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Dopamine Receptor
货号 | 产品名 | CAS号 | 信息 |
---|---|---|---|
CSN11417 | 10-(3-(4-Methylpiperazin-1-yl)propyl)-2-(trifluoromethyl)-10H-phenothiazine dihydrochloride | 440-17-5 | Trifluoperazine 2HCl is a dopamine D2 receptor inhibitor with anti-dopaminergic and anti-adrenergic actions, which belongs to the phenothiazine compounds. |
CSN21106 | Pimozide | 2062-78-4 | Pimozide is a dopamine receptor antagonist, with Kis of 1.4 nM, 2.5 nM and 588 nM for dopamine D2, D3 and D1 receptors, respectively, and also has affinity at α1-adrenoceptor, with a Ki of 39 nM; also inhibits STAT3 and STAT5. |
CSN10189 | Paliperidone | 144598-75-4 | Paliperidone is a potent serotonin-2A and dopamine-2 receptor antagonist, it is the main active metabolite of risperidone and used in the treatment of schizophrenia. |
CSN10153 | 5-(2-Aminoethyl)benzene-1,2,4-triol hydrobromide | 636-00-0 | Oxidopamine hydrobromide is a selective catecholaminergic neurotoxin, depletes brain catecholamine levels via uptake and accumulation by a transport mechanism specific to these neurons. |
CSN10154 | Oxidopamine HCl | 28094-15-7 | Oxidopamine HCl is a neurotoxic synthetic organic compound, selectively destroys dopaminergic and noradrenergic neurons in the brain. |
CSN11425 | 4-Amino-5-chloro-N-(2-(diethylamino)ethyl)-2-methoxybenzamide | 364-62-5 | Metoclopramide is an antagonist of dopamine D2 and is commonly used as an antiemetic. |
CSN11426 | Metoclopramide HCl | 7232-21-5 | Metoclopramide HCl is a selective dopamine D2 receptor antagonist, used for the treatment of nausea and vomiting. |
CSN11293 | Levosulpiride | 23672-07-3 | Levosulpiride, an atypical antipsychotic, can selectively inhibit D2 receptor and it is the (S)-enantiomer of sulpiride. |
CSN11238 | Itopride | 122898-67-3 | Itopride is a prokinetic benzamide derivative unlike metoclopramide or domperidone, and is indicated for the treatment of functional dyspepsia and other gastrointestinal conditions. |
CSN19483 | GR 103691 | 162408-66-4 | GR 103691 is an effective and selective receptor antagonist of the dopamine D3 receptor (D3DR). |
CSN11042 | Fluphenazine 2HCl | 146-56-5 | Fluphenazine 2HCl is a inhibitor of D1DR and D2DR. It has been used to deliver fluphenazine to biological systems and also used as an antipsychotic. |
CSN10871 | Droperidol | 548-73-2 | Droperidol is an antagonist of dopamine-2 receptor. |
CSN12935 | Domperidone | 57808-66-9 | Domperidone is an antagonist of dopamine D2 receptor and the IC50 value for rat D2 receptor is 13.6 nM. |
CSN10685 | Clozapine | 5786-21-0 | Clozapine, an antipsychotic drug, is antagonist of dopamine and other receptors used to treat schizophrenia with a Ki value of 9.5 nM for M1 receptor. |
CSN10662 | Clebopride malate | 57645-91-7 | Clebopride malate, with antiemetic and prokinetic properties, is a dopamine antagonist drug used to treat gastrointestinal dysfunction. |
CSN17057 | CL-216303 Hydrochloride | 86215-36-3 | CL-216303 HCl is a dopamine transporter inhibitor and a 5-HT inhibitor potentially for the treatment of depression. |
CSN10490 | Bromopride | 4093-35-0 | Bromopride is a dopamine antagonist with prokinetic properties, widely used as an antiemetic. |
CSN10487 | Bromocriptine mesylate | 22260-51-1 | Bromocriptine mesylate is a potent dopamine D2/D3 receptoragonist, which binds D2 dopamine receptor with pKi of 8.05±0.2. |
CSN10446 | Talipexole 2HCl | 36085-73-1 | B-HT 920 is a dopamine D2 receptor agonist, α2-adrenoceptor agonist and 5-HT3 receptor antagonist, which displays antiParkinsonian activity. |
CSN10288 | Amisulpride | 71675-85-9 | Amisulpride is a selective dopamine antagonist wit Ki of 2.8 nM for D2 receptor and Ki of 3.2 nM D3 receptor, it's used as an antipsychotic drug. |
CSN10011 | 1-Adamantanamine HCl | 665-66-7 | Amantadine HCl is an antiviral and an antiparkinsonian drug. It is used to treat or prevent infections of the respiratory tract caused by a certain virus. |
CSN10242 | Alizapride | 59338-93-1 | Alizapride is a dopamine antagonist with prokinetic and antiemetic effects used in the treatment of nausea and vomiting, including postoperative nausea and vomiting. |
CSN10243 | Alizapride HCl | 59338-87-3 | Alizapride HCl is a dopamine receptor antagonist used in the administration of nausea and vomiting. |
CSN10654 | A68930 HCl | 130465-39-3 | A-68930 HCl is a potent and selective D1-like dopamine receptor agonist (EC50 values are 2.1 and 3910 nM for D1-like and D2-like receptors respectively). |
CSN52424 | 6-Chloro-1-(4-hydroxyphenyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepine-7,8-diol methanesulfonate | 67227-57-0 |