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Cannabinoid Receptor

Cannabinoid Receptor

货号 产品名 CAS号 信息
CSN21516 β-Caryophyllene 87-44-5 β-Caryophyllene is an agonist of the cannabinoid (CB) receptor CB2 with Ki of 155 nM.
CSN25626 TM38837 1253641-65-4 TM38837 is a novel, largely peripherally restricted CB1 antagonist with limited penetrance to the brain. Oral dose of TM38837 (100 mg/kg) induced a significant increase in freezing behavior.
CSN18972 Taranabant (1R,2R)stereoisomer 701977-08-4 Taranabant(1R,2R)stereoisomer is the R-Enantiomer of taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist.
CSN24661 RVD-Hpα 1193362-76-3 RVD-Hpα is a N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist and positive CB2 allosteric modulator (Ki = 50 nM). It can increase intracellular Ca2+ levels in cells expressing CB1 receptors in vitro.
CSN19427 Rimonabant 168273-06-1 Rimonabant is a selective central cannabinoid (CB1) receptor inverse agonist with Ki of 1.8 nM.
CSN10030 Rimonabant HCl 158681-13-1 Rimonabant HCl is a selective central cannabinoid (CB1) receptor inverse agonist with Ki of 1.8 nM.
CSN13721 Org 27569 868273-06-7 Org 27569 is an allosteric modulator of cannabinoid CB1 receptor, induces a CB1 receptor state that is characterized by enhanced agonist affinity and decreased inverse agonist affinity.
CSN13453 MDA 19 1048973-47-2 MDA 19 is a selective human CB2 receptor agonist with Ki of 43.3 nM.
CSN25339 MAFP 188404-10-6 MAFP is a potent, irreversible inhibitor of fatty acid amide hydrolase (FAAH, anandamide amidase), the enzyme responsible for anandamide hydrolysis (IC50 = 2.5 nM). MAFP also binds irreversibly to CB1 receptors with IC50 of 20 nM.
CSN19472 LY320135 176977-56-3 LY-320135 is a potent and selective Canniboid CB1 receptor antagonist/inverse agonist. LY-320135 is selective (~70 fold) over Canniboid CB2 receptors. This compound shows weak binding to both 5-HT2 (Ki = 6.4 μM) and muscarinic receptors (Ki = 2.1 μM).
CSN24685 Leelamine HCl 16496-99-4 Leelamine hydrochloride is an agonist of cannabinoid Receptor 1 (CB1).
CSN24684 JTE 907 282089-49-0 JTE 907 is a highly selective cannabinoid CB2 receptor inverse agonist that binds with high affinity to rat, mouse and human CB2 receptors with Ki of 0.38, 1.55 and 35.9 nM respectively.
CSN24687 Hemopressin (rat) 568588-77-2 Hemopressin can act as a cannabinoid CB1 inverse agonist. It could reduce appetite and block signaling by CB1 receptors but not by other members of family A G protein-coupled receptors (including the closely related CB2 receptors. Hemopressin is an endogenous hypotensive nonapeptide derived from hemoglobin.
CSN24686 Hemopressin (human, mouse) 1314035-51-2 Hemopressin (human, mouse) is a selective CB1 receptor inverse agonist with antinociceptive activity. It is the bioactive endogenous peptide substrate for endopeptidase 24.15 (ep24.15), neurolysin (ep24.16) and ACE with Ki values of 27.76, 3.43 and 1.87 μM respectively.
CSN21228 CB2R-IN-1 1257555-79-5 CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 0.9 nM.
CSN10473 BML-190 2854-32-2 BML-190 is a selective cannabinoid CB2 receptor inverse agonist with Ki of 435 nM, with 50-fold selectivity over CB1 receptor.
CSN10421 beta-Amyrin 559-70-6 beta-Amyrin, a natural cannabinoid receptors agonist isolated and purified from the stem bark of Alstonia boonei, has anti-inflammatory activity. Beta-Amyrin significantly inhibits PGE2, IL-6 secretion, and NF-κB activation in a concentration-dependent manner on LPS-induced hPBMCs.
CSN15642 beta-Amyrin Acetate 1616-93-9 beta-Amyrin acetrate, a natural cannabinoid receptor isolated and purified from the herbs of Alstonia boone, shows significant HMG-CoA-reductase and sEH inhibitory activities.
CSN27633 BAY-38-7271 212188-60-8 BAY 38-7271 is selective agonist of cannabinoid CB1/CB2 receptor with Kis of 1.85 nM and 5.96 nM respectively. It has strong neuroprotective properties.
CSN25672 Arvanil 128007-31-8 Arvanil is an antagonist of cannabinoid CB1 and vanilloid TRPV1 (VR1) with Ki values are 0.5 and 0.3 μM respectively.
CSN12783 (-)-Gallocatechin 3371-27-5 (-)-Gallocatechin, a natural product isolated and purified from the wood of Acacia catechu (L.F.) Willd., has moderate affinity to the human cannabinoid receptor.
CSN15641 (+)-Gallocatechin 970-73-0 (+)-Gallocatechin, a natural product isolated and purified from the wood of Acacia catechu (L.F.) Willd., has moderate affinity to the human cannabinoid receptor.
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