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Melanocortin Receptor

货号 产品名 CAS号 信息
CSN24285 α-MSH (swine) trifluoroacetate 171869-93-5 α-MSH is endogenous agonist of melanocortin receptor with Ki values of 0.12, 31, 660 and 5700 nM for MC1, MC3, MC4 and MC5 receptors respectively.
CSN21474 α-MSH 581-05-5 α-MSH is endogenous agonist of melanocortin receptor with Ki values of 0.12, 31, 660 and 5700 nM for MC1, MC3, MC4 and MC5 receptors respectively.
CSN27581 THIQ 312637-48-2 THIQ is the first selective agonist of the melanocortin-4 receptor (MC4R), with high affinity and potency for hMC4R (IC50=1.2 nM, EC50=2.1 nM) and rMC4R (IC50=0.6 nM, EC50=2.9 nM). THIQ maintains low potency at MC1R, MC3R and MC5R. THIQ plays a role in eliciting erectile activity in rodents. THIQ acts as a pharmacoperone of the MC4R rescuing the cell surface expression and signaling of some intracellularly retained MC4R mutants .
CSN20790 Melanotan II 121062-08-6 Melanotan II, an analog of α-melanocyte stimulating hormone, is agonist of MC3-R/MC4-R melanocortin that induces melanogenesis and thus increases skin pigmentation.
CSN21457 Melanotan I 75921-69-6 Melanotan I, a synthetic analog of α-MSH, is an agonist of melanocortin receptors with Ki values of 0.085, 0.4, 3.8 and 5.1 nM for MC1, MC3, MC4 and MC5 receptors respectively.
CSN21460 ACTH (1-39), Human 12279-41-3 ACTH (1-39) is agonist of melanocortin receptor 2 (MC2R) with an EC50 of 57 pM in HeLa cells expressing the mouse receptor.
CSN24141 ACTH (1-39) (mouse, rat) 77465-10-2 ACTH (1-39) (mouse, rat) is a potent melanocortin 2 (MC2) receptor agonist.
CSN21459 ACTH (1-17) 7266-47-9 ACTH (1-17), a peptide fragment of adrenocorticotropic hormone, is an agonist of MC1R. It is a
CSN21434 ACTH (1-10), Human 2791-05-1 ACTH (1-10), human is an agonist of melanocortin receptor 3 (MC3R) and MC4R with EC50s of 2.6 and 200 nM, respectively.
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