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Cannabinoid Receptor
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN21516 | β-Caryophyllene | 87-44-5 | β-Caryophyllene is an agonist of the cannabinoid (CB) receptor CB2 with Ki of 155 nM. |
| CSN18972 | Taranabant (1R,2R)stereoisomer | 701977-08-4 | Taranabant(1R,2R)stereoisomer is the R-Enantiomer of taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist. |
| CSN13721 | Org 27569 | 868273-06-7 | Org 27569 is an allosteric modulator of cannabinoid CB1 receptor, induces a CB1 receptor state that is characterized by enhanced agonist affinity and decreased inverse agonist affinity. |
| CSN25339 | MAFP | 188404-10-6 | MAFP is a potent, irreversible inhibitor of fatty acid amide hydrolase (FAAH, anandamide amidase), the enzyme responsible for anandamide hydrolysis (IC50 = 2.5 nM). MAFP also binds irreversibly to CB1 receptors with IC50 of 20 nM. |
| CSN19472 | LY320135 | 176977-56-3 | LY-320135 is a potent and selective Canniboid CB1 receptor antagonist/inverse agonist. LY-320135 is selective (~70 fold) over Canniboid CB2 receptors. This compound shows weak binding to both 5-HT2 (Ki = 6.4 μM) and muscarinic receptors (Ki = 2.1 μM). |
| CSN24684 | JTE 907 | 282089-49-0 | JTE 907 is a highly selective cannabinoid CB2 receptor inverse agonist that binds with high affinity to rat, mouse and human CB2 receptors with Ki of 0.38, 1.55 and 35.9 nM respectively. |
| CSN21228 | CB2R-IN-1 | 1257555-79-5 | CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 0.9 nM. |
| CSN10473 | BML-190 | 2854-32-2 | BML-190 is a selective cannabinoid CB2 receptor inverse agonist with Ki of 435 nM, with 50-fold selectivity over CB1 receptor. |
| CSN10421 | beta-Amyrin | 559-70-6 | beta-Amyrin, a natural cannabinoid receptors agonist isolated and purified from the stem bark of Alstonia boonei, has anti-inflammatory activity. Beta-Amyrin significantly inhibits PGE2, IL-6 secretion, and NF-κB activation in a concentration-dependent manner on LPS-induced hPBMCs. |
| CSN15642 | beta-Amyrin Acetate | 1616-93-9 | beta-Amyrin acetrate, a natural cannabinoid receptor isolated and purified from the herbs of Alstonia boone, shows significant HMG-CoA-reductase and sEH inhibitory activities. |
| CSN12783 | (-)-Gallocatechin | 3371-27-5 | (-)-Gallocatechin, a natural product isolated and purified from the wood of Acacia catechu (L.F.) Willd., has moderate affinity to the human cannabinoid receptor. |
| CSN15641 | (+)-Gallocatechin | 970-73-0 | (+)-Gallocatechin, a natural product isolated and purified from the wood of Acacia catechu (L.F.) Willd., has moderate affinity to the human cannabinoid receptor. |
