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mGluR
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN23124 | Spaglumic Acid | 3106-85-2 | Spaglumic Acid is a neuropeptide found in millimolar concentrations in brain. |
| CSN23116 | SIB 1757 | 31993-01-8 | SIB-1757 is a highly selective antagonist for the mGlu5 metabotropic glutamate receptor subtype. SIB-1757 displays an IC50 value of 0.4 μM at hmGlu5 compared with > 30 μM at hmGlu1b, hmGlu2, hmGlu4, hmGlu6, hmGlu7 and hmGlu8. |
| CSN23187 | VU 29 | 890764-36-0 | Potent positive allosteric modulator of mGlu5 receptors |
| CSN23007 | NPS 2390 | 226878-01-9 | NPS 2390 is a Group I mGlu antagonist. |
| CSN22913 | MMPEP | 823198-78-3 | MPEP HCl is both a selective non-competitive mGlu5 receptor antagonist with IC50 value of 36 nM, and a mGlu4 receptor positive allosteric modulator. |
| CSN18024 | LY354740 | 176199-48-7 | LY354740 is a highly potent, efficacious and selective group II (mGlu2/3) receptor agonist, produces > 90% suppression of forskolin-stimulated cAMP formation with an EC50 of 5.1 ± 0.3 nM. |
| CSN27529 | L-Cysteinesulfinic acid monohydrate | 207121-48-0 | L-Cysteinesulfinic acid monohydrate is a potent agonist at several rat metabotropic glutamate receptors (mGluRs) with pEC50s of 3.92, 4.6, 3.9, 2.7, 4.0, and 3.94 for mGluR1, mGluR5, mGluR2, mGluR4, mGluR6, and mGluR8, respectively. |
| CSN22881 | L-CCG-l | 117857-93-9 | L-CCG-l is a potent group II metabotropic glutamate receptor agonist. |
| CSN23016 | H-Ser(PO3H2)-OH | 407-41-0 | H-Ser(PO3H2)-OH is both a Group III metabotropic glutamate receptor (mGluR4, mGluR7, and mGluR8) agonist, and a competitive NMDA antagonist. |
| CSN22778 | CPPG | 183364-82-1 | CPPG is a potent group II/III mGlu receptor antagonist, with IC50s of 46.2 and 2.2 nM respectively. |