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Cannabinoid Receptor

Cannabinoid Receptor

货号 产品名 CAS号 信息
CSN19427 Rimonabant 168273-06-1 Rimonabant is a selective central cannabinoid (CB1) receptor inverse agonist with Ki of 1.8 nM.
CSN10030 Rimonabant HCl 158681-13-1 Rimonabant HCl is a selective central cannabinoid (CB1) receptor inverse agonist with Ki of 1.8 nM.
CSN13721 Org 27569 868273-06-7 Org 27569 is an allosteric modulator of cannabinoid CB1 receptor, induces a CB1 receptor state that is characterized by enhanced agonist affinity and decreased inverse agonist affinity.
CSN25339 MAFP 188404-10-6 MAFP is a potent, irreversible inhibitor of fatty acid amide hydrolase (FAAH, anandamide amidase), the enzyme responsible for anandamide hydrolysis (IC50 = 2.5 nM). MAFP also binds irreversibly to CB1 receptors with IC50 of 20 nM.
CSN19472 LY320135 176977-56-3 LY-320135 is a potent and selective Canniboid CB1 receptor antagonist/inverse agonist. LY-320135 is selective (~70 fold) over Canniboid CB2 receptors. This compound shows weak binding to both 5-HT2 (Ki = 6.4 μM) and muscarinic receptors (Ki = 2.1 μM).
CSN10473 BML-190 2854-32-2 BML-190 is a selective cannabinoid CB2 receptor inverse agonist with Ki of 435 nM, with 50-fold selectivity over CB1 receptor.
CSN10421 beta-Amyrin 559-70-6 beta-Amyrin, a natural cannabinoid receptors agonist isolated and purified from the stem bark of Alstonia boonei, has anti-inflammatory activity. Beta-Amyrin significantly inhibits PGE2, IL-6 secretion, and NF-κB activation in a concentration-dependent manner on LPS-induced hPBMCs.
CSN15642 beta-Amyrin Acetate 1616-93-9 beta-Amyrin acetrate, a natural cannabinoid receptor isolated and purified from the herbs of Alstonia boone, shows significant HMG-CoA-reductase and sEH inhibitory activities.
CSN18739 BAY 59-3074 406205-74-1 Bay 59-3074 is a selective CB1/CB2 receptor partial agonist with Kis of 48.3 and 45.5 nM at human CB1 and CB2 receptors respectively .
CSN25672 Arvanil 128007-31-8 Arvanil is an antagonist of cannabinoid CB1 and vanilloid TRPV1 (VR1) with Ki values are 0.5 and 0.3 μM respectively.
CSN21999 (±)-SLV319 362519-49-1 (±)-SLV319 is a selective antagonist of cannabinoid-1 (CB1) receptor with Ki value of 7.8 nM and it has a weaker activation effect on CB2.
CSN12783 (-)-Gallocatechin 3371-27-5 (-)-Gallocatechin, a natural product isolated and purified from the wood of Acacia catechu (L.F.) Willd., has moderate affinity to the human cannabinoid receptor.
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