| CSN22353 |
AZ3451
|
2100284-59-9 |
AZ3451 is a protease-activated receptor-2 (PAR2) antagonist. |
| CSN22357 |
Beperidium Iodide
|
86434-57-3 |
Beperidium iodide shows a competitive antagonistic effect against acetylcholine receptor with a pA2 of 7.93. |
| CSN22337 |
Adavivint
|
1467093-03-3 |
Adavivint is a potent and selective inhibitor of canonical Wnt signaling, with an EC50 of 19.5 nM via a high-throughput TCF/LEF-reporter assay in SW480 colon cancer cells. |
| CSN22471 |
Nedocromil Sodium
|
69049-74-7 |
Nedocromil Sodium is a potent TNF-α inhibitor with an IC50 value of 1.67 μM for Blood eosinophils. |
| CSN22454 |
Lymecycline
|
992-21-2 |
Lymecycline is a tetracycline derivative, with broad-spectrum antibacterial activity and also has anti-inflammatory property. |
| CSN22371 |
Cephalosporin C Zinc Salt
|
59143-60-1 |
Cephalosporin C zinc salt is a potent inhibitor of SAMHD1 with an IC50 of 1.1 μM. |
| CSN22191 |
MK-0429
|
227963-15-7 |
MK-0429 is a potent integrin antagonist with IC50s of 12.2 nM (α5β1 integrin) and 2.8 nM (αvβ3 integrin), respectively. |
| CSN22375 |
Cl-amidine
|
913723-61-2 |
Cl-amidine is a peptidylarginine deminase (PAD) inhibitor, with an IC50 5.9±0.3 μM for PAD4. |
| CSN22333 |
A-69412
|
123606-23-5 |
A-69412 is a reversible, specific inhibitor of the hydrophilic 5-lipoxygenase (5-LO). |
| CSN22409 |
Gefapixant
|
1015787-98-0 |
Gefapixant is an orally active P2X3 receptor (P2X3R) antagonist with IC50s of ~30 nM versus recombinant hP2X3 homotrimers and 100-250 nM at hP2X2/3 heterotrimeric receptors. |
| CSN22527 |
TY-51469
|
603987-59-3 |
TY-51469 is a chymase inhibitor with IC50s for simian and human chymases of 0.4 and 7.0 nM, respectively. |
400-920-2911
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