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GPCR

GPCR

货号 产品名 CAS号 信息
CSN23913 TUG-1375 2247372-59-2 TUG-1375 is a free fatty acid receptor 2 (FFA2/GPR43) inhibitor with pKi of 6.69.
CSN23156 TC-O 9311 444932-31-4 TC-O 9311 is a potent orphan G protein-coupled receptor 139 (GPR139) agonist with an EC50 of 39 nM[1].
CSN25229 SBI-115   882366-16-7 SBI-115 is a GPBAR1 (TGR5) antagonist.
CSN24134 PMX 53 219639-75-5 PMX 53 is a potent C5a receptor antagonist.
CSN22253 Monosodium Taurocholate 145-42-6 Monosodium taurocholate is an agonist of GPBAR1 and is potential of the treatment of type 2 diabetes and obesity in rats.
CSN22976 ML 193 713121-80-3 ML 193 is a selective GPR55 antagonist with IC50 of 221 nM.
CSN22972 MK 1903 1268882-43-4 MK 1903 is a potent and selective hydroxycarboxylic acid receptor 2 (HCA2, GPR109A) full agonist.
CSN22968 MEDICA 16 87272-20-6 MEDICA 16 is a free fatty acid 1 (FFA1/GPR40) receptor agonist.
CSN23711 MCHr1 Antagonist 1 391610-37-0 MCHr1 antagonist 1 is a selective antagonist of MCH1 receptor with Kb of 1 nM and Ki of 4 nM at human MCHR1, may be used to reduce the body mass.
CSN25201 Hyodeoxycholic acid 83-49-8 Hyodeoxycholic(HDCA) acid is a secondary bile acid, one of the metabolic byproducts of intestinal bacteria.
CSN23532 AF64394 1637300-25-4 F64394 is an inverse agonist of GPR3 with pIC50 of 7.3.
CSN20629 Diphenyleneiodonium Chloride 4673-26-1 Diphenyleneiodonium chloride is an agonist of GPR3 with EC50 of 1 μM. It can activate adenylate cyclase.
CSN25392 Deoxycholic acid sodium salt 302-95-4 Deoxycholic acid sodium salt is specifically responsible for activating the G protein-coupled bile acid receptor TGR5 that stimulates brown adipose tissue (BAT) thermogenic activity.
CSN20443 CYM 5541 945128-26-7 CYM-5541 is an allosteric agonist of S1P3 with EC50 of 72 nM - 132 nM.
CSN23236 CID 1375606 313493-80-0 CID 1375606 is an agonist of GPR27 (SREB1) that induces coupling of the receptor to β-arrestin 2.
CSN22671 AH 7614 6326-06-3 AH 7614 is a selective free fatty acid receptor 4 (FFA4/GPR120) antagonist with pIC50 of 7.1 for human FFA4.
CSN20400 AEZS-108 139570-93-7 AEZS-108 is a peptide agonist of the gonadotropin releasing hormone-1 receptor (GnRH-1R).
CSN25414 3-chloro-5-hydroxybenzoic Acid 53984-36-4 3-chloro-5-hydroxybenzoic Acid is a selective GPR81 agonist that exhibited favorable in vivo effects on lipolysis in a mouse model of obesity.
CSN23486 3,5-Dihydroxybenzoic acid 99-10-5 3, 5-dihydroxybenzoic acid is a metabolite of alkylresinols with a certain activation effect on HCA1. It can be used as intermediates in organic synthesis.
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