |
| CSN20165 | GDC-0425 | 1200129-48-1 | GDC-0425 is an oral, selective Chk1 inhibitor. GDC-0425 enhances gemcitabine (gem) efficacy in tumor xenograft models, and shows greater chemopotentiation in cancer cell lines lacking p53 activity. |
| CSN20047 | Seco-Duocarmycin SA | 144667-38-9 | Seco-duocarmycin SA is a DNA alkylator agent belonging to duocarmycins family that inhibits DNA synthesis. |
| CSN20166 | SU11652 | 326914-10-7 | SU11652 is a sunitinib analog with anti-tyrosine-kinase activity, also is identified as a potential inhibitor for Leishmania major (Lm) nucleoside diphosphate kinases NDK and structural studies indicated that this molecule binds to the active site of LmNDK in a similar conformation to nucleotides, mimicking natural substrates. |
| CSN20049 | Duocarmycin SA | 130288-24-3 | Duocarmycin SA is a DNA alkylator agent belonging to duocarmycins family that inhibits DNA synthesis. |
| CSN20159 | SC-43 | 1400989-25-4 | SC-43 is an src-homology protein tyrosine phosphatase-1 (SHP-1) agonist which reduces liver fibrosis. |
| CSN20051 | Duocarmycin MB | 1613286-58-0 | Seco-duocarmycin MB is a DNA alkylator agent belonging to duocarmycins family that inhibits DNA synthesis. |
| CSN20162 | CAM4066 | 2101206-81-7 | CAM4066 is a selective Casein Kinase 2α (CK2α) inhibitor. |
| CSN20052 | Seco-Duocarmycin TM | 236102-87-7 | Seco-duocarmycin TM is a DNA alkylator agent belonging to duocarmycins family that inhibits DNA synthesis. |
| CSN20163 | Tegatrabetan | 1227637-23-1 | beta-Catenin inhibitor BC2059 is efficacious as monotherapy or in combination with proteasome inhibitor bortezomib in multiple myeloma. |
| CSN20172 | EML-631 | 2101206-36-2 | EML631 interacts with the Tudor-domain-containing protein Spindlin1 (SPIN1), blocking its ability to 'read' H3K4me3 marks and inhibit its transcriptional-coactivator activity. |
| CSN20164 | PP2A-β-Catenin Inhibitor CS-11 | N/A | PP2A-β-Catenin inhibitor CS-11 a small molecule inhibitor of PP2A-β-catenin signaling that limits both in vivo tumor growth and metastasis. |
