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NMDAR
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN21328 | UK-240455 | 178908-09-3 | UK-240455 is a potent and selective N-methyl D-aspartate (NMDA) glycine site antagonist. |
| CSN12978 | Traxoprodil | 134234-12-1 | Traxoprodil a selective antagonist of the NR2B subunit of the NMDA receptor. |
| CSN24287 | Traxoprodil mesylate | 189894-57-3 | Traxoprodil a selective antagonist of the NR2B subunit of the NMDA receptor. |
| CSN11907 | SDZ 220-581 | 174575-17-8 | SDZ 220-581 is a potent, competitive antagonist at the NMDA glutamate receptor subtype (pKi= 7.7). |
| CSN15699 | Sarcosine | 107-97-1 | Sarcosine is an NMDAR co-agonist at the glycine binding site. It is an intermediate and byproduct in glycine synthesis and degradation. |
| CSN17353 | Ro 25-6981 | 169274-78-6 | Ro 25-6981 is a potent and selective activity-dependent blocker of NMDA receptors containing the NR2B subunit. |
| CSN17520 | Rapastinel | 117928-94-6 | Rapastinel is a putative NMDAR functional glycine-site partial agonist. |
| CSN23784 | Radiprodil | 496054-87-6 | Radiprodil is a selective antagonist of NMDA NR2B that used in treatment of neuropathic pain. |
| CSN23523 | Quinolinic acid | 89-00-9 | Quinolinic acid is both a selective agonist at NMDA receptors and also a precursor for the formation of NAD+. |
| CSN16857 | QNZ46 | 1237744-13-6 | QNZ46 is a noncompetitive and voltage-independent GluN2C/GluN2D-selective NMDA antagonist with IC50 values of 3, 6, 229 μM for GluN2D, GluN2C, GluN2A, respectively. |
| CSN11780 | Procyclidine HCl | 1508-76-5 | Procyclidine HCl is an potent anti-cholinergic agent, and is also known to have NMDA antagonist properties. |
| CSN11639 | Oxysophoridine | 54809-74-4 | Oxysophoridine is a natural product isolated and purified from the herb of Sophora alopecuroidos L. Oxysophoridine inhibited N-methyl-D-aspartate NR1 mRNA and protein expression in the cerebral cortex of mice with cerebral ischemia/reperfusion injury. |
| CSN11619 | Orphenadrine HCl | 341-69-5 | Orphenadrine HCl is an uncompetitive N-methyl-D-aspartate (NMDA) receptor antagonist with Ki of 6.0 ±0.7 μM. |
| CSN11618 | Orphenadrine Citrate | 4682-36-4 | Orphenadrine Citrate is both an uncompetitive NMDA receptor antagonist IC50 value of 16.2 µM and a mAChR antagonist with IC50 value of 0.37 µM. |
| CSN13790 | NMDA | 6384-92-5 | NMDA is an amino acid derived specific agonist at the NMDA receptor. |
| CSN11379 | Mephenesin | 59-47-2 | Mephenesin is a centrally acting muscle relaxant which may work as an NMDA receptor antagonist. |
| CSN11501 | Memantine | 19982-08-2 | Memantine is the first in a class of Alzheimer's disease medications acting on the glutamatergic system by blocking NMDA receptors. |
| CSN13695 | MDL-29951 | 130798-51-5 | MDL-29951 is a glycine antagonist of NMDA receptor activation (Ki=0.14 mM, [3H]glycine binding) in vitro and in vivo. |
| CSN20030 | Lanicemine | 153322-05-5 | Lanicemine is a low-trapping NMDA receptor antagonist. Lanicemine is used the management of severe and treatment-resistant depression. Lanicemine was originally developed as a neuroprotective agent, but was redeveloped as an antidepressant. |
| CSN17128 | L-701,324 | 142326-59-8 | L-701324 is an orally active and long acting anticonvulsant with high affinity and selectivity for the glycine site on the NMDA receptor. |
| CSN11186 | Ifenprodil Tartrate | 23210-58-4 | Ifenprodil Tartrate is a high affinity and atypical noncompetitive NMDA receptor antagonist with IC50 of 0.3 μM. |
| CSN21125 | Ibotenic Acid | 2552-55-8 | Ibotenic acid has agonist activity at both the N-methyl-D-aspartate (NMDA) and trans-ACPD or metabolotropic quisqualate (Qm) receptor sites. |
| CSN10988 | Felbamate | 25451-15-4 | Felbamate is a potent nonsedative anticonvulsant whose clinical effect may be related to the inhibition of N-methyl-D-aspartate (NMDA) . |
| CSN10256 | Eliprodil | 119431-25-3 | Eliprodil can antogonize GluN2B-selective NMDA in a non-competitive manner with IC50 value of 1 μM. It is also a σ1 ligand with Ki value of 0.013 μM. |
| CSN10502 | Budipine | 57982-78-2 | Budipine is an uncompetitive NMDAR antagonist used as an antiparkinson agent. |
| CSN24923 | 6-Methoxy-2-naphthoic acid | 2471-70-7 | 6-Methoxy-2-naphthoic acid is an modulator of NMDAR. |
| CSN25440 | ACBC | 22264-50-2 | 1-Aminocyclobutanecarboxylic acid is a NMDA receptor partial agonist acting at the glycine site, NR1. |
| CSN23429 | L-Glutamic Acid | 56-86-0 | (S)-Glutamic acid acts as an excitatory neurotransmitter in the central nervous system. |
| CSN25441 | (-)-Aspartic acid | 1783-96-6 | (-)-Aspartic acid is an endogenous NMDA receptor agonist. |
| CSN13883 | (+)-MK 801 Maleate | 77086-22-7 | (+)-MK 801 Maleate is a highly potent, selective and non-competitive NMDA receptor antagonist with Ki of 30.5 nM. |