Epigenetic Reader Domain

Epigenetic Reader Domain
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货号	产品名	CAS号	信息
CSN22252	KG-501	18228-17-6	KG-501 is histochemical substrate of alkaline phosphatases and can inhibit CREB-CBP interaction.
CSN18953	GSK6853	1910124-24-1	GSK6853 selectively inhibits the BRPF1 bromodomain with the pKd value of 9.5.
CSN18952	BI-9564	1883429-22-8	BI-9564 is an inhibitor of BRD9 (IC50 = 75 nM) and BRD7 (IC50 = 3.4 µM).
CSN18046	ARV-825	1818885-28-7	ARV-825 is a PROTAC targeting on BRD4, consisting of a BRD4-ligand JQ-1 linked to a cereblon E3 ligase ligand Pomalidomide, with K_ds values of 90nM and 28nM for affinity to BD1 and BD2.
CSN24157	666-15	1433286-70-4	666-15 is a potent and cell-permeable inhibitor of cAMP-response element binding protein (CREB) with efficacious anti-cancer activity both in vitro and in vivo.
CSN18086	JQ-1 Carboxylic Acid	202592-23-2	(+)-JQ1 carboxylic acid is a warhead ligand with a carboxylic acid functional group for conjugation reactions of PROTAC targeting on BET.