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Cannabinoid Receptor
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN25626 | TM38837 | 1253641-65-4 | TM38837 is a novel, largely peripherally restricted CB1 antagonist with limited penetrance to the brain. Oral dose of TM38837 (100 mg/kg) induced a significant increase in freezing behavior. |
| CSN18972 | Taranabant (1R,2R)stereoisomer | 701977-08-4 | Taranabant(1R,2R)stereoisomer is the R-Enantiomer of taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist. |
| CSN19427 | Rimonabant | 168273-06-1 | Rimonabant is a selective central cannabinoid (CB1) receptor inverse agonist with Ki of 1.8 nM. |
| CSN10030 | Rimonabant HCl | 158681-13-1 | Rimonabant HCl is a selective central cannabinoid (CB1) receptor inverse agonist with Ki of 1.8 nM. |
| CSN13721 | Org 27569 | 868273-06-7 | Org 27569 is an allosteric modulator of cannabinoid CB1 receptor, induces a CB1 receptor state that is characterized by enhanced agonist affinity and decreased inverse agonist affinity. |
| CSN13453 | MDA 19 | 1048973-47-2 | MDA 19 is a selective human CB2 receptor agonist with Ki of 43.3 nM. |
| CSN25339 | MAFP | 188404-10-6 | MAFP is a potent, irreversible inhibitor of fatty acid amide hydrolase (FAAH, anandamide amidase), the enzyme responsible for anandamide hydrolysis (IC50 = 2.5 nM). MAFP also binds irreversibly to CB1 receptors with IC50 of 20 nM. |
| CSN19472 | LY320135 | 176977-56-3 | LY-320135 is a potent and selective Canniboid CB1 receptor antagonist/inverse agonist. LY-320135 is selective (~70 fold) over Canniboid CB2 receptors. This compound shows weak binding to both 5-HT2 (Ki = 6.4 μM) and muscarinic receptors (Ki = 2.1 μM). |
| CSN21228 | CB2R-IN-1 | 1257555-79-5 | CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 0.9 nM. |
| CSN10473 | BML-190 | 2854-32-2 | BML-190 is a selective cannabinoid CB2 receptor inverse agonist with Ki of 435 nM, with 50-fold selectivity over CB1 receptor. |
| CSN10421 | beta-Amyrin | 559-70-6 | beta-Amyrin, a natural cannabinoid receptors agonist isolated and purified from the stem bark of Alstonia boonei, has anti-inflammatory activity. Beta-Amyrin significantly inhibits PGE2, IL-6 secretion, and NF-κB activation in a concentration-dependent manner on LPS-induced hPBMCs. |
| CSN15642 | beta-Amyrin Acetate | 1616-93-9 | beta-Amyrin acetrate, a natural cannabinoid receptor isolated and purified from the herbs of Alstonia boone, shows significant HMG-CoA-reductase and sEH inhibitory activities. |
| CSN25672 | Arvanil | 128007-31-8 | Arvanil is an antagonist of cannabinoid CB1 and vanilloid TRPV1 (VR1) with Ki values are 0.5 and 0.3 μM respectively. |
| CSN12849 | AM630 | 164178-33-0 | AM630 is a selectivity CB2 antagonist with Ki of 31.2 nM with a > 150 fold selectivity over CB1 receptor. |
| CSN10272 | AM251 | 183232-66-8 | AM251 is a potent CB1 receptor antagonist (IC50 = 8 nM, Ki = 7.49 nM) that displays 306-fold selectivity over CB2 receptors and also a potent GPR55 agonist (EC50 = 39 nM). |
| CSN21999 | (±)-SLV319 | 362519-49-1 | (±)-SLV319 is a selective antagonist of cannabinoid-1 (CB1) receptor with Ki value of 7.8 nM and it has a weaker activation effect on CB2. |
| CSN12783 | (-)-Gallocatechin | 3371-27-5 | (-)-Gallocatechin, a natural product isolated and purified from the wood of Acacia catechu (L.F.) Willd., has moderate affinity to the human cannabinoid receptor. |
| CSN15641 | (+)-Gallocatechin | 970-73-0 | (+)-Gallocatechin, a natural product isolated and purified from the wood of Acacia catechu (L.F.) Willd., has moderate affinity to the human cannabinoid receptor. |
