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Opioid Receptor

Opioid Receptor

货号 产品名 CAS号 信息
CSN21444 [Leu5]-Enkephalin 58822-25-6 [Leu5]-Enkephalin, an endogenous opioid neurotransmitter or neuromodulator, is an agonist of µ and δ opioid receptors.
CSN20210 TRV0109101 1401027-29-9 TRV0109101, a G protein-biased agonist of the µ-opioid receptor, which may be an effective therapeutic avenue for managing chronic pain with reduced propensity for opioid-induced hyperalgesia.
CSN20211 TRV0109101 HCl 2101210-22-2 TRV0109101 HCl, a G protein-biased agonist of the µ-opioid receptor, which may be an effective therapeutic avenue for managing chronic pain with reduced propensity for opioid-induced hyperalgesia.
CSN26718 SB-612111 371980-98-2 SB-612111 is a novel and potent human opiate receptor-like orphan receptor (ORL-1) antagonist with a high affinity for hORL-1 (Ki=0.33 nM). SB-612111 exhibits selectivity for μ-, κ- and δ-receptors with Ki values of 57.6 nM, 160.5 nM and 2109 nM, respecticely. SB-612111 effectively antagonizes the pronociceptive action of Nociceptin (HY-P0183) in an acute pain model[1].
CSN21214 PZM21 1997387-43-5 PZM21 is a potent and selective μ opioid receptor agonist with an EC50 of 1.8 nM.
CSN12166 Porcine dynorphin A(1-13) 72957-38-1 Porcine dynorphin A(1-13) is a potent, endogenous κ-agonist.
CSN21766 Nociceptin 170713-75-4 Nociceptin, a 17 amino acid neuropeptide, is endogenous ligand for the opioid-like G-protein coupled receptor, ORL1 (opioid receptor-like 1).
CSN26717 LY2940094 1307245-86-8 LY2940094 is a potent and selective nociceptin receptor antagonist which inhibits excessive feeding behavior in rodents.
CSN20227 LY2444296 1346133-11-6 LY2444296 is a short-acting kappa opioid receptor antagonist.
CSN23719 LY2940094 tartrate 1307245-87-9 LY-2940094 tartrate is the tartrate form of LY-2940094 which is an antagonist of nociceptin receptor that is used for the treatment of major depressive disorder and alcoholism.
CSN20601 Aticaprant 1174130-61-0 LY-2456302 is a potent and centrally-penetrant kappa opioid receptor antagonist with a Ki of 0.807 nM.
CSN21596 Gluten Exorphin C 142479-62-7 Gluten exorphin C, an opioid peptide derived from wheat gluten, can inhibit μ opioid and δ opioid with IC50 values of 40 μM and 13.5 μM in the GPI and MVD assays.
CSN21628 Endomorphin 2 141801-26-5 Endomorphin 2, an endogenous neuropeptide, is agonist of μ-opioid receptor with Ki of 0.69 nM that has analgesic and gastrointestinal properties.
CSN21627 Endomorphin 1 189388-22-5 Endomorphin 1 is a selective agonist of μ-opioid receptor with reasonable affinities for kappa3 binding sites (Ki value between 20 and 30 nM).
CSN35445 Difelikefalin 1024828-77-0 Difelikefalin (CR-845; FE-202845) is a peripherally restricted and selective agonist of kappa opioid receptor (KOR). Difelikefalin produces anti-inflammatory effects and has the potential in modulating pruritus in conditions such as chronic kidney disease.
CSN21597 Deltorphin I 122752-15-2 Deltorphin I is a selective agonist of δ-opioid receptor.
CSN22567 DAMGO 78123-71-4 DAMGO is a highly selective peptide agonist for the μ opioid receptor.
CSN33173 BTRX-335140 2244614-14-8 BTRX-335140 is a potent and selective KOR antagonist with IC50 (KOR)=0.8 nM.
CSN25444 BRL 52537 hydrochloride 112282-24-3 BRL-52537 hydrochloride is a potent and highly selective κ-opioid agonist. It has neuroprotective effects in animal studies, and is used for research into potential treatments for stroke and heart attack as well as more general brain research.
CSN27537 Bevenopran 676500-67-7 Bevenopran is a peripheral μ-opioid receptor antagonist.
CSN24259 BAN ORL 24diHCl- 475150-69-7 BAN ORL 24 is a potent and selective NOP receptor antagonist. (IC50 values are 0.27, 2500, 6700 and > 10000 nM for NOP, κ-, μ- and δ-receptors respectively).
CSN21495 Asimadoline 153205-46-0 Asimadoline is an agonist of κ-opioid receptor (KOR) with IC50 of 1.2 nM.
CSN23662 AR-M 1000390 hydrochloride 209808-47-9 AR-M 1000390 HCl is a non-peptidic and low-internalizing δ-selective opioid receptor agonist.
CSN27869 SCH 32615 83861-02-3
CSN41142 Dynorphin A 80448-90-4
CSN40048 Allomatrine 641-39-4
CSN36635 β-Endorphin, human 61214-51-5
CSN36630 Endomorphin 2 TFA 1276124-00-5
CSN33751 CTOP 103429-31-8
CSN35755 Dermorphin 77614-16-5
CSN63176 DIPPA hydrochloride 155512-52-0
CSN63462 BMS-986122 313669-88-4
CSN75683 ICI 199441 115199-84-3
CSN75308 Acetyl tetrapeptide-15 928007-64-1
CSN80506 AT-076 1657028-64-2
CSN81431 ML138 1355243-24-1
CSN104006 rel-4-((R)-((2S,5R)-4-allyl-2,5-dimethylpiperazin-1-yl)(3-hydroxyphenyl)methyl)-N,N-diethylbenzamide 150428-54-9
CSN104173 2-(3-(1-(2-(3,4-Dichlorophenyl)-N-methylacetamido)-2-(pyrrolidin-1-yl)ethyl)phenoxy)acetic acid hydrochloride 121264-04-8
CSN102444 N,N-Diethyl-3-hydroxy-4-(spiro[chromene-2,4'-piperidin]-4-yl)benzamide 850176-30-6
CSN104190 (2S,5S,14S)-15-Allyl-5-benzyl-14-(4-hydroxybenzyl)-2-isobutyl-8,8,11,11-tetramethyl-4,7,10,13-tetraoxo-3,6,9,12,15-pentaazaoctadec-17-en-1-oic acid 92535-15-4
CSN107811 2-Methyl-N-((2'-(pyrrolidin-1-ylsulfonyl)-[1,1'-biphenyl]-4-yl)methyl)propan-1-amine hydrochloride 1322001-35-3
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