优势价格
快速发货
品质保证
技术支持
400-920-2911 sales@csnpharm.cn
Opioid Receptor
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN22049 | [Met5]-Enkephalin Amide | 60117-17-1 | [Met5]-Enkephalin, amide is an agonist for δ opioid receptors as well as putative ζ (zeta) opioid receptors. |
| CSN21444 | [Leu5]-Enkephalin | 58822-25-6 | [Leu5]-Enkephalin, an endogenous opioid neurotransmitter or neuromodulator, is an agonist of µ and δ opioid receptors. |
| CSN18678 | [D-Ala2]Leucine-Enkephalin | 64963-01-5 | [D-Ala2]Leucine-Enkephalin is a potent, long-acting Leu-enkephalin analog agonist of delta opioid receptor. |
| CSN26718 | SB-612111 | 371980-98-2 | SB-612111 is a novel and potent human opiate receptor-like orphan receptor (ORL-1) antagonist with a high affinity for hORL-1 (Ki=0.33 nM). SB-612111 exhibits selectivity for μ-, κ- and δ-receptors with Ki values of 57.6 nM, 160.5 nM and 2109 nM, respecticely. SB-612111 effectively antagonizes the pronociceptive action of Nociceptin (HY-P0183) in an acute pain model[1]. |
| CSN12166 | Porcine Dynorphin A(1-13) | 72957-38-1 | Porcine dynorphin A(1-13) is a potent, endogenous κ-agonist. |
| CSN22475 | ORL1 Antagonist 1 | 1174985-59-1 | ORL1 antagonist 1 is an opioid receptor-like 1 (ORL1) antagonist with an IC50 of 61 nM. |
| CSN21766 | Nociceptin | 170713-75-4 | Nociceptin, a 17 amino acid neuropeptide, is endogenous ligand for the opioid-like G-protein coupled receptor, ORL1 (opioid receptor-like 1). |
| CSN16622 | JTC-801 | 244218-51-7 | JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, and weakly inhibits receptors δ, κ, and μ. |
| CSN16488 | JDTic | 361444-66-8 | JDTic is a highly selective antagonist for the κ-opioid receptor and without affecting the μ- or δ-opioid receptors. |
| CSN18435 | JDTic 2HCl | 785835-79-2 | JDTic 2HCl is a highly selective antagonist for the κ-opioid receptor without affecting the μ- or δ-opioid receptors. |
| CSN21596 | Gluten Exorphin C | 142479-62-7 | Gluten exorphin C, an opioid peptide derived from wheat gluten, can inhibit μ opioid and δ opioid with IC50 values of 40 μM and 13.5 μM in the GPI and MVD assays. |
| CSN21628 | Endomorphin 2 | 141801-26-5 | Endomorphin 2, an endogenous neuropeptide, is agonist of μ-opioid receptor with Ki of 0.69 nM that has analgesic and gastrointestinal properties. |
| CSN21627 | Endomorphin 1 | 189388-22-5 | Endomorphin 1 is a selective agonist of μ-opioid receptor with reasonable affinities for kappa3 binding sites (Ki value between 20 and 30 nM). |
| CSN21597 | Deltorphin I | 122752-15-2 | Deltorphin I is a selective agonist of δ-opioid receptor. |
| CSN21598 | Deltorphin 2 | 122752-16-3 | Deltorphin 2 is selective δ2 opioid receptor agonist. |
| CSN25444 | BRL 52537 hydrochloride | 112282-24-3 | BRL-52537 hydrochloride is a potent and highly selective κ-opioid agonist. It has neuroprotective effects in animal studies, and is used for research into potential treatments for stroke and heart attack as well as more general brain research. |
| CSN17791 | BAN ORL 24 | 1401463-54-4 | BAN ORL 24 is a potent and selective NOP receptor antagonist. (IC50 values are 0.27, 2500, 6700 and > 10000 nM for NOP, κ-, μ- and δ-receptors respectively). |
| CSN24259 | BAN ORL 24diHCl- | 475150-69-7 | BAN ORL 24 is a potent and selective NOP receptor antagonist. (IC50 values are 0.27, 2500, 6700 and > 10000 nM for NOP, κ-, μ- and δ-receptors respectively). |
| CSN21495 | Asimadoline | 153205-46-0 | Asimadoline is an agonist of κ-opioid receptor (KOR) with IC50 of 1.2 nM. |
| CSN23662 | AR-M 1000390 HCl | 209808-47-9 | AR-M 1000390 HCl is a non-peptidic and low-internalizing δ-selective opioid receptor agonist. |
| CSN17774 | Alvimopan Monohydrate | 1383577-62-5 | Alvimopan is a peripherally acting mu-opioid receptor (PAM-OR, IC50= 1.7 nM) antagonist for accelerating gastrointestinal recovery after surgery. |
| CSN19330 | (+)-Matrine | 519-02-8 | (+)-Matrine is a naturally occuring κ-opioid and μ-opioid receptor agonist. |
| CSN29545 | SNC 80 | 156727-74-1 | Highly selective non-peptide δ agonist |
| CSN27869 | SCH 32615 | 83861-02-3 |
