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Cannabinoid Receptor
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN21516 | β-Caryophyllene | 87-44-5 | β-Caryophyllene is an agonist of the cannabinoid (CB) receptor CB2 with Ki of 155 nM. |
| CSN12586 | WIN 55,212-2 Mesylate | 131543-23-2 | WIN 55212-2 mesylate is a potent aminoalkylindole cannabinoid (CB) receptor agonist with a Ki of 62.3 and 3.3 nM for human recombinant CB1 and CB2 receptors, respectively. |
| CSN25682 | (5Z,8Z,11Z,14Z)-N-(4-Hydroxy-2-methylphenyl)icosa-5,8,11,14-tetraenamide | 313998-81-1 | VDM 11 is a selective inhibitor of the anandamide membrane transporter (AMT) with IC50 values of 4 - 11 μM. |
| CSN25626 | TM38837 | 1253641-65-4 | TM38837 is a novel, largely peripherally restricted CB1 antagonist with limited penetrance to the brain. Oral dose of TM38837 (100 mg/kg) induced a significant increase in freezing behavior. |
| CSN18972 | Taranabant ((1R,2R)stereoisomer) | 701977-08-4 | Taranabant(1R,2R)stereoisomer is the R-Enantiomer of taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist. |
| CSN12382 | Taranabant | 701977-09-5 | Taranabant is a cannabinoid 1 receptor inverse agonist with IC50 of 0.3 nM. |
| CSN19427 | Rimonabant | 168273-06-1 | Rimonabant is a selective central cannabinoid (CB1) receptor inverse agonist with Ki of 1.8 nM. |
| CSN10030 | Rimonabant Hydrochloride | 158681-13-1 | Rimonabant HCl is a selective central cannabinoid (CB1) receptor inverse agonist with Ki of 1.8 nM. |
| CSN24663 | PF 514273 | 851728-60-4 | PF 514273 is a selective CB1 receptor antagonist with Ki values of 1 and > 10000 nM at CB1 and CB2 receptors respectively. |
| CSN18394 | Otenabant | 686344-29-6 | Otenabant is a selective, potent and competitive CB1 receptor antagonist with Ki of 0.7 nM. |
| CSN16613 | Otenabant Hydrochloride | 686347-12-6 | Otenabant HCl is a recently discovered selective, high affinity, competitive CB1 receptor antagonist with Ki of 0.7 nM. |
| CSN13721 | Org 27569 | 868273-06-7 | Org 27569 is an allosteric modulator of cannabinoid CB1 receptor, induces a CB1 receptor state that is characterized by enhanced agonist affinity and decreased inverse agonist affinity. |
| CSN24683 | OMDM-2 | 616884-63-0 | OMDM-2 is a stable and selective inhibitor of anandamide cellular uptake with Ki of 3 μM. |
| CSN25339 | MAFP | 188404-10-6 | MAFP is a potent, irreversible inhibitor of fatty acid amide hydrolase (FAAH, anandamide amidase), the enzyme responsible for anandamide hydrolysis (IC50 = 2.5 nM). MAFP also binds irreversibly to CB1 receptors with IC50 of 20 nM. |
| CSN19472 | LY320135 | 176977-56-3 | LY-320135 is a potent and selective Canniboid CB1 receptor antagonist/inverse agonist. LY-320135 is selective (~70 fold) over Canniboid CB2 receptors. This compound shows weak binding to both 5-HT2 (Ki = 6.4 μM) and muscarinic receptors (Ki = 2.1 μM). |
| CSN24685 | Leelamine hydrochloride | 16496-99-4 | Leelamine hydrochloride is an agonist of cannabinoid Receptor 1 (CB1). |
| CSN24684 | JTE-907 | 282089-49-0 | JTE 907 is a highly selective cannabinoid CB2 receptor inverse agonist that binds with high affinity to rat, mouse and human CB2 receptors with Ki of 0.38, 1.55 and 35.9 nM respectively. |
| CSN20218 | JD-5037 | 1392116-14-1 | JD-5037 is a peripherally restricted CB1R antagonist with an IC50 of 1.5 nM. |
| CSN19173 | GW842166X | 666260-75-9 | GW842166X is a potent and highly selective agonist of cannabinoid receptor CB2 receptor with EC50 of 63 nM, shows no significant activity at CB1 receptor. |
| CSN21228 | CB2R-IN-1 | 1257555-79-5 | CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 0.9 nM. |
| CSN20330 | CB2 Agonist C8 | 2052602-31-8 | CB2 agonist C8 is an agonists of cannabinoid receptor type 2. |
| CSN20331 | CB2 Agonist C36 | 2097512-96-2 | CB2 agonist C36 is an agonists of cannabinoid receptor type 2. |
| CSN17330 | CB1-IN-1 | 1429239-98-4 | CB1-IN-1 is a peripherally restricted CB1R antagonist, with Ki of 0.3 nM and 21 nM for CB1R (EC50 = 3 nM) and CB2R, respectively. |
| CSN10473 | BML-190 | 2854-32-2 | BML-190 is a selective cannabinoid CB2 receptor inverse agonist with Ki of 435 nM, with 50-fold selectivity over CB1 receptor. |
| CSN10421 | β-Amyrin | 559-70-6 | beta-Amyrin, a natural cannabinoid receptors agonist isolated and purified from the stem bark of Alstonia boonei, has anti-inflammatory activity. Beta-Amyrin significantly inhibits PGE2, IL-6 secretion, and NF-κB activation in a concentration-dependent manner on LPS-induced hPBMCs. |
| CSN15642 | β-Amyrin acetate | 1616-93-9 | beta-Amyrin acetrate, a natural cannabinoid receptor isolated and purified from the herbs of Alstonia boone, shows significant HMG-CoA-reductase and sEH inhibitory activities. |
| CSN18739 | Bay 59-3074 | 406205-74-1 | Bay 59-3074 is a selective CB1/CB2 receptor partial agonist with Kis of 48.3 and 45.5 nM at human CB1 and CB2 receptors respectively . |
| CSN25672 | Arvanil | 128007-31-8 | Arvanil is an antagonist of cannabinoid CB1 and vanilloid TRPV1 (VR1) with Ki values are 0.5 and 0.3 μM respectively. |
| CSN12849 | 6-Iodopravadoline | 164178-33-0 | AM630 is a selectivity CB2 antagonist with Ki of 31.2 nM with a > 150 fold selectivity over CB1 receptor. |
| CSN24665 | CB1 antagonist 2 | 614726-85-1 | AM 4113 is selective CB1 antagonist with Kd of 0.89 nM. |
| CSN24666 | Arachidonylcyclopropylamide | 229021-64-1 | ACPA is a selective agonist of CB1 with Ki of 2.2 nM. |
| CSN18640 | A-836339 | 959746-77-1 | A-836339 is a cannabinoid CB2 receptor-selective agonist and exhibits high potencies at CB(2) and selectivity over CB(1) receptors. |
| CSN21999 | (±)-Ibipinabant | 362519-49-1 | (±)-SLV319 is a selective antagonist of cannabinoid-1 (CB1) receptor with Ki value of 7.8 nM and it has a weaker activation effect on CB2. |
| CSN24668 | (R)-Methanandamide | 157182-49-5 | (R)-(+)-Methanandamide, the stable anandamide analog, is a selective agonist for the CB1 receptor with Ki values of 20 and 815 nM for CB1 and CB2 receptors respectively. |
| CSN12783 | (-)-Gallocatechin | 3371-27-5 | (-)-Gallocatechin, a natural product isolated and purified from the wood of Acacia catechu (L.F.) Willd., has moderate affinity to the human cannabinoid receptor. |
| CSN15641 | (+)-Gallocatechin | 970-73-0 | (+)-Gallocatechin, a natural product isolated and purified from the wood of Acacia catechu (L.F.) Willd., has moderate affinity to the human cannabinoid receptor. |
