400-920-2911
上海市杨浦区翔殷路128号1号楼101
Chk
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN17165 | PF-477736 | 952021-60-2 | PF-477736 is a selective, potent and ATP-competitive Chk1 inhibitor with Ki of 0.49 nM and also inhibits VEGFR2, Aurora-A, FGFR3, Flt3, Fms (CSF1R), Ret and Yes and shows ~100-fold selectivity for Chk1 than Chk2. |
| CSN23009 | NSC 109555 Ditosylate | 66748-43-4 | NSC 109555 Ditosylate is a selective, reversible, ATP-competitive Chk2 inhibitor with IC50 of 0.2 μM. |
| CSN17600 | LY2606368 2HCl | 1234015-54-3 | LY2606368 (Prexasertib) is a selective Chk1 inhibitor with IC50 value <1nM, modest to Chk2 and Rsk with IC50 values of 8nM and <10nM. |
| CSN16323 | BML-277 | 516480-79-8 | BML-277 is a selective Chk2 (checkpoint kinase 2) inhibitor with IC50 of 15 nM. |