Dual Specificity Tyrosine-phosphorylation-regulated Kinase | Protein Tyrosine Kinase/RTK|Cell Cycle| CSNpharm

DYRK

DYRK
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货号	产品名	CAS号	信息
CSN25712	ProINDY	719277-30-2	ProINDY, the prodrug form of INDY, is an inhibitor of DYRK1A and DYRK1B.
CSN23650	Ml 315	1440251-53-5	ML 315 HCl is inhibitor of Clk and DYRK kinases with IC50s of 68, 68 and 231 nM for Clk1, Clk4 and Clk2, 282 and 1156 nM for Dyrk1A and Dyrk1B.
CSN17778	Mirk-IN-1	1386979-55-0	Mirk-IN-1 is a potent inhibitor of Dyrk1B (Mirk kianse) and Dyrk1A with IC50 of 68±48 nM and 22±8 nM respectively.
CSN25711	INDY	1169755-45-6	INDY is inhibitor of DYRK1B and DYRK1A with IC50 values of 0.23 and 0.24 μM respectively.
CSN17160	ID-8	147591-46-6	ID-8 is an inhibitor of DYRK inhibitor that can sustain embryonic stem cell self-renewal and survival without differentiation.
CSN22843	GSK-626616	1025821-33-3	GSK 626616 is a potent and selective DYRK inhibitor with IC50 of 0.7 nM for DYRK3, similar potency for DYRK1 and 2.
CSN24803	GNF4877	2041073-22-5	GNF4877 is a potent DYRK1A and GSK3β inhibitor with IC50s of 6 nM and 16 nM, respectively
CSN22699	AZ-Dyrk1B-33	1679330-37-0	AZ Dyrk1B 33 is a potent and selective ATP-competitive Dyrk1B kinase inhibitor with IC50 of 7 nM.
CSN15862	AZ191	1594092-37-1	AZ 191 is a potent and selective DYRK1B inhibitor with IC50 of 17 nM in a cell-free assay, about 5- and 110-fold selectivity over DYRK1A and DYRK2, respectively.