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E1/E2/E3 Enzyme

E1/E2/E3 Enzyme

货号 产品名 CAS号 信息
CSN23792 VL285 1448188-57-5 VL285 is a potent VHL ligand, degrading HaloTag7 fusion proteins.
CSN20606 VH-298 2097381-85-4 VH-298 is a highly affinity inhibitor of E3 ubiquitin ligase VHL inhibitor (Kd = 80-90 nM) which can block the interaction of VHL and HIF-α, thus initiating hypoxic response.
CSN17382 TZ9 1002789-86-7 TZ9 is an inhibitor of Rad6 ubiquitin conjugating enzyme (E2 enzyme) and inhibits MDA-MB-231 cell proliferation with IC50 of ~6 μM.
CSN22266 E3 Ligand-Linker Conjugate 10 1957236-22-4 Thalidomide-O-amido-PEG4-C2-Amine is a PROTAC block consist of Thalidomide and a linker with Amine functional group for conjugation reactions.
CSN22271 E3 Ligand-Linker Conjugate 7 2022182-59-6 Thalidomide-O-amido-PEG-C2-Amine is a PROTAC block consist of Thalidomide and a linker with Amine functional group for conjugation reactions.
CSN22272 E3 Ligand-Linker Conjugate 6 2022182-57-4 Thalidomide-O-amido-C3-Amine is a PROTAC block consist of Thalidomide linked to alkyl with Amine functional group for conjugation reactions.
CSN24768 Thalidomide-linker 2 2245697-85-0 Thalidomide-linker 2 is a PROTAC block consist of Thalidomide and a linker with Amine functional group for conjugation reactions.
CSN21424 E3 ligase Ligand 3 1061605-21-7 TC E3 5031 is a thalidomide derivate for conjugation reactions of PROTAC, which can hijack cereblon as the E3 ubiquitin ligase component.
CSN17260 SZL P1-41 222716-34-9 SZL P1-41 is Skp2 inhibitor, selectively suppresses Skp2 E3 ligase activity, but not activity of other SCF complexes.
CSN25714 SMER 3 67200-34-4 SMER 3 is a selective inhibitor of yeast SCF family E3 ubiquitin ligase (SCFMet30) in vitro and in vivo.
CSN18199 PRT4165 31083-55-3 PRT4165, an inhibitor of bim1 and ring1A, could block PRC1 (Polycomb-repressive complex 1)-mediated H2A ubiquitylation.
CSN22492 PROTAC Linker 1 1835705-53-7 PROTAC Linker 1 is a linker used to link the warhead and the E3 ligase ligand.
CSN19741 PK11195 85532-75-8 PK11195 is a 2‑Phenylindolylglyoxylyldipeptide Murine Double Minute2 (MDM2)/Translocator Protein (TSPO)/Human Constitutive Androstane Receptor (hCAR) Inhibitor, and is potentially useful for the Treatment of Gliomas.
CSN17303 NSC 697923 343351-67-7 NSC 697923 is a cell-permeable and selective inhibitor of the Ub-conjugating enzyme (E2) complex Ubc13-Uev1A.
CSN27723 MID-1   312608-54-1 MID-1 is a MG53-IRS-1 interaction disruptor. It abolished MG53-mediated IRS-1 ubiquitination and degradation, as well as sensitized insulin signaling and increased insulin-elicited glucose uptake with an elevated level of IRS-1 in C2C12 myotubes.
CSN20357 MDK7526 1448297-52-6 MDK7526 is a ligand of Von Hippel–Lindau protein, that can be used for making proteolysis targeting chimeras (PROTACs).
CSN32744 EMBL 445222-91-3 EMBL is an inhibitor of MuRF1.
CSN28743 E3 ligase Ligand 9 87304-15-2 E3 ligase Ligand 9 is a Bestatin-based E3 ligase ligand.
CSN21237 E3 Ligase Ligand 6 1631137-51-3 E3 Ligase Ligand 6 is used for conjugation reactions of PROTAC, which can hijack VHL as the E3 ubiquitin ligase component.
CSN21420 E3 ligase Ligand 2 5054-59-1 E3 ligase Ligand 2 is a thalidomide derivate for conjugation reactions of PROTAC, which can hijack cereblon as the E3 ubiquitin ligase component.
CSN33243 tert-Butyl 4-(2-(2,6-dioxopiperidin-3-yl)-3-oxoisoindolin-5-yl)piperazine-1-carboxylate 2229723-91-3
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