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Histamine Receptor

Histamine Receptor

货号 产品名 CAS号 信息
CSN20447 VUF 10460 1028327-66-3 VUF 10460 is a selective agonist of histamine H4 receptor with pKi of 8.22.
CSN21872 Triprolidine HCl 6138-79-0 Triprolidine Hydrochloride is the first generation histamine H1 antagonist used in allergic rhinitis.
CSN19848 Thioperamide 106243-16-7 Thioperamide is a potent HRH4 antagonist and selective HRH3 antagonist capable of crossing the blood–brain barrier.
CSN17265 Setastine 64294-95-7 Setastine is an antihistamine used to treat allergies and rhinitis.
CSN21281 S 38093 862896-30-8 S 38093 is a brain-penetrant antagonist/inverse agonist of H3 receptors.
CSN26180 PU-02   313984-77-9 PU-02 is an antagonist of serotonin (5-HT) receptor subtype 5-HT3.
CSN17113 Promethazine HCl 58-33-3 Promethazine HCl is the effective antagonist of the H1 receptor and moderate antagonist of mACh receptor.
CSN18242 Pitolisant Oxalate 362665-57-4 Pitolisant oxalate is a potent, and selective nonimidazole inverse agonist at the recombinant human H3 receptor (Ki=0.16 nM).
CSN17352 Pitolisant 362665-56-3 Pitolisant is a potent, and selective nonimidazole inverse agonist at the recombinant human H3 receptor (Ki=0.16 nM).
CSN21315 Pirolate 55149-05-8 Pirolate (CP-32,387) is an antihistamine drug with a tricyclic chemical structure which was patented as an "antiallergen".
CSN18828 Osthole 484-12-8 Osthole, an O-methylated coumarin, is a histamine H1 receptor inhibitior. It exhibits immunomodulatory, antioxidative and anti-inflammatory activities.
CSN21105 N-omega-Acetylhistamine 673-49-4 N-acetylhistamine is a histamine metabolite. N-acetylhistamine can be used as a potential biomarker of histidine metabolism for anaphylactoid reactions.
CSN21134 Mebhydrolin 524-81-2 Mebhydrolin is a specific histamine H1 receptor antagonist.
CSN14575 Marmin 14957-38-1 Marmin, a natural product isolated and purified from the herbs of Citrus maxima with potent anti-ulcer, antibacterial, fungicidal, and algicidal properties, can inhibit contraction of the guinea-pig tracheal smooth muscle, especially by interfering histamine receptor, inhibiting the histamine release from mast, inhibiting intracellular Ca2+ release from the intracellular store and the Ca2+ influx through voltage-dependent Ca2+ channels, is potential to develop as antihistamine agents, especially as histamine H1 receptor antagonists by interacting with amino acid residues, Asp107, Lys179, Lys191, Asn198, and Trp428 of histamine H1 receptor, shows a cell-growth inhibitory effect against L1210 and K562 in vitro.
CSN19403 Ketotifen Fumarate 34580-14-8 Ketotifen fumarate is a noncompetitive H1 receptor antagonist and mast cell stabilizer that is used to treat asthma.
CSN16759 JNJ-7777120 459168-41-3 JNJ-7777120 is a selective antagonist of histamine-4 receptor (H4R) with Ki of 4 ± 1 nM.
CSN25273 JNJ-5207852 398473-34-2 JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.
CSN17063 Hydroxyzine 68-88-2 Hydroxyzine is a histamine H1-receptor antagonist.
CSN16784 Famotidine 76824-35-6 Famotidine is antagonist of histamine H2–receptor with IC50 of 0.6 mM that used to treat heartburn and other digestive conditions.
CSN19386 Epinastine 80012-43-7 Epinastine is mast cell stabilizer and antihistamine that is used to treat allergic conjunctivitis.
CSN21346 Cyclizine 82-92-8 Cyclizine, a piperazine derivative, is an antihistaminic antiemetic that is useful in the prevention and treatment of nausea and vomiting associated with motion sickness.
CSN22573 Cyclizine 2HCl 5897-18-7 Cyclizine is a histamine H1 receptor antagonist of the piperazine class.
CSN21347 Cyclizine HCl 303-25-3 Cyclizine HCl is a piperazine derivative with anti-emetic activity that is useful in the prevention and treatment of nausea and vomiting associated with motion sickness.
CSN20584 Clobenpropit Dihydrobromide 145231-35-2 Clobenpropit hydrobromide is a selective histamine H3 receptor antagonist that crosses the blood-brain barrier, inhibiting histamine binding in rat brain.
CSN18049 Ciproxifan 184025-18-1 Ciproxifan is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity at other receptor subtypes.
CSN22139 Cipralisant 213027-19-1 Cipralisant is a potent and selective histamine H3 receptor antagonist in vivo, and an agonist in vitro, with a pKi of 9.9 for histamine H3 receptor and a Ki of 0.47 nM for rat histamine H3 receptor; Cipralisant has entered in clinical trials for the treatment of attention-deficit hyperactivity disorder.
CSN23808 Chlorcyclizine HCl 14362-31-3 Chlorcyclizine hydrochloride is a histamine H1 antagonist.
CSN25269 Bromazine HCl 1808-12-4 Bromazine hydrochloride is an antagonist of histamine H1 receptor.
CSN22167 BMY-25271 78441-82-4 BMY-25271 is a histamine H2 receptor antagonist.
CSN25225 Betahistine 5638-76-6 Betahistine is a histamine analog and H1 receptor agonist.
CSN17080 Betahistine 2HCl 5579-84-0 Betahistine 2HCl is histamine H3 receptor inhibitor with IC50 of 1.9 μM. It is an antivertigo drug.
CSN24137 Bepotastine 125602-71-3 Bepotastine is a non-sedating and selective antagonist of the histamine 1 (H1) receptor.
CSN16768 Azelastine 58581-89-8 Azelastine is a potent, second-generation, selective, histamine antagonist.
CSN16787 Azelastine HCl 79307-93-0 Azelastine HCl is a selective antagonist of histamine receptor used in the treatment of rhinitis.
CSN18662 Antazoline HCl 2508-72-7 Antazoline HCl is a antihistamine with anticholinergic properties. It is used to relieve nasal congestion.
CSN23462 5-Hydroxyindole-3-acetic acid 54-16-0 5-Hydroxyindole-3-acetic acid (5-HIAA), the major metabolite of serotonin, is a histamine H1 receptor antagonist and can be used to treat allergies.
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