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OX Receptor

OX Receptor

货号 产品名 CAS号 信息
CSN27292 YNT 185 1804978-81-1 YNT 185 is potent and selective orexin OX2 receptor agonist with EC50 of 28 nM at human OX2 expressed in CHO cells. YNT 185 displays approximately 100-fold selectivity for OX2 over OX1 (EC50 = 2.75 μM at human OX1 expressed in CHO cells).
CSN18978 TCS-OX2-29 372523-75-6 TCS-OX2-29 is a potent and selective orexin 2 (OX2) receptor antagonist with IC50 of 40 nM.
CSN16236 TCS 1102 916141-36-1 TCS 1102 is a potent, dual orexin receptor antagonist (Ki values are 0.2 and 3 nM for OX2 and OX1 receptors respectively).
CSN16826 SB-674042 483313-22-0 SB-674042 is a potent and selective non-peptide orexin OX1 receptor antagonist (Kd = 3.76 nM) exhibiting 100-fold selectivity for OX1 over OX2 receptors.
CSN20633 SB-649868 380899-24-1 SB-649868 is a potent and selective orally active orexin (OX) 1 and OX2 receptor antagonist (pKi =9.4 and 9.5 at the OX1 and OX2 receptor, respectively).
CSN16521 SB-408124 288150-92-5 SB-408124 is a non-peptide antagonist for OX1 receptor with Ki of 57 nM and 27 nM in both whole cell and membrane, respectively, and exhibits 50-fold selectivity over OX2 receptor.
CSN11490 SB-334867 249889-64-3 SB-334867 is a selective non-peptide orexin OX1 receptor antagonist with a pKb value of 7.2.
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