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| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN22437 | JNJ-46778212 | 1363281-27-9 | JNJ-46778212 is an mGlu5 positive allosteric modulator with an EC50 of 260 nM. |
| CSN22348 | AP521 | 151227-08-6 | AP521 is an agonist of human 5-HT1A receptor with an IC50 of 94 nM. |
| CSN22374 | CI-943 | 89239-35-0 | CI-943 is a potential antipsychotic agent. |
| CSN22450 | Lurasidone Metabolite 14283 HCl | 186204-32-0 | Lurasidone Metabolite 14283 HCl is a major active metabolite of Lurasidone. Lurasidone is a FDA approved drug for the treatment of schizophrenia. |
| CSN22241 | NBQX | 118876-58-7 | NBQX is a potent, selective and competitive AMPAR antagonist, which shows activity of neuroprotective and anticonvulsant. |
| CSN22445 | L-APB | 23052-81-5 | L-APB is a potent and specific agonist for the group III mGluRs, with EC50s of 0.13±0.02, 0.29±0.07, 1.0±0.3, 249±107 μM for mGlu4, mGlu8, mGlu6 and mGlu7 receptors, respectively. |
| CSN22913 | MMPEP | 823198-78-3 | MPEP HCl is both a selective non-competitive mGlu5 receptor antagonist with IC50 value of 36 nM, and a mGlu4 receptor positive allosteric modulator. |
| CSN22503 | Saredutant | 142001-63-6 | Saredutant is a selective NK2 receptor antagonist. |
| CSN22192 | AR-A 2 | 220051-79-6 | AR-A 2 is a selective 5-HT1B receptor antagonist, with high affinity to guinea pig cortex 5HT1B/1D and recombinant guinea pig 5-HT1B receptors (Ki=0.24 and 0.47 nM) and with 10-fold lower affinity to guinea pig 5-HT1D receptor (Ki=5 nM), and shows an EC50 of 4.5 nM for the guinea pig 5-HT1B receptor; AR-A 2 can be used in the research of depression and anxiety. |
| CSN22187 | W-2429 | 37795-69-0 | W-2429 is a non-narcotic analgesic agent. |
| CSN22216 | NS1652 | 1566-81-0 | NS1652 is a reversible anion conductance inhibitor, blocks chloride channel, with an IC50 of 1.6 μM in human and mouse red blood cells. |
| CSN22325 | (+)-Phenserine | 116839-68-0 | Posiphen is a selective cholinesterase noncompetitive inhibitor with an IC50 of 45.3 μM. |
| CSN22401 | Fluxametamide | 928783-29-3 | Fluxametamide is an insecticide with wide spectrum, acts as an antagonist of GABA- and glutamate-gated chloride channels, with IC50 of 1.95 nM and 225 nM for M. domestica GABACls and GluCls. |
| CSN22323 | (+)-Dihydrexidine HCl | 158704-02-0 | (+)-Dihydrexidine HCl is a dopamine D1 receptor agonist with an EC50 of 72± 21 nM. |
| CSN22396 | Eplivanserin | 130579-75-8 | Eplivanserin is a potent, selective and orally available 5-HT2 receptor antagonist, with an IC50 of 5.8 nM in rat cortical membrane, and a Kd of 1.14 nM. |
| CSN22469 | MSOP | 66515-29-5 | MSOP is a selective group III metabotropic glutamate receptor antagonist with apparent KD of 51 μM for the L-AP4-sensitive presynaptic mGluR. |
| CSN22538 | β-Secretase Inhibitor IV | 797035-11-1 | β-Secretase Inhibitor IV is a potent, cell-active BACE-1 inhibitor with IC50s of 15.6 and 16.3nM under BACE-1 concentrations of 2 nM and 100 pM, respectively. |
| CSN23242 | Cyromazin | 66215-27-8 | Cyromazine is a triazine insecticide and an acaricide. |
