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HSP
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN13116 | VER-155008 | 1134156-31-2 | VER-155008 is a potent Hsp70 family inhibitor with IC50 of 0.5 μM, 2.6 μM, and 2.6 μM in cell-free assays for HSP70, HSC70, and GRP78, respectively, > 100-fold selectivity over HSP90. |
| CSN20344 | TRC051384 HCl | 1333327-56-2 | TRC051384 is an inducer of heat shock protein Hsp70. it reduces stroke-associated neuronal injury and increases survival in a rat model of transient ischemic stroke and activates heat shock factor-1 and results in elevated chaperone and anti-inflammatory activity. |
| CSN12051 | Teprenone | 6809-52-5 | Teprenone is used as an anti-ulcer drug, a cardioprotective agent, a hepatoprotective agent, a nephroprotective agent, a neuroprotective agent and a Hsp70 inducer. |
| CSN22232 | TAS-116 | 1260533-36-5 | TAS-116 is a potent and selective HSP90α/β inhibitor with Kis of 34.7 nM, 21.3 nM, respectively. |
| CSN15760 | PU-WS13 | 1454619-14-7 | PU-WS13 is a potent, Grp94-specific Hsp90 inhibitor of the purine scaffold class. |
| CSN16046 | PU-H 71 | 873436-91-0 | PU-H71 is a potent Hsp90 inhibitor with IC50 of 50 nM. |
| CSN17514 | PF-04929113 Mesylate | 1173111-67-5 | PF-04929113 mesylate is a potent and selective Hsp90 inhibitor with an IC50 of median 50 nM. |
| CSN17387 | ML346 | 100872-83-1 | ML346 is an activator of Hsp70 with EC50 of 4600 nM in HeLa cell toxicity assay. |
| CSN21425 | MKT-077 | 147366-41-4 | MKT-077 (FJ-776) is a water-soluble rhodacyanine dye with antitumor activity. It can bind to Hsp70 family member mortalin-2 and inhibit its interactions with p53. |
| CSN18942 | KRIBB11 | 342639-96-7 | KRIBB11 is an inhibitor of heat shock factor (HSF) inhibitor, with IC50 of 1.2 μM. |
| CSN17321 | KNK437 | 218924-25-5 | KNK437 is a pan-HSP inhibitor, which inhibits the synthesis of inducible HSPs, including HSP105, HSP72, and HSP40. |
| CSN11085 | Geldanamycin | 30562-34-6 | Geldanamycin is a natural existing HSP90 inhibitor with Kd of 1.2 μM. |
| CSN22828 | Gedunin | 2753-30-2 | Gedunin is a Hsp90 inhibitor and exhibits anticancer and antimalarial activity. |
| CSN25416 | Ethoxyquin | 91-53-2 | Ethoxyquin is an antioxidant which has been used in animal feed for many years and also an inhibitor of heat shock protein 90 (Hsp90). |
| CSN27185 | Col003 | 328565-16-8 | Col003 is a cell penetrant, selective and potent inhibitor of the interaction of Hsp47 with collagen. Col003 is the cleavage product of AK778.It competitively inhibited the interaction and caused the inhibition of collagen secretion by destabilizing the collagen triple helix. |
| CSN22743 | CCT 018159 | 171009-07-7 | CCT 018159 is a novel inhibitor of heat shock protein 90 (Hsp90) ATPase activity with IC50 of 5.7 μM. |
| CSN18941 | Apoptozole | 1054543-47-3 | Apoptozole is an inhibitor of heat shock protein 70 (HSP70) and Hsc70. It induces caspase-dependent apoptosis. |
| CSN18284 | Alvespimycin HCl | 467214-21-7 | Alvespimycin HCl is a potent, water-soluble HSP90 inhibitor with IC50 of 62 nM. |
| CSN17209 | 17-AAG | 75747-14-7 | 17-AAG is a potent HSP90 inhibitor with IC50 of 5 nM, having a 100-fold higher binding affinity for HSP90 derived from tumour cells than HSP90 from normal cells. |
