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MMP
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN26232 | UK 356618 | 230961-08-7 | UK-356618 is a matrix metalloproteinase-3 (MMP-3) inhibitor with an IC50 of 5.9 nM. It displays selectivity over a range of MMPs (IC50 values are 73, 840, 1790, 1900 and 51000 for MMP-13, MMP-9, MMP-2, MMP-14 and MMP-1 respectively). |
| CSN19037 | TAPI-2 | 187034-31-7 | TAPI-2 is a broad-spectrum inhibitor of matrix metalloprotease (MMP), tumour necrosis factorα-converting enzyme (TACE) and a disintegrin and metalloproteinase (ADAM), with an IC50 of 20±10 μM for MMP. |
| CSN18802 | (S,S)-TAPI-1 | 171235-71-5 | TAPI-1 is an ADAM17/TACE inhibitor, which blocks shedding of cytokine receptors. |
| CSN17979 | TAPI-1 | 163847-77-6 | TAPI-1 is a specific TACE (TNF-α-converting enzyme) inhibitor. |
| CSN20402 | TACE Inhibitor C3 | 1219812-22-2 | TACE inhibitor C3 is a prodrug of hydantoin based TNF-α converting enzyme (TACE) inhibitor. |
| CSN24080 | T-26c | 869296-13-9 | T-26c is highly potent and selective matrix metalloproteinase-13 (MMP-13) inhibitor with an IC50 of 6.75 pM and more than 2600-fold selectivity over the other related metalloenzymes[1]. |
| CSN23111 | SD 2590 HCl | 226395-93-3 | SD-2590 HCl is an inhibitor of MMP-2,-3, -9, -8, 13, and -14. |
| CSN21234 | S-methyl-KE-298 | 143584-75-2 | S-methyl-KE-298 is an active metabolite of KE-298. KE-298 inhibits matrix metalloproteinase (MMP-1) production from rheumatoid arthritis (RA) synovial cells. |
| CSN21340 | S 3304 | 203640-27-1 | S 3304 is a novel MMP inhibitor. |
| CSN22013 | Prinomastat | 192329-42-3 | Prinomastat is a spectrum inhibitor of MMP with IC50s of 79, 6.3 and 5.0 nM for MMP-1, MMP-3 and MMP-9 respectively. |
| CSN11720 | Pimaric acid | 127-27-5 | Pimaric acid is a natural product isolated and purified from the herbs of Aralia cordata having a potent anti-atherosclerotic activity with inhibitory action on matrix metalloproteinase-9 production and cell migration in TNF-α-induced human aortic smooth muscle cells. |
| CSN19193 | Phosphoramidon Disodium | 164204-38-0 | Phosphoramidon disodium is a metalloendopeptidase inhibitor, widely used as a biochemical tool. |
| CSN19679 | MMP13-IN-2 | 935759-55-0 | MMP13-In-1 is a selective Matrix Metalloproteinase (MMP)-13 inhibitors. |
| CSN25314 | MMP-9-IN-1 | 502887-71-0 | MMP-9-IN-1 is a specific matrix metalloproteinase-9 (MMP-9) inhibitor that selectively targets the hemopexin (PEX) domain of MMP-9. |
| CSN32640 | Tiludronate disodium | 149845-07-8 | MMP-2 (Gelatinase A) Inhibitors, Parathyroid Hormone Receptor Antagonists, Signal Transduction Modulators |
| CSN25429 | JNJ0966 | 315705-75-0 | JNJ0966 is a selective inhibitor of MMP-9 zymogen (IC50 = 440nM) that inhibits subsequent generation of the catalytically active enzyme. It showed no effect on the catalytic activity of MMP-1, MMP-2, MMP-3, MMP-9, or MMP-14, and did not inhibit the activation of MMP-2 zymogen. |
| CSN23138 | T 26c Disodium Salt | 869298-22-6 | Highly potent and selective MMP13 inhibitor |
| CSN19851 | GI254023X | 260264-93-5 | GI 254023X is a potent and selective ADAM10 metalloproteinase inhibitor. |
| CSN10218 | Ethyl gallate | 831-61-8 | Ethyl gallate is a natural product isolated and purifeid from the herbs of Coriaria nepalensis, and it can inhibit the abilities of invasion of breast cancer in vitro by inhibiting the mRNA levels of MMP-9/MMP-2, phosphorylation of Akt and protein expression of NF-κB. |
| CSN23852 | EGTA | 67-42-5 | EGTA is a calcium chelating agent, it's also a useful chemical in a variety of buffers. It also inhibits the zinc-dependent endopeptidases, MMPs. |
| CSN32654 | PKF-241-466 | 205807-58-5 | Disintegrin and Metalloproteinase Domain-Containing Protein 17 (ADAM17; TACE) Inhibitors, MMP-1 (Interstitial Collagenase) Inhibitors, MMP-13 (Collagenase 3) Inhibitors, MMP-2 (Gelatinase A) Inhibitors, MMP-9 (Gelatinase B) Inhibitors, Signal Transduction Modulators |
| CSN32653 | TMI-1 | 287403-39-8 | Disintegrin and Metalloproteinase Domain-Containing Protein 17 (ADAM17; TACE) Inhibitors, MMP-1 (Interstitial Collagenase) Inhibitors, MMP-13 (Collagenase 3) Inhibitors, MMP-2 (Gelatinase A) Inhibitors, MMP-7 (Matrilysin) Inhibitors, MMP-9 (Gelatinase B) Inhibitors, Signal Transduction Modulators |
| CSN32655 | PKF-242-484 | 205807-59-6 | Disintegrin and Metalloproteinase Domain-Containing Protein 17 (ADAM17; TACE) Inhibitors, MMP-1 (Interstitial Collagenase) Inhibitors, MMP-13 (Collagenase 3) Inhibitors, MMP-2 (Gelatinase A) Inhibitors, MMP-3 (Stromelysin 1) Inhibitors, MMP-9 (Gelatinase B) Inhibitors, Signal Transduction Modulators |
| CSN18069 | CTS-1027 | 193022-04-7 | CTS-1027 is a potent small molecule inhibitor of MMPs (IC50=0.4 nM/0.6 nM for MMP2/MMP13), displaying > 1,000 fold selectivity over MMP1. |
| CSN26236 | ARP-100 | 704888-90-4 | ARP-100 is a potent and selective matrix metalloproteinase MMP-2 inhibitor (IC50=12 nM). |
| CSN32647 | 4-(Dodecylamino)phenol | 25848-37-7 | Antioxidants, Apoptosis Inducers, Free Radical Scavengers, Lipid Peroxidation Inhibitors, MMP-2 (Gelatinase A) Inhibitors, MMP-9 (Gelatinase B) Inhibitors |
| CSN32641 | Incyclinide | 15866-90-7 | Angiogenesis Inhibitors, MMP-2 (Gelatinase A) Inhibitors, MMP-9 (Gelatinase B) Inhibitors, Signal Transduction Modulators, Vascular Endothelial Growth Factor (VEGF) Inhibitors |
| CSN32643 | ABT-518 | 286845-00-9 | Angiogenesis Inhibitors, MMP-2 (Gelatinase A) Inhibitors, MMP-9 (Gelatinase B) Inhibitors |
| CSN32644 | CGS 27023A free | 161314-70-1 | Angiogenesis Inhibitors, MMP-2 (Gelatinase A) Inhibitors, MMP-8 (Neutrophil Collagenase) Inhibitors, MMP-9 (Gelatinase B) Inhibitors |
| CSN32642 | CGS 27023A hydrochloride | 169799-04-6 | Angiogenesis Inhibitors, MMP-2 (Gelatinase A) Inhibitors, MMP-8 (Neutrophil Collagenase) Inhibitors, MMP-9 (Gelatinase B) Inhibitors |
| CSN32645 | Tanomastat | 179545-77-8 | Angiogenesis Inhibitors, MMP-2 (Gelatinase A) Inhibitors, MMP-3 (Stromelysin 1) Inhibitors, MMP-9 (Gelatinase B) Inhibitors |
| CSN19813 | Aderbasib | 791828-58-5 | Aderbasib is a sheddase inhibitor, is also an orally bioavailable inhibitor of the ADAM (A disintegrin and metalloprotease) family of multifunctional membrane-bound proteins with potential antineoplastic activity. |
| CSN20301 | ADAMTS Inhibitor C7 | 1607004-34-1 | ADAMTS inhibitor C7 is an inhibitor of aggrecanase 1 and 2 (ADAMTS-4 and ADAMTS-5) had good oral pharmacokinetics in rats and showed efficacy in a rat chemical model of os-teoarthritis. |
| CSN24958 | Abametapir | 1762-34-1 | Abametapir is the active ingredient of Xeglyze Lotion. Abametapir inhibits metalloproteinases; enzymes that are essential to physiological processes critical for egg development and the survival of nymph and adult lice. In vitro and ex vivo research has demonstrated that abametapir not only kills the lice, but also prevents hatching of their eggs. Xeglyze Lotion is emerging as a differentiated development candidate to treat head lice infestations. |
| CSN29447 | PD-166793 | 199850-67-4 | Broad spectrum MMP inhibitor |
| CSN26955 | Palmitoyl Tripeptide-5 TFA | 623172-56-5 | |
| CSN33198 | GW280264X | 866924-39-2 | |
| CSN39987 | Apratastat | 287405-51-0 | |
| CSN42022 | ADAMTS-5 Inhibitor | 929634-33-3 | |
| CSN39089 | ZLDI-8 | 667880-38-8 | |
| CSN68121 | Aldumastat | 1957278-93-1 | |
| CSN75578 | WAY-170523 | 307002-73-9 | |
| CSN79104 | ADAMTS-5-IN-3 | 2688733-96-0 | |
| CSN77766 | JG26 | 1464910-32-4 | |
| CSN80889 | TAPI-0 | 163958-73-4 | |
| CSN83124 | TAPI | 143457-40-3 | |
| CSN84053 | Imidapril | 89371-37-9 | |
| CSN84136 | PPNDS tetrasodium | 1021868-77-8 | |
| CSN105563 | (3R,4R)-N-Hydroxy-4-(4-((2-(trifluoromethyl)-1H-benzo[d]imidazol-1-yl)methyl)benzamido)tetrahydro-2H-pyran-3-carboxamide | 503166-51-6 | |
| CSN107659 | (R)-N1-((S)-1-(((S)-1-((2-Aminoethyl)amino)-1-oxopropan-2-yl)amino)-3,3-dimethyl-1-oxobutan-2-yl)-N4-hydroxy-2-isobutylsuccinamide | 689284-12-6 |
