货号 | 产品名 | CAS号 | 信息 |
---|---|---|---|
CSN21291 | ML171 | 6631-94-3 | ML171 is a novel and selective NOX1 inhibitor with IC50 value of 0.25 μM for blocking NOX1-dependent ROS generation in a HEK293-NOX1 recombinant cell system. |
CSN21155 | L-NMMA Acetate | 53308-83-1 | L-NMMA acetate is a nitric oxide synthase inhibitor of all NOS isoforms including NOS1, NOS2, and NOS3. The Ki values for nNOS (rat), eNOS (human), and iNOS (mouse) are approximately 0.18, 0.4, and 6 µM, respectively. |
CSN21258 | Tecadenoson | 204512-90-3 | Tecadenoson is a selective A1 adenosine receptor agonist. |
CSN21296 | AGN 192836 | 171102-29-7 | AGN 192836 is a potent and selective α2 adrenergic agonist with EC50s of 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor, respectively. |
CSN22330 | RP 54275 | 81364-78-5 | 2-Octadecyl-1H-indole-5-carboxylic acid is a novel hypocholesterolaemic drug. |
CSN22149 | Prolylleucine | 61596-47-2 | Prolylleucine is a dipeptide containing branched-chain amino acids. |
CSN22110 | Bepridil HCl | 68099-86-5 | Bepridil HCl is a calcium channel blocker, with antianginal activity. |
CSN22159 | ICI 153110 | 87164-90-7 | ICI 153110 is an orally active phosphodiesterase inhibitor with both vasodilating and inotropic properties which is designed for the treatment of congestive cardiac failure. |
CSN21356 | S107 HCl | 1357476-46-0 | S107 HCl is a RyR-selective 1,4-benzothiazepine derivative that stabilizes RyR2 channels by enhancing the binding affinity of calstabin2 to mutant and/or PKA-phosphorylated channels. |
CSN22181 | OM-189 | 55381-18-5 | OM-189 is a selective synthetic thrombin inhibitor. |
CSN22174 | CE-245677 | 717899-97-3 | CE-245677 is a potent reversible inhibitor of Tie2 and TrkA/B kinases with a cellular IC50s of 4.7 and 1 nM. |
CSN22154 | F 16915 | 92510-91-3 | F 16915 is a docosahexaenoic acid derivative which can prevent heart failure-induced atrial fibrillation. |
CSN22168 | FKK | 78299-79-3 | FKK is an indazole derivative and also a novel bronchodilator. |
CSN22235 | Almokalant | 123955-10-2 | Almokalant is a class III antiarrhythmic drug, acts as a potassium channel blocker, and inhibits a specific component (Ikr) of the time-dependent delayed rectifier K+ current. |
CSN22444 | L-765314 | 189349-50-6 | L-765314 is a potent and selective α1b adrenergic receptor antagonist with Kis of 5.4±0.6 nM and 2.0±0.66 nM for rat and human α1b adrenergic receptor, respectively. |
CSN22536 | ZD-0892 | 171964-73-1 | ZD-0892 is a selective and potent inhibitor of a neutrophil elastase with Kis of 6.7 and 200 nM for human neutrophil elastase and porcine pancreatic elastase, respectively. |