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Histamine Receptor
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN25848 | N-(3-(3-(Piperidin-1-ylmethyl)phenoxy)propyl)benzo[d]thiazol-2-amine dimaleate | 104076-39-3 | Zolantidine dimaleate is a selective and brain penetrating H2 receptor antagonist. |
| CSN25862 | VUF 8430 dihydrobromide | 100130-32-3 | VUF 8430 dihydrobromide is a full agonist of histamine H4 receptor with pKi of 7.5 and pEC50 of 7.3. |
| CSN25841 | Triprolidine hydrochloride | 550-70-9 | Trans-Triprolidine hydrochloride is a potent H1 receptor antagonist. |
| CSN25844 | Tiotidine | 69014-14-8 | Tiotidine is antagonist of histamine H2-receptor with negligible activity against H1- and H3- receptors. |
| CSN26513 | SUN 1334H | 607736-84-5 | SUN-1334H is a histamine H1 receptor antagonist potentially for the treatment of allergic conjunctivitis and allergic rhinitis |
| CSN24554 | SEN12333 | 874450-44-9 | SEN 12333 is a selective agonist of α7 nicotinic acetylcholine receptor (nAChR) with EC50 and Ki of 1.6 μM, 260 nM in rat. It also displays functional antagonism at histamine H3 receptors (IC50 = 103 nM). |
| CSN21826 | Rocastine | 91833-77-1 | Rocastine is a selective antagonist of nonsedative H1 antagonist for antihistamines. |
| CSN26180 | PU02 | 313984-77-9 | PU-02 is an antagonist of serotonin (5-HT) receptor subtype 5-HT3. |
| CSN17113 | Promethazine hydrochloride | 58-33-3 | Promethazine HCl is the effective antagonist of the H1 receptor and moderate antagonist of mACh receptor. |
| CSN25855 | 2-(1H-Imidazol-4-yl)-N-methylethanamine dihydrochloride | 16503-22-3 | Nα-Methylhistamine dihydrochloride is H2R agonist that acts directly on histamine H(2) receptors (H2Rs) in animals to stimulate acid secretion and it dose dependently stimulated cAMP productions in CHO-H2R cells. |
| CSN11591 | Nylidrin hydrochloride | 849-55-8 | Nylidrin HCl was an effective inhibitor of IgE-mediated release of histamine from passively sensitized rat peritoneal mast cells and human basophils, and of IgG1-mediated release of histamine from passively sensitized guinea pig lung slices. |
| CSN21744 | Niperotidine | 84845-75-0 | Niperotidine is an antagonist of histamine H2-receptor. |
| CSN11531 | Nedocromil | 69049-73-6 | Nedocromil is an inhaled anti-inflammatory agent for the preventive management of asthma. |
| CSN25565 | LML134 | 1542135-76-1 | LML134 is an orally active and high selective Histamine 3 receptor (H3R) inverse agonist with Kis of 0.3 nM and 12 nM for hH3R cAMP and hH3R bdg. LML134 penetrates the brain rapidly, leading to high H3R occupancy, and disengages its target with a fast kinetic profile. LML134 has the potential for excessive sleep disorders. |
| CSN25273 | JNJ-5207852 | 398473-34-2 | JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor. |
| CSN25851 | Impentamine dihydrobromide | 149629-70-9 | Impentamine dihydrobromide is highly selective antagonist of histamine H3 receptor with pA2 of 8.4. |
| CSN25847 | Ici162,846 | 84545-30-2 | ICI 162,846 is a potent histamine H2 receptor antagonist. |
| CSN25852 | GT-2016 | 152241-24-2 | GT 2016 is a high affinity antagonist of H3 receptor with Ki of 43.8 nM. |
| CSN22023 | FRG8701 | 108498-50-6 | FRG-8701 is a new Histamine H2-receptor antagonist with IC50 of ranging from 0.25 to 0.43 μM. |
| CSN21734 | Minocromil | 85118-44-1 | FPL59360, a anti-asthmatic compound, is histamine I receptor antagonist that prevents exercise-induced asthma. |
| CSN24500 | Emedastine | 87233-61-2 | Emedastine is a potent, high affinity histamine H1-receptor-selective antagonist with Ki of 1.3 ±0.1 nM for H1-receptors while considerably weaker at H2- (Ki = 49,067 ± 11,113 nM) and H3-receptors (Ki = 12,430 ± 1,282 nM). |
| CSN25845 | Dimaprit dihydrochloride | 23256-33-9 | Dimaprit dihydrochloride is a selective H2 agonist with central effects upon systemic administration. |
| CSN25857 | Conessine | 546-06-5 | Conessine is a steroid alkaloid that acts as a specific antagonist of histamine H3 receptor with Ki of 5.37. |
| CSN26664 | Cimetidine sulfoxide | 54237-72-8 | Cimetidine sulfoxide (Cimetidine sulphoxide) is a sulfoxide metabolite of Cimetidine. Cimetidine is a histamine H2-receptor antagonist. Cimetidine has the potential for peptic ulcer disease and upper gastrointestinal haemorrhage treatment[1]. |
| CSN26201 | Chloropyramine hydrochloride | 6170-42-9 | Chloropyramine hydrochloride is a histamine receptor H1 antagonist which can also inhibit the biochemical function of VEGFR-3. Chloropyramine hydrochloride may be useful in the treatment of invasive breast cancer. |
| CSN25269 | Bromodiphenhydramine hydrochloride | 1808-12-4 | Bromazine hydrochloride is an antagonist of histamine H1 receptor. |
| CSN24556 | AR-R17779 hydrochloride | 178419-42-6 | AR-R 17779 hydrochloride is a selective alpha7 nicotinic agonist with Ki value of 190 nM for rat. |
| CSN25846 | Amthamine dihydrobromide | 142457-00-9 | Amthamine dihydrobromide is a highly selective agonist of H2 receptor. |
| CSN25843 | Aminopotentidine | 140873-26-3 | Aminopotentidine is antagonist of H2 with KB value of 220 nM. |
| CSN21455 | Acrivastine | 87848-99-5 | Acrivastine, an H1-receptor antagonist, is a second-generation antihistamine. |
| CSN26178 | N-(3-Chloro-2-methylphenyl)quinoxaline-2-carboxamide | 930478-88-9 | 5-HT3 antagonist-4i is a 5-HT3 receptor antagonist which modulates the serotonergic system. |
| CSN25863 | 4-Methylhistamine dihydrochloride | 36376-47-3 | 4-Methylhistamine dihydrochloride is a high affinity agonist of H4 receptor with Ki of 7 nM. |
| CSN25840 | 2-(Pyridin-2-yl)ethanamine dihydrochloride | 3343-39-3 | 2-Pyridylethylamine dihydrochloride is an agonist of histamine H1 receptor that produces vasoconstriction. |
| CSN24562 | (S)-(+)-Dimethindene maleate | 136152-65-3 | (S)-(+)-Dimethindene maleate is a subtype-selective M2 muscarinic receptor antagonist with pKi of 7.78 and is also a H1 histamine receptor antagonist with pKi of 7.48. |
| CSN25856 | (R)-(-)-α-Methylhistamine dihydrobromide | 868698-49-1 | (R)-(-)-α-Methylhistamine dihydrobromide is a very potent agonist of H3 receptor with Kd of 50.3 nM that crosses the blood-brain barrier and inhibits histamine synthesis and release at nanomolar concentrations. |
| CSN36535 | Pimethixene maleate | 13187-06-9 | |
| CSN34474 | QF0301B | 149247-12-1 | |
| CSN63870 | Paliperidone-d4 | 1020719-55-4 | |
| CSN68409 | 4,4-Diphenylbutylamine hydrochloride | 22101-90-2 | |
| CSN68935 | Histamine H4 receptor antagonist-1 | 1246207-84-0 | |
| CSN83992 | Melitracen | 5118-29-6 | |
| CSN85193 | Izuforant | 1429374-83-3 | |
| CSN90189 | Dimethothiazine | 7456-24-8 | |
| CSN104778 | 3-(4-(Dibenzo[b,f][1,4]oxazepin-6-yl)piperazin-1-yl)-2,2-dimethylpropanoic acid | 879409-35-5 | |
| CSN105278 | 1-(6-((3-Cyclobutyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yl)oxy)pyridin-3-yl)pyrrolidin-2-one | 720691-69-0 | |
| CSN105231 | (R)-2-((1-(4-(4-(3-(Azepan-1-yl)propoxy)phenyl)butyl)pyrrolidin-2-yl)methyl)-4-(4-chlorobenzyl)phthalazin-1(2H)-one | 955359-72-5 |
