Cannabinoid Receptor

Cannabinoid Receptor
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货号	产品名	CAS号	信息
CSN21516	β-Caryophyllene	87-44-5	β-Caryophyllene is an agonist of the cannabinoid (CB) receptor CB2 with Ki of 155 nM.
CSN25626	TM38837	1253641-65-4	TM38837 is a novel, largely peripherally restricted CB1 antagonist with limited penetrance to the brain. Oral dose of TM38837 (100 mg/kg) induced a significant increase in freezing behavior.
CSN18972	Taranabant (1R,2R)stereoisomer	701977-08-4	Taranabant(1R,2R)stereoisomer is the R-Enantiomer of taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist.
CSN24661	RVD-Hpα	1193362-76-3	RVD-Hpα is a N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist and positive CB2 allosteric modulator (Ki = 50 nM). It can increase intracellular Ca2+ levels in cells expressing CB1 receptors in vitro.
CSN19427	Rimonabant	168273-06-1	Rimonabant is a selective central cannabinoid (CB1) receptor inverse agonist with Ki of 1.8 nM.
CSN10030	Rimonabant HCl	158681-13-1	Rimonabant HCl is a selective central cannabinoid (CB1) receptor inverse agonist with Ki of 1.8 nM.
CSN13721	Org 27569	868273-06-7	Org 27569 is an allosteric modulator of cannabinoid CB1 receptor, induces a CB1 receptor state that is characterized by enhanced agonist affinity and decreased inverse agonist affinity.
CSN13453	MDA 19	1048973-47-2	MDA 19 is a selective human CB2 receptor agonist with Ki of 43.3 nM.
CSN25339	MAFP	188404-10-6	MAFP is a potent, irreversible inhibitor of fatty acid amide hydrolase (FAAH, anandamide amidase), the enzyme responsible for anandamide hydrolysis (IC50 = 2.5 nM). MAFP also binds irreversibly to CB1 receptors with IC50 of 20 nM.
CSN19472	LY320135	176977-56-3	LY-320135 is a potent and selective Canniboid CB1 receptor antagonist/inverse agonist. LY-320135 is selective (~70 fold) over Canniboid CB2 receptors. This compound shows weak binding to both 5-HT2 (Ki = 6.4 μM) and muscarinic receptors (Ki = 2.1 μM).
CSN24685	Leelamine HCl	16496-99-4	Leelamine hydrochloride is an agonist of cannabinoid Receptor 1 (CB1).
CSN24684	JTE 907	282089-49-0	JTE 907 is a highly selective cannabinoid CB2 receptor inverse agonist that binds with high affinity to rat, mouse and human CB2 receptors with Ki of 0.38, 1.55 and 35.9 nM respectively.
CSN24687	Hemopressin (rat)	568588-77-2	Hemopressin can act as a cannabinoid CB1 inverse agonist. It could reduce appetite and block signaling by CB1 receptors but not by other members of family A G protein-coupled receptors (including the closely related CB2 receptors. Hemopressin is an endogenous hypotensive nonapeptide derived from hemoglobin.
CSN24686	Hemopressin (human, mouse)	1314035-51-2	Hemopressin (human, mouse) is a selective CB1 receptor inverse agonist with antinociceptive activity. It is the bioactive endogenous peptide substrate for endopeptidase 24.15 (ep24.15), neurolysin (ep24.16) and ACE with Ki values of 27.76, 3.43 and 1.87 μM respectively.
CSN21228	CB2R-IN-1	1257555-79-5	CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 0.9 nM.
CSN10473	BML-190	2854-32-2	BML-190 is a selective cannabinoid CB2 receptor inverse agonist with Ki of 435 nM, with 50-fold selectivity over CB1 receptor.
CSN10421	beta-Amyrin	559-70-6	beta-Amyrin, a natural cannabinoid receptors agonist isolated and purified from the stem bark of Alstonia boonei, has anti-inflammatory activity. Beta-Amyrin significantly inhibits PGE2, IL-6 secretion, and NF-κB activation in a concentration-dependent manner on LPS-induced hPBMCs.
CSN15642	beta-Amyrin Acetate	1616-93-9	beta-Amyrin acetrate, a natural cannabinoid receptor isolated and purified from the herbs of Alstonia boone, shows significant HMG-CoA-reductase and sEH inhibitory activities.
CSN27633	BAY-38-7271	212188-60-8	BAY 38-7271 is selective agonist of cannabinoid CB1/CB2 receptor with Kis of 1.85 nM and 5.96 nM respectively. It has strong neuroprotective properties.
CSN25672	Arvanil	128007-31-8	Arvanil is an antagonist of cannabinoid CB1 and vanilloid TRPV1 (VR1) with Ki values are 0.5 and 0.3 μM respectively.
CSN12783	(-)-Gallocatechin	3371-27-5	(-)-Gallocatechin, a natural product isolated and purified from the wood of Acacia catechu (L.F.) Willd., has moderate affinity to the human cannabinoid receptor.
CSN15641	(+)-Gallocatechin	970-73-0	(+)-Gallocatechin, a natural product isolated and purified from the wood of Acacia catechu (L.F.) Willd., has moderate affinity to the human cannabinoid receptor.

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