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Opioid Receptor

Opioid Receptor

货号 产品名 CAS号 信息
CSN22049 [Met5]-Enkephalin Amide 60117-17-1 [Met5]-Enkephalin, amide is an agonist for δ opioid receptors as well as putative ζ (zeta) opioid receptors.
CSN21444 [Leu5]-Enkephalin 58822-25-6 [Leu5]-Enkephalin, an endogenous opioid neurotransmitter or neuromodulator, is an agonist of µ and δ opioid receptors.
CSN18678 [D-Ala2]Leucine-Enkephalin 64963-01-5 [D-Ala2]Leucine-Enkephalin is a potent, long-acting Leu-enkephalin analog agonist of delta opioid receptor.
CSN26718 SB-612111 371980-98-2 SB-612111 is a novel and potent human opiate receptor-like orphan receptor (ORL-1) antagonist with a high affinity for hORL-1 (Ki=0.33 nM). SB-612111 exhibits selectivity for μ-, κ- and δ-receptors with Ki values of 57.6 nM, 160.5 nM and 2109 nM, respecticely. SB-612111 effectively antagonizes the pronociceptive action of Nociceptin (HY-P0183) in an acute pain model[1].
CSN12166 Porcine Dynorphin A(1-13) 72957-38-1 Porcine dynorphin A(1-13) is a potent, endogenous κ-agonist.
CSN22475 ORL1 Antagonist 1 1174985-59-1 ORL1 antagonist 1 is an opioid receptor-like 1 (ORL1) antagonist with an IC50 of 61 nM.
CSN21766 Nociceptin 170713-75-4 Nociceptin, a 17 amino acid neuropeptide, is endogenous ligand for the opioid-like G-protein coupled receptor, ORL1 (opioid receptor-like 1).
CSN16622 JTC-801 244218-51-7 JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, and weakly inhibits receptors δ, κ, and μ.
CSN16488 JDTic 361444-66-8 JDTic is a highly selective antagonist for the κ-opioid receptor and without affecting the μ- or δ-opioid receptors.
CSN18435 JDTic 2HCl 785835-79-2 JDTic 2HCl is a highly selective antagonist for the κ-opioid receptor without affecting the μ- or δ-opioid receptors.
CSN21596 Gluten Exorphin C 142479-62-7 Gluten exorphin C, an opioid peptide derived from wheat gluten, can inhibit μ opioid and δ opioid with IC50 values of 40 μM and 13.5 μM in the GPI and MVD assays.
CSN21628 Endomorphin 2 141801-26-5 Endomorphin 2, an endogenous neuropeptide, is agonist of μ-opioid receptor with Ki of 0.69 nM that has analgesic and gastrointestinal properties.
CSN21627 Endomorphin 1 189388-22-5 Endomorphin 1 is a selective agonist of μ-opioid receptor with reasonable affinities for kappa3 binding sites (Ki value between 20 and 30 nM).
CSN21597 Deltorphin I 122752-15-2 Deltorphin I is a selective agonist of δ-opioid receptor.
CSN21598 Deltorphin 2 122752-16-3 Deltorphin 2 is selective δ2 opioid receptor agonist.
CSN25444 BRL 52537 hydrochloride 112282-24-3 BRL-52537 hydrochloride is a potent and highly selective κ-opioid agonist. It has neuroprotective effects in animal studies, and is used for research into potential treatments for stroke and heart attack as well as more general brain research.
CSN17791 BAN ORL 24 1401463-54-4 BAN ORL 24 is a potent and selective NOP receptor antagonist. (IC50 values are 0.27, 2500, 6700 and > 10000 nM for NOP, κ-, μ- and δ-receptors respectively).
CSN24259 BAN ORL 24diHCl- 475150-69-7 BAN ORL 24 is a potent and selective NOP receptor antagonist. (IC50 values are 0.27, 2500, 6700 and > 10000 nM for NOP, κ-, μ- and δ-receptors respectively).
CSN21495 Asimadoline 153205-46-0 Asimadoline is an agonist of κ-opioid receptor (KOR) with IC50 of 1.2 nM.
CSN23662 AR-M 1000390 HCl 209808-47-9 AR-M 1000390 HCl is a non-peptidic and low-internalizing δ-selective opioid receptor agonist.
CSN17774 Alvimopan Monohydrate 1383577-62-5 Alvimopan is a peripherally acting mu-opioid receptor (PAM-OR, IC50= 1.7 nM) antagonist for accelerating gastrointestinal recovery after surgery.
CSN19330 (+)-Matrine 519-02-8 (+)-Matrine is a naturally occuring κ-opioid and μ-opioid receptor agonist.
CSN29545 SNC 80 156727-74-1 Highly selective non-peptide δ agonist
CSN27869 SCH 32615 83861-02-3
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