Kainate receptors, or kainic acid receptors (KARs), are ionotropic receptors that respond to the neurotransmitter glutamate.
|CSN23175||UBP 282||544697-47-4||UBP-282 is an α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) and kainate receptor antagonist.|
|CSN24615||UBP 310||902464-46-4||UBP 310 is an antagonist of GluK1 (formerly GLUK5) kainate receptor with IC50 of 130 nM.|
|CSN24617||(S)-2-((3-(2-Amino-2-carboxyethyl)-2,6-dioxo-2,3-dihydropyrimidin-1(6H)-yl)methyl)benzoic acid||745055-91-8||UBP 302 is a potent and selective GluK1 (formally GluR5)-subunit containing kainate receptor antagonist with KD of 402 nM.|
|CSN16600||L-Theanine||3081-61-6||L-theanine is an amino acid found most commonly in tea leaves and binds to ionotropic glutamate receptors in the micromolar range, including the AMPA and kainate receptors and, to a lesser extent, the NMDA receptor.|
|CSN19846||Kainic Acid||487-79-6||Kainic acid is a selective agonist at kainate receptors. Potent excitant and neurotoxin.|
|CSN24616||ATPA||140158-50-5||ATPA is a selective and potent GluK1 kainate receptor agonist with Ki of 4.3 nM.|
|CSN11876||(S)-Willardiine||21416-43-3||(S)-Willardiine is a potent agonist of AMPA/kainate receptors with EC50 of 44.8 μM.|