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Epigenetic Reader Domain

Epigenetic Reader Domain

货号 产品名 CAS号 信息
CSN22252 KG-501 18228-17-6 KG-501 is histochemical substrate of alkaline phosphatases and can inhibit CREB-CBP interaction.
CSN18953 GSK6853 1910124-24-1 GSK6853 selectively inhibits the BRPF1 bromodomain with the pKd value of 9.5.
CSN17637 GSK525768A 1260530-25-3 GSK525768A is the enantiomer compound of GSK 525762A, which is a potent small molecule inhibitor that disrupt the function of the BET family of bromodomains (Brd2, Brd3, and Brd4) and has NO activity towards BET.
CSN22423 GSK1379725A 1802251-00-8 GSK1379725A is an inhibitor of Brd4 and a selective BPTF ligand (Kd=2.8 μM).
CSN27738 CBP/EP300-IN-1 2443789-32-8 CBP/EP300-IN-1 is a CBP/EP300 bromodomain inhibitor.
CSN18957 BET-BAY 002 S-Enantiomer 2070009-49-1 BET-BAY 002 S-enantiomer is the S-enantiomer of BET-BAY 002.
CSN17940 BET-BAY 002 1588521-78-1 BET-BAY 002 is a potent BET inhibitor and shows efficacy in a multiple myeloma model.
CSN21392 AT6 2098836-50-9 AT6 is a PROTAC targeting on Brd4.
CSN18046 ARV-825 1818885-28-7 ARV-825 is a PROTAC targeting on BRD4, consisting of a BRD4-ligand JQ-1 linked to a cereblon E3 ligase ligand Pomalidomide, with Kds values of 90nM and 28nM for affinity to BD1 and BD2.
CSN18086 JQ-1 Carboxylic Acid 202592-23-2 (+)-JQ1 carboxylic acid is a warhead ligand with a carboxylic acid functional group for conjugation reactions of PROTAC targeting on BET.
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