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Kinesin
货号 | 产品名 | CAS号 | 信息 |
---|---|---|---|
CSN13619 | SB-743921 hydrochloride | 940929-33-9 | SB-743921 is a potent KIF11 inhibitor with Ki value of 0.1 nM. |
CSN18934 | PF-2771 | 2070009-55-9 | PF-2771 is a potent, selective CENP-E inhibitor, PF-2771 inhibits CENP-E motor activity with an IC50 of 16.1 ± 1.2 nM. |
CSN18931 | Monastrol | 329689-23-8 | Monastrol is a specific and allosteric inhibitor of mitotic molecular motor kinesin Eg5 with IC50 value of 14 μM. |
CSN18557 | Litronesib | 910634-41-2 | Litronesib is a selective, allosteric inhibitor of Eg5, which may result in mitotic disruption, apoptosis and consequently cell death in tumor cells that are actively dividing. |
CSN18383 | Kif15-IN-2 | 672926-33-9 | Kif15-IN-2 is a potent Kif15 kinesin inhibitor and inhibits cellular proliferation in tumor cell lines. |
CSN18382 | Kif15-IN-1 | 672926-32-8 | Kif15-IN-1 is a potent Kif15 kinesin inhibitor and inhibits cellular proliferation in tumor cell lines. |
CSN18408 | K858 (Racemic) | 72926-24-0 | K858 is a selective and ATP-uncompetitive mitotic kinesin Eg5 inhibitor with IC50 value of 1.3 μM. |
CSN12370 | Ispinesib | 336113-53-2 | Ispinesib is a quinazolinone-derived, specific and reversible kinesin spindle protein inhibitor with Kiapp value of 1.7 nM. |
CSN23527 | S-Trityl-L-cysteine | 2799-07-7 | H-Cys(Trt)-OH is a potent and selective inhibitor of mitotic kinesin Eg5 with IC50 value of 140 nM. |
CSN13157 | GSK-923295 | 1088965-37-0 | GSK923295 is a specific allosteric CENP-E inhibito with Ki value of 3.2 nM. |
CSN18490 | Dimethylenastron | 863774-58-7 | Dimethylenastron is specific and reversible mitotic motor kinesin Eg5 inhibitor with IC50 value of 200 nM. |
CSN16978 | CW-069 | 1594094-64-0 | CW069 is a selective and allosteric microtubule motor protein HSET inhibitor with IC50 value of 75 μM. |
CSN25421 | BRD9876 | 32703-82-5 | BRD9876 is a selective inhibitor of MM1S growth. It is selective for microtubule bound Eg5 and causes a rapid arrest in G2/M phase. |
CSN32365 | AZ82 | 1449578-65-7 | AZ82 is a small molecule inhibitor of KIFC1/HSET. |
CSN16565 | (R)-Filanesib | 885060-08-2 | ARRY-520 R-Enantiomer is the R form of ARRY-520, which is a synthetic, small molecule kinesin spindle protein (KSP) inhibitor with IC50 of 6 nM. |
CSN18527 | Filanesib | 885060-09-3 | ARRY-520 is a synthetic, small molecule kinesin spindle protein (KSP) inhibitor with IC50 of 6 nM. |
CSN19191 | ARQ 621 | 1095253-39-6 | ARQ 621 is an allosteric, and selective Eg5 mitotic motor protein inhibitor. |