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| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN16069 | IMD-0354 | 978-62-1 | IMD-0354 is a synthetic selective NF-kB inhibitor and blocks IκBα phosphorylation in NF-κB pathway. |
| CSN16093 | Dalcetrapib | 211513-37-0 | Dalcetrapib is a rhCETP inhibitor with IC50 of 0.2 μM. |
| CSN16211 | Sacubitril/Valsartan | 936623-90-4 | LCZ 696 is a mixture of neprilysin inhibitor sacubitril and the angiotensin receptor blocker valsartan in a ratio of 1:1. |
| CSN16408 | Dipyridamole | 58-32-2 | Dipyridamole is a phosphodiesterase inhibitor that blocks uptake and metabolism of adenosine by erythrocytes and vascular endothelial cells. |
| CSN16438 | (S)-1-((S)-3-mercapto-2-methylpropanoyl)pyrrolidine-2-carboxylic acid | 62571-86-2 | Captopril is an angiotensin-converting enzyme (ACE) inhibitor with IC50 of 6 nM. |
| CSN16475 | Ozagrel | 82571-53-7 | Ozagrel is an antiplatelet agent working as a thromboxane A2 synthesis inhibitor. |
| CSN16692 | Eplerenone | 107724-20-9 | Eplerenone is both a selective aldosterone blocker and a CYP3A4 substrate. |
| CSN16785 | (E)-3-(4-((1H-Imidazol-1-yl)methyl)phenyl)acrylic acid hydrochloride | 78712-43-3 | Ozagrel HCl is a selective thromboxane A(2) (TXA(2)) synthetase inhibitor with IC50 of 11 nM for rabbit platelet, used for the improvement of postoperative cerebrovascular contraction and accompanying cerebral ischaemia. |
| CSN16790 | Amlodipine | 88150-42-9 | Amlodipine is a long-acting calcium channel blocker used to lower blood pressure and prevent chest pain. |
| CSN16791 | Amlodipine maleate | 88150-47-4 | Amlodipine Maleate is a long-acting calcium channel blocker. |
| CSN16825 | Selexipag | 475086-01-2 | NS-304 is an agonist of prostacyclin IP1 receptor with Ki of 260 nM. It is used for the treatment of pulmonary arterial hypertension. |
| CSN16917 | AVE 0991 | 304462-19-9 | AVE 0991 is a nonpeptide Ang-(1-7) receptor Mas agonist. |
| CSN17009 | Fosinopril sodium | 88889-14-9 | Fosinopril sodium is a phosphinic acid-containing ester ACE inhibitor used to treat high blood pressure. |
| CSN16090 | UNC2881 | 1493764-08-1 | UNC2881 is a Mer kinase inhibitor and can inhibit the phosphorylation of Mer with IC50 of 4.3 nM. |
| CSN16691 | 2-Methylpropan-2-amine (2S,3aS,7aS)-1-((S)-2-(((S)-1-ethoxy-1-oxopentan-2-yl)amino)propanoyl)octahydro-1H-indole-2-carboxylate | 107133-36-8 | Perindopril erbumine Perindopril is a long-acting ACE inhibitor with IC50 of 1.05 nM, used in treatment for hypertension. |
| CSN16652 | 5-((3,4-Dimethoxyphenethyl)(methyl)amino)-2-(3,4-dimethoxyphenyl)-2-isopropylpentanenitrile hydrochloride | 152-11-4 | Verapamil HCl is a phenylalkylamine class L-type calcium channel blocker. |
| CSN16147 | 1-Butyl-N-(2,6-dimethylphenyl)piperidine-2-carboxamide | 38396-39-3 | Bupivacaine, an amide local anesthetic, reversibly binds to specific sodium ion channels that decreases the stabilization of membrane . |
| CSN16086 | KY02111 | 1118807-13-8 | KY02111 can inhibit Wnt signaling and promote differentiation of hPSCs to cardiomyocytes. |
| CSN16171 | 5-(2-Cyclopropyl-1-(2-fluorophenyl)-2-oxoethyl)-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-2-yl acetate | 150322-43-3 | Prasugrel is a platelet inhibitor with IC50 value of 1.8 μM. |
| CSN17034 | (S)-3-((S)-2-(((S)-1-Ethoxy-1-oxo-4-phenylbutan-2-yl)amino)propanoyl)-1-methyl-2-oxoimidazolidine-4-carboxylic acid hydrochloride | 89396-94-1 | Imidapril HCl is the HCl salt of imidapril, an angiotensin-converting enzyme (ACE) inhibitor with antihypertensive activity. |
| CSN17095 | Nisoldipine | 63675-72-9 | Nisoldipine is a calcium channel blocker belonging to the dihydropyridines class, specific for L-type Cav1.2 with IC50 of 10 nM. |
| CSN16729 | Gliclazide | 21187-98-4 | Gliclazide is a blocker of pancreatic β-cell ATP-sensitive potassium channels with IC50 of 184 nM in murine. It belongs to the sulfonylurea class of insulin secretagoguesIt. Gliclazide is an antihyperglycemic agent used for the treatment of non-insulin-dependent diabetes mellitus (NIDDM). |
| CSN16465 | Enalapril | 75847-73-3 | Enalapril is an angiotensin converting enzyme (ACE) inhibitor. |
| CSN16953 | (S)-4-Fluoro-5-((2-methyl-1,4-diazepan-1-yl)sulfonyl)isoquinoline | 223645-67-8 | K-115, an isoquinolinesulfonamide compound, is a highly selective and potent (IC50 = 31 nM) Rho-kinase inhibitor, and used for treating POAG or ocular hypertension. |
| CSN16473 | Zofenopril Calcium | 81938-43-4 | Zofenopril calcium is sulfhydryl ACE inhibitor with antihypertensive activity. |
| CSN17378 | BMS-687453 | 1000998-59-3 | BMS-687453 is a potent and selective PPARα agonist, with an EC50 of 10 nM for human PPARα and 410-fold selectivity vs human PPARγ in PPAR-GAL4 transactivation assays. |
| CSN16645 | (1S,2S)-2-(2-((3-(1H-Benzo[d]imidazol-2-yl)propyl)(methyl)amino)ethyl)-6-fluoro-1-isopropyl-1,2,3,4-tetrahydronaphthalen-2-yl cyclopropanecarboxylate dihydrochloride | 357400-13-6 | NNC 55-0396, Mibefradil derivative, is a highly selective T-type calcium channel blocker, displaying IC50 values of 6.8 and > 100 μM for inhibition of Cav3.1 T-type channels and HVA currents respectively in INS-1 cells. |
| CSN16320 | GS967 | 1262618-39-2 | GS-967 is a selective inhibitor of cardiac late sodium current (late INa ). The IC50 values in ventricular myocytes and isolated hearts are 0.13 μM and 0.21 μM. |
| CSN16099 | SAR407899 HCl | 923262-96-8 | SAR407899 HCl is a potent, ATP-competitive ROCK inhibitor woth Ki value of 36 nM/41 nM for human ROCK/Rat ROCK respectively. |
| CSN17027 | Fenoldopam | 67227-56-9 | Fenoldopam is a drug and synthetic benzazepine derivative which acts as a selective D1 receptor partial agonist. |
| CSN16760 | 2-(4-((5,6-Diphenylpyrazin-2-yl)(isopropyl)amino)butoxy)acetic acid | 475085-57-5 | MRE-269 can act as an agonist of IP receptor and it is an active metabolite of selexipag. |
| CSN17409 | TPO agonist 1 | 1033040-23-1 | TPO agonist 1 can increase production of platelets by stimulating the TPO receptor in people with chronic ITP. |
| CSN17348 | BQ-788 sodium salt | 156161-89-6 | BQ-788 sodium salt is a potent, selective ETB receptor antagonist with IC50 of 1.2 nM for inhibition of ET-1 binding to human Girardi heart cells, poorly inhibiting the binding to ETA receptors in human neuroblastoma cell line SK-N-MC cells with IC50 of 1300 nM. |
| CSN17393 | VTP-27999 TFA | 1013937-63-7 | VTP-27999 trifluoroacetate is an alkyl amine Renin inhibitor and is useful for Hypertension and End-Organ Diseases. |
| CSN16922 | AVE 0991 sodium salt | 306288-04-0 | AVE 0991 sodium is a nonpeptide Ang-(1-7) receptor Mas agonist, represents an important step for exploration of the effects of Ang-(1-7) and testing of its potential as a cardiovascular drug. |
| CSN16302 | Efonidipine | 111011-63-3 | Efonidipine is a dual T-type and L-type calcium channel blocker (CCB). |
| CSN17076 | Nicainoprol | 76252-06-7 | Nicainoprol is a sodium channels blocker which is used as an antiarrhythmic agent. |
| CSN16272 | XEN445 | 1515856-92-4 | XEN445 is a potent and selective endothelial lipase inhibitor with IC50 of 0.237 μM. |
| CSN16232 | Omecamtiv mecarbil | 873697-71-3 | Omecamtiv mecarbil is a selective sarcomere-directed cardiac myosin activator with an EC50 of 0.6 μM. |
| CSN16875 | PD 123319 ditrifluoroacetate | 136676-91-0 | PD123319 Ditrifluoroacetate is a potent, selective and non-peptide angiotensin AT2 receptor antagonist. |
| CSN16264 | Calcium 4-(((2S,4R)-1-([1,1'-biphenyl]-4-yl)-5-ethoxy-4-methyl-5-oxopentan-2-yl)amino)-4-oxobutanoate | 1369773-39-6 | AHU-377 Hemicalcium is a potent Neprilysin inhibitor with an IC50 of 5 nM. |
| CSN16280 | SEA0400 | 223104-29-8 | SEA0400 is a selective inhibitor of the Na+-Ca2+ exchanger with IC50 of 5-33 nM (inhibiting Na+-dependent Ca2+ uptake in cultured neurons, astrocytes, and microglia). |
| CSN16501 | Trandolapril | 87679-37-6 | Trandolapril is an ACE inhibitor used to treat high blood pressure. |
| CSN16723 | (6R,12aR)-6-(Benzo[d][1,3]dioxol-5-yl)-2-methyl-2,3,12,12a-tetrahydropyrazino[1',2':1,6]pyrido[3,4-b]indole-1,4(6H,7H)-dione | 171596-29-5 | Tadalafil is a PDE5 inhibitor with an IC50 value of 1.8 nM. |
| CSN17090 | Nifekalant HCl | 130656-51-8 | Nifekalant HCl is an antiarrhythmic shown to be effective against ventricular tachyarrhythmias by inhibiting HERG channels in a voltage- and frequency-dependent manner. |
| CSN16080 | GSK 3 Inhibitor IX | 667463-62-9 | BIO is an inhibitor of GSK-3 and CDK1–cyclinB complex. The IC50s of GSK-3αβ, CDK1, CDK5 are 5 nM, 320 nM and 83 nM, respectively. |
