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| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN11339 | Lubiprostone | 136790-76-6 | Lubiprostone is an ClC-2 chloride channel activator used in the treatment of idiopathic chronic constipation. |
| CSN10030 | Rimonabant HCl | 158681-13-1 | Rimonabant HCl is a selective central cannabinoid (CB1) receptor inverse agonist with Ki of 1.8 nM. |
| CSN10050 | (S)-2-(4-(((2-Amino-4-oxo-3,4-dihydropteridin-6-yl)methyl)amino)benzamido)pentanedioic acid | 59-30-3 | Folic acid, a B vitamin, plays an important role in cell division and in the synthesis of amino acids and nucleic acids like DNA. |
| CSN10055 | Glibenclamide | 10238-21-8 | Glibenclamide is a sulfonylurea compound that modulates insulin production. |
| CSN10130 | Miglitol | 72432-03-2 | Miglitol is a desoxynojirimycin-derived inhibitor of alpha-glucosidase with antihyperglycemic activity. |
| CSN10172 | Sitagliptin phosphate monohydrate | 654671-77-9 | Sitagliptin Phosphate Monohydrate is a potent inhibitor of DPP4 with IC50 of 19 nM in Caco-2 cell extracts. |
| CSN10199 | (2R,3R,4R,5R)-4-(((2R,3R,4R,5S,6R)-5-(((2R,3R,4S,5S,6R)-3,4-Dihydroxy-6-methyl-5-(((1S,4R,5S,6S)-4,5,6-trihydroxy-3-(hydroxymethyl)cyclohex-2-en-1-yl)amino)tetrahydro-2H-pyran-2-yl)oxy)-3,4-dihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)oxy)-2,3,5,6-tetrahydroxyhexanal | 56180-94-0 | Acarbose is an intestinal alpha-glucosidase inhibitor and can be used to treat type 2 diebetes. |
| CSN10251 | (R)-2-((6-(3-Aminopiperidin-1-yl)-3-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)methyl)benzonitrile | 850649-61-5 | Alogliptin is a dipeptidyl peptidase 4 (DPP-4) inhibitor with IC50 of 6.9 nM that exhibits greater selective than DPP-2, DPP-8 and DPP-9. |
| CSN10462 | Bisacodyl | 603-50-9 | Bisacodyl is a Na+/K+-ATPase inhibitor used as a stimulant laxative drug. |
| CSN10464 | Bisindolylmaleimide I | 133052-90-1 | GF109203X is a potent PKC inhibitor with IC50 of 20 nM, 17 nM, 16 nM, and 20 nM for PKCα, PKCβI, PKCβII, and PKCγ in cell-free assays, respectively, showing more than 3000-fold selectivity for PKC as compared to EGFR, PDGFR and insulin receptor. |
| CSN10987 | 2-(3-Cyano-4-isobutoxyphenyl)-4-methylthiazole-5-carboxylic acid | 144060-53-7 | Febuxostat is an inhibitor of xanthine oxidase with Ki of 0.6 nM and can affect the progression of renal disease. |
| CSN11129 | GW 4064 | 278779-30-9 | GW4064 is a selective, non-steroidal farnesoid X receptor (FXR) agonist (EC50 = 15 nM). |
| CSN11264 | Lafutidine | 118288-08-7 | Lafutidine is an antagonist of histamine H(2)-receptor that inhibits gastric acid secretion. |
| CSN11335 | (S)-(1S,3R,7S,8S,8aR)-8-(2-((2R,4R)-4-Hydroxy-6-oxotetrahydro-2H-pyran-2-yl)ethyl)-3,7-dimethyl-1,2,3,7,8,8a-hexahydronaphthalen-1-yl 2-methylbutanoate | 75330-75-5 | Lovastatin is a HMG-CoA reductase used to treat high blood cholesterol and reduce the risk of cardiovascular disease, a naturally occuring fungal metabolite. |
| CSN11395 | Methocarbamol | 532-03-6 | Methocarbamol is a central muscle relaxant used to treat skeletal muscle spasms. |
| CSN11418 | Methyl-5,6-dimethylbenzimidazolylcobalamin | 13422-55-4 | Methylcobalamin is a form of vitamin B12, used to prevent or treat pathology arising from a lack of vitamin B12 intake. |
| CSN11584 | Repaglinide | 135062-02-1 | Repaglinide is a carbamoylmethyl benzoic acid (CMBA) derivative, which recently has become available for the treatment of type II diabetes. |
| CSN10171 | 7,8-Dihydroxy-2-phenyl-4H-chromen-4-one | 38183-03-8 | 7,8-Dihydroxyflavone acts as an agonist of TrkB receptor with Kd of 320 nM with neuroprotective effect. |
| CSN10236 | Alfacalcidol | 41294-56-8 | Alfacalcidol is a non-selective VDR activator medication. |
| CSN11492 | Camostat Mesylate | 59721-29-8 | Camostat mesylate is a trypsin-like protease inhibitor, inhibits airway epithelial sodium channel (ENaC) function with IC50 of 50 nM, less potent to trypsin, prostasin and matriptase. |
| CSN11433 | 2-Methyl-1,2-di(pyridin-3-yl)propan-1-one | 54-36-4 | Metyrapone is an inhibitor of cytochrome P450-mediated ω/ω-1 hydroxylase activity and CYP11B1. |
| CSN11101 | Glipizide | 29094-61-9 | Glipizide is used to treat high blood sugar levels caused by a type of diabetes mellitus called type 2 diabetes. |
| CSN11539 | Neostigmine bromide | 114-80-7 | Neostigmine bromide is a cholinesterase inhibitor used in the treatment of myasthenia gravis. Neostigmine bromide is a reversible AchR inhibitor but can not cross the blood-brain barrier. |
| CSN10123 | Rosiglitazone HCl | 302543-62-0 | Rosiglitazone HCl is a blood glucose-lowering drug, stimulating insulin secretion by binding to the PPAR receptors in fat cells. |
| CSN10441 | Bethanechol chloride | 590-63-6 | Bethanechol chloride is a selective mAchR receptor agonist as a parasympathomimetic choline carbamate. |
| CSN10151 | Tioxolone | 4991-65-5 | Tioxolone, a metalloenzyme carbonic anhydrase I inhibitor with a Ki of 91 nM, is an anti-acne preparation. |
| CSN10234 | Aleglitazar | 475479-34-6 | Aleglitazar is a dual PPAR-α/γ agonist with IC50 of 2.8 nM/4.6 nM. |
| CSN17401 | MK-5046 | 1022152-70-0 | MK-5046 is a BRS-3 agonist, binds to BRS-3 with high affinity (mouse Ki = 1.6 nM, human Ki = 25 nM). |
| CSN10525 | Calcipotriol monohydrate | 147657-22-5 | Calcipotriol is a synthetic VitD3 analogue with a high affinity for the vitamin D receptor. |
| CSN10979 | Falecalcitriol | 83805-11-2 | Falecalcitriol is an analog of calcitriol with a higher potency both in vivo and in vitro systems, and longer duration of action in vivo. |
| CSN10729 | Cysteine Protease inhibitor | 921625-62-9 | Cysteine protease inhibitor is an inhibitor of cysteine protease. |
| CSN18585 | Camicinal HCl | 923565-22-4 | GSK962040 HCl is a small molecule, selective motilin receptor agonist with pEC50 of 7.9. |
| CSN10662 | Clebopride malate | 57645-91-7 | Clebopride malate, with antiemetic and prokinetic properties, is a dopamine antagonist drug used to treat gastrointestinal dysfunction. |
| CSN11254 | KN-62 | 127191-97-3 | KN-62 is a selective and potent inhibitor of calmodulin-dependent protein kinase II (CaMK-II) with IC50 of 0.9 μM, KN-62 also displays noncompetitive antagonism at P2X7 receptors in HEK293 cells, with an IC50 value of approximately 15 nM.. |
| CSN18584 | Camicinal | 923565-21-3 | GSK962040 is a small molecule, selective motilin receptor agonist with pEC50 of 7.9. |
| CSN10978 | Fadrozole | 102676-47-1 | Fadrozole is a selective aromatase inhibitor that has been introduced in Japan for the treatment of breast cancer. |
| CSN10374 | Bafilomycin A1 | 88899-55-2 | Bafilomycin A1 is an inhibitor of vacuolar H+-ATPase with IC50 of 0.44 nM. |
| CSN10667 | 2,2'-((Cyclohexane-1,1-diylbis(4,1-phenylene))bis(oxy))bis(2-methylbutanoic acid) | 30299-08-2 | Clinofibrate is a HMG-CoA reductase inhibitor with IC50 value of 470 μM which can reduce plasma cholesterol levels and shows antihyperlipidemic effects. |
| CSN19058 | BMS-779788 | 918348-67-1 | BMS-779788 is a LXR partial agonist with IC50 values of 68 nM for LXRα and 14 nM for LXRβ. |
| CSN22238 | PF-04991532 | 1215197-37-7 | PF-04991532 is a potent, hepatoselective glucokinase activator with EC50s of 80 and 100 nM in human and rat, respectively. |
