货号 | 产品名 | CAS号 | 信息 |
---|---|---|---|
CSN22437 | JNJ-46778212 | 1363281-27-9 | JNJ-46778212 is an mGlu5 positive allosteric modulator with an EC50 of 260 nM. |
CSN22374 | CI-943 | 89239-35-0 | CI-943 is a potential antipsychotic agent. |
CSN22241 | NBQX | 118876-58-7 | NBQX is a potent, selective and competitive AMPAR antagonist, which shows activity of neuroprotective and anticonvulsant. |
CSN22445 | L-APB | 23052-81-5 | L-APB is a potent and specific agonist for the group III mGluRs, with EC50s of 0.13±0.02, 0.29±0.07, 1.0±0.3, 249±107 μM for mGlu4, mGlu8, mGlu6 and mGlu7 receptors, respectively. |
CSN22913 | MMPEP | 823198-78-3 | MPEP HCl is both a selective non-competitive mGlu5 receptor antagonist with IC50 value of 36 nM, and a mGlu4 receptor positive allosteric modulator. |
CSN22187 | W-2429 | 37795-69-0 | W-2429 is a non-narcotic analgesic agent. |
CSN22216 | NS1652 | 1566-81-0 | NS1652 is a reversible anion conductance inhibitor, blocks chloride channel, with an IC50 of 1.6 μM in human and mouse red blood cells. |
CSN22401 | Fluxametamide | 928783-29-3 | Fluxametamide is an insecticide with wide spectrum, acts as an antagonist of GABA- and glutamate-gated chloride channels, with IC50 of 1.95 nM and 225 nM for M. domestica GABACls and GluCls. |
CSN22323 | (+)-Dihydrexidine HCl | 158704-02-0 | (+)-Dihydrexidine HCl is a dopamine D1 receptor agonist with an EC50 of 72± 21 nM. |
CSN22469 | MSOP | 66515-29-5 | MSOP is a selective group III metabotropic glutamate receptor antagonist with apparent KD of 51 μM for the L-AP4-sensitive presynaptic mGluR. |
CSN22538 | β-Secretase Inhibitor IV | 797035-11-1 | β-Secretase Inhibitor IV is a potent, cell-active BACE-1 inhibitor with IC50s of 15.6 and 16.3nM under BACE-1 concentrations of 2 nM and 100 pM, respectively. |
CSN23242 | Cyromazin | 66215-27-8 | Cyromazine is a triazine insecticide and an acaricide. |