| CSN21291 |
ML171
|
6631-94-3 |
ML171 is a novel and selective NOX1 inhibitor with IC50 value of 0.25 μM for blocking NOX1-dependent ROS generation in a HEK293-NOX1 recombinant cell system. |
| CSN21155 |
L-NMMA Acetate
|
53308-83-1 |
L-NMMA acetate is a nitric oxide synthase inhibitor of all NOS isoforms including NOS1, NOS2, and NOS3. The Ki values for nNOS (rat), eNOS (human), and iNOS (mouse) are approximately 0.18, 0.4, and 6 µM, respectively. |
| CSN21258 |
Tecadenoson
|
204512-90-3 |
Tecadenoson is a selective A1 adenosine receptor agonist. |
| CSN21296 |
AGN 192836
|
171102-29-7 |
AGN 192836 is a potent and selective α2 adrenergic agonist with EC50s of 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor, respectively. |
| CSN22330 |
RP 54275
|
81364-78-5 |
2-Octadecyl-1H-indole-5-carboxylic acid is a novel hypocholesterolaemic drug. |
| CSN22149 |
Prolylleucine
|
61596-47-2 |
Prolylleucine is a dipeptide containing branched-chain amino acids. |
| CSN22110 |
Bepridil HCl
|
68099-86-5 |
Bepridil HCl is a calcium channel blocker, with antianginal activity. |
| CSN22159 |
ICI 153110
|
87164-90-7 |
ICI 153110 is an orally active phosphodiesterase inhibitor with both vasodilating and inotropic properties which is designed for the treatment of congestive cardiac failure. |
| CSN21356 |
S107 HCl
|
1357476-46-0 |
S107 HCl is a RyR-selective 1,4-benzothiazepine derivative that stabilizes RyR2 channels by enhancing the binding affinity of calstabin2 to mutant and/or PKA-phosphorylated channels. |
| CSN22181 |
OM-189
|
55381-18-5 |
OM-189 is a selective synthetic thrombin inhibitor. |
| CSN22174 |
CE-245677
|
717899-97-3 |
CE-245677 is a potent reversible inhibitor of Tie2 and TrkA/B kinases with a cellular IC50s of 4.7 and 1 nM. |
| CSN22154 |
F 16915
|
92510-91-3 |
F 16915 is a docosahexaenoic acid derivative which can prevent heart failure-induced atrial fibrillation. |
| CSN22168 |
FKK
|
78299-79-3 |
FKK is an indazole derivative and also a novel bronchodilator. |
| CSN22235 |
Almokalant
|
123955-10-2 |
Almokalant is a class III antiarrhythmic drug, acts as a potassium channel blocker, and inhibits a specific component (Ikr) of the time-dependent delayed rectifier K+ current. |
| CSN22444 |
L-765314
|
189349-50-6 |
L-765314 is a potent and selective α1b adrenergic receptor antagonist with Kis of 5.4±0.6 nM and 2.0±0.66 nM for rat and human α1b adrenergic receptor, respectively. |
| CSN22536 |
ZD-0892
|
171964-73-1 |
ZD-0892 is a selective and potent inhibitor of a neutrophil elastase with Kis of 6.7 and 200 nM for human neutrophil elastase and porcine pancreatic elastase, respectively. |
400-920-2911
上海市杨浦区翔殷路128号1号楼101
