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NMDAR
货号 | 产品名 | CAS号 | 信息 |
---|---|---|---|
CSN12978 | Traxoprodil | 134234-12-1 | Traxoprodil a selective antagonist of the NR2B subunit of the NMDA receptor. |
CSN11907 | SDZ 220-581 | 174575-17-8 | SDZ 220-581 is a potent, competitive antagonist at the NMDA glutamate receptor subtype (pKi= 7.7). |
CSN11780 | Procyclidine HCl | 1508-76-5 | Procyclidine HCl is an potent anti-cholinergic agent, and is also known to have NMDA antagonist properties. |
CSN11619 | Orphenadrine HCl | 341-69-5 | Orphenadrine HCl is an uncompetitive N-methyl-D-aspartate (NMDA) receptor antagonist with Ki of 6.0 ±0.7 μM. |
CSN11618 | Orphenadrine citrate | 4682-36-4 | Orphenadrine Citrate is both an uncompetitive NMDA receptor antagonist IC50 value of 16.2 µM and a mAChR antagonist with IC50 value of 0.37 µM. |
CSN11379 | Mephenesin | 59-47-2 | Mephenesin is a centrally acting muscle relaxant which may work as an NMDA receptor antagonist. |
CSN11501 | Memantine | 19982-08-2 | Memantine is the first in a class of Alzheimer's disease medications acting on the glutamatergic system by blocking NMDA receptors. |
CSN13695 | MDL-29951 | 130798-51-5 | MDL-29951 is a glycine antagonist of NMDA receptor activation (Ki=0.14 mM, [3H]glycine binding) in vitro and in vivo. |
CSN11186 | 4-(2-(4-Benzylpiperidin-1-yl)-1-hydroxypropyl)phenol hemi((2R,3R)-2,3-dihydroxysuccinate) | 23210-58-4 | Ifenprodil Tartrate is a high affinity and atypical noncompetitive NMDA receptor antagonist with IC50 of 0.3 μM. |
CSN10988 | 2-Phenylpropane-1,3-diyl dicarbamate | 25451-15-4 | Felbamate is a potent nonsedative anticonvulsant whose clinical effect may be related to the inhibition of N-methyl-D-aspartate (NMDA) . |
CSN10256 | Eliprodil | 119431-25-3 | Eliprodil can antogonize GluN2B-selective NMDA in a non-competitive manner with IC50 value of 1 μM. It is also a σ1 ligand with Ki value of 0.013 μM. |
CSN10502 | Budipine | 57982-78-2 | Budipine is an uncompetitive NMDAR antagonist used as an antiparkinson agent. |