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OX Receptor
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN27292 | YNT 185 | 1804978-81-1 | YNT 185 is potent and selective orexin OX2 receptor agonist with EC50 of 28 nM at human OX2 expressed in CHO cells. YNT 185 displays approximately 100-fold selectivity for OX2 over OX1 (EC50 = 2.75 μM at human OX1 expressed in CHO cells). |
| CSN18978 | TCS-OX2-29 | 372523-75-6 | TCS-OX2-29 is a potent and selective orexin 2 (OX2) receptor antagonist with IC50 of 40 nM. |
| CSN16236 | TCS 1102 | 916141-36-1 | TCS 1102 is a potent, dual orexin receptor antagonist (Ki values are 0.2 and 3 nM for OX2 and OX1 receptors respectively). |
| CSN16826 | SB-674042 | 483313-22-0 | SB-674042 is a potent and selective non-peptide orexin OX1 receptor antagonist (Kd = 3.76 nM) exhibiting 100-fold selectivity for OX1 over OX2 receptors. |
| CSN20633 | SB-649868 | 380899-24-1 | SB-649868 is a potent and selective orally active orexin (OX) 1 and OX2 receptor antagonist (pKi =9.4 and 9.5 at the OX1 and OX2 receptor, respectively). |
| CSN16521 | SB-408124 | 288150-92-5 | SB-408124 is a non-peptide antagonist for OX1 receptor with Ki of 57 nM and 27 nM in both whole cell and membrane, respectively, and exhibits 50-fold selectivity over OX2 receptor. |
| CSN11490 | SB-334867 | 249889-64-3 | SB-334867 is a selective non-peptide orexin OX1 receptor antagonist with a pKb value of 7.2. |
