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Opioid Receptor
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN21444 | [Leu5]-Enkephalin | 58822-25-6 | [Leu5]-Enkephalin, an endogenous opioid neurotransmitter or neuromodulator, is an agonist of µ and δ opioid receptors. |
| CSN20210 | Trv0109101 | 1401027-29-9 | TRV0109101, a G protein-biased agonist of the µ-opioid receptor, which may be an effective therapeutic avenue for managing chronic pain with reduced propensity for opioid-induced hyperalgesia. |
| CSN20211 | TRV0109101 Hydrochloride | 2101210-22-2 | TRV0109101 HCl, a G protein-biased agonist of the µ-opioid receptor, which may be an effective therapeutic avenue for managing chronic pain with reduced propensity for opioid-induced hyperalgesia. |
| CSN26718 | SB-612111 | 371980-98-2 | SB-612111 is a novel and potent human opiate receptor-like orphan receptor (ORL-1) antagonist with a high affinity for hORL-1 (Ki=0.33 nM). SB-612111 exhibits selectivity for μ-, κ- and δ-receptors with Ki values of 57.6 nM, 160.5 nM and 2109 nM, respecticely. SB-612111 effectively antagonizes the pronociceptive action of Nociceptin (HY-P0183) in an acute pain model[1]. |
| CSN21214 | PZM21 | 1997387-43-5 | PZM21 is a potent and selective μ opioid receptor agonist with an EC50 of 1.8 nM. |
| CSN12166 | Porcine dynorphin A(1-13) | 72957-38-1 | Porcine dynorphin A(1-13) is a potent, endogenous κ-agonist. |
| CSN21766 | Nociceptin | 170713-75-4 | Nociceptin, a 17 amino acid neuropeptide, is endogenous ligand for the opioid-like G-protein coupled receptor, ORL1 (opioid receptor-like 1). |
| CSN26717 | LY2940094 | 1307245-86-8 | LY2940094 is a potent and selective nociceptin receptor antagonist which inhibits excessive feeding behavior in rodents. |
| CSN20227 | LY2444296 | 1346133-11-6 | LY2444296 is a short-acting kappa opioid receptor antagonist. |
| CSN23719 | LY2940094 tartrate | 1307245-87-9 | LY-2940094 tartrate is the tartrate form of LY-2940094 which is an antagonist of nociceptin receptor that is used for the treatment of major depressive disorder and alcoholism. |
| CSN20601 | Aticaprant | 1174130-61-0 | LY-2456302 is a potent and centrally-penetrant kappa opioid receptor antagonist with a Ki of 0.807 nM. |
| CSN21596 | Gluten Exorphin C | 142479-62-7 | Gluten exorphin C, an opioid peptide derived from wheat gluten, can inhibit μ opioid and δ opioid with IC50 values of 40 μM and 13.5 μM in the GPI and MVD assays. |
| CSN21628 | Endomorphin 2 | 141801-26-5 | Endomorphin 2, an endogenous neuropeptide, is agonist of μ-opioid receptor with Ki of 0.69 nM that has analgesic and gastrointestinal properties. |
| CSN21627 | Endomorphin 1 | 189388-22-5 | Endomorphin 1 is a selective agonist of μ-opioid receptor with reasonable affinities for kappa3 binding sites (Ki value between 20 and 30 nM). |
| CSN35445 | Difelikefalin | 1024828-77-0 | Difelikefalin (CR-845; FE-202845) is a peripherally restricted and selective agonist of kappa opioid receptor (KOR). Difelikefalin produces anti-inflammatory effects and has the potential in modulating pruritus in conditions such as chronic kidney disease. |
| CSN21597 | Deltorphin I | 122752-15-2 | Deltorphin I is a selective agonist of δ-opioid receptor. |
| CSN22567 | DAMGO | 78123-71-4 | DAMGO is a highly selective peptide agonist for the μ opioid receptor. |
| CSN33173 | Navacaprant | 2244614-14-8 | BTRX-335140 is a potent and selective KOR antagonist with IC50 (KOR)=0.8 nM. |
| CSN25444 | BRL 52537 hydrochloride | 112282-24-3 | BRL-52537 hydrochloride is a potent and highly selective κ-opioid agonist. It has neuroprotective effects in animal studies, and is used for research into potential treatments for stroke and heart attack as well as more general brain research. |
| CSN27537 | Bevenopran | 676500-67-7 | Bevenopran is a peripheral μ-opioid receptor antagonist. |
| CSN24259 | (R)-N-(3-(3H-Spiro[isobenzofuran-1,4'-piperidin]-1'-yl)propyl)-1-benzylpyrrolidine-2-carboxamide | 475150-69-7 | BAN ORL 24 is a potent and selective NOP receptor antagonist. (IC50 values are 0.27, 2500, 6700 and > 10000 nM for NOP, κ-, μ- and δ-receptors respectively). |
| CSN21495 | Asimadoline | 153205-46-0 | Asimadoline is an agonist of κ-opioid receptor (KOR) with IC50 of 1.2 nM. |
| CSN23662 | AR-M 1000390 hydrochloride | 209808-47-9 | AR-M 1000390 HCl is a non-peptidic and low-internalizing δ-selective opioid receptor agonist. |
| CSN27869 | SCH 32615 | 83861-02-3 | |
| CSN41142 | Dynorphin A | 80448-90-4 | |
| CSN40048 | Allomatrine | 641-39-4 | |
| CSN36635 | β-Endorphin, human | 61214-51-5 | |
| CSN36630 | Endomorphin 2 TFA | 1276124-00-5 | |
| CSN33751 | CTOP | 103429-31-8 | |
| CSN35755 | Dermorphin | 77614-16-5 | |
| CSN63176 | DIPPA hydrochloride | 155512-52-0 | |
| CSN63462 | BMS-986122 | 313669-88-4 | |
| CSN75683 | ICI 199441 | 115199-84-3 | |
| CSN75308 | Acetyl tetrapeptide-15 | 928007-64-1 | |
| CSN80506 | AT-076 | 1657028-64-2 | |
| CSN81431 | ML138 | 1355243-24-1 | |
| CSN104006 | rel-4-((R)-((2S,5R)-4-allyl-2,5-dimethylpiperazin-1-yl)(3-hydroxyphenyl)methyl)-N,N-diethylbenzamide | 150428-54-9 | |
| CSN102444 | N,N-Diethyl-3-hydroxy-4-(spiro[chromene-2,4'-piperidin]-4-yl)benzamide | 850176-30-6 | |
| CSN104190 | (2S,5S,14S)-15-Allyl-5-benzyl-14-(4-hydroxybenzyl)-2-isobutyl-8,8,11,11-tetramethyl-4,7,10,13-tetraoxo-3,6,9,12,15-pentaazaoctadec-17-en-1-oic acid | 92535-15-4 | |
| CSN107811 | 2-Methyl-N-((2'-(pyrrolidin-1-ylsulfonyl)-[1,1'-biphenyl]-4-yl)methyl)propan-1-amine hydrochloride | 1322001-35-3 |
