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Epigenetic Reader Domain
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN22252 | KG-501 | 18228-17-6 | KG-501 is histochemical substrate of alkaline phosphatases and can inhibit CREB-CBP interaction. |
| CSN18953 | GSK6853 | 1910124-24-1 | GSK6853 selectively inhibits the BRPF1 bromodomain with the pKd value of 9.5. |
| CSN17637 | GSK525768A | 1260530-25-3 | GSK525768A is the enantiomer compound of GSK 525762A, which is a potent small molecule inhibitor that disrupt the function of the BET family of bromodomains (Brd2, Brd3, and Brd4) and has NO activity towards BET. |
| CSN22423 | GSK1379725A | 1802251-00-8 | GSK1379725A is an inhibitor of Brd4 and a selective BPTF ligand (Kd=2.8 μM). |
| CSN27738 | CBP/EP300-IN-1 | 2443789-32-8 | CBP/EP300-IN-1 is a CBP/EP300 bromodomain inhibitor. |
| CSN18957 | BET-BAY 002 S-Enantiomer | 2070009-49-1 | BET-BAY 002 S-enantiomer is the S-enantiomer of BET-BAY 002. |
| CSN17940 | BET-BAY 002 | 1588521-78-1 | BET-BAY 002 is a potent BET inhibitor and shows efficacy in a multiple myeloma model. |
| CSN21392 | AT6 | 2098836-50-9 | AT6 is a PROTAC targeting on Brd4. |
| CSN18046 | ARV-825 | 1818885-28-7 | ARV-825 is a PROTAC targeting on BRD4, consisting of a BRD4-ligand JQ-1 linked to a cereblon E3 ligase ligand Pomalidomide, with Kds values of 90nM and 28nM for affinity to BD1 and BD2. |
| CSN18086 | JQ-1 Carboxylic Acid | 202592-23-2 | (+)-JQ1 carboxylic acid is a warhead ligand with a carboxylic acid functional group for conjugation reactions of PROTAC targeting on BET. |
