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P-gp

P-gp

货号 产品名 CAS号 信息
CSN12903 Zosuquidar 167354-41-8 Zosuquidar is P-gp modulator that inhibited Pgp-ATPase activity 50-60% at 2 and 10μM and had no effect at 0.08 and 0.4μM (measured by P-gp ATPase activity).
CSN12751 Zosuquidar trihydrochloride 167465-36-3 Zosuquidar 3HCl is the 3HCl form of Zosuquidar. Zosuquidar is P-gp modulator that inhibited Pgp-ATPase activity 50-60% at 2 and 10μM and had no effect at 0.08 and 0.4μM.
CSN12182 Valspodar 121584-18-7 Valspodar is a P-glycoprotein (P-gp) inhibitor widely used in preclinical and clinical studies for overcoming multidrug resistance (MDR).
CSN14774 Taxinine B 18457-44-8 Taxinine B, a natural product isolated and purified from the barks of Taxus chinensis, can inhibit the drug transport by P-glycoprotein in multidrug-resistant cells, and shows stronger inhibitory effects than acetylsalicylic acid (ASA) on platelet aggregation induced by arachidonic acid (AA).
CSN18364 Tariquidar methanesulfonate, hydrate 625375-83-9 Tariquidar methanesulfonate is a potent and specific inhibitor of P-glycoprotein (P-gp) with the high affinity (Kd=5.1±0.9 nM).
CSN12910 Tariquidar 206873-63-4 Tariquidar is a potent and selective noncompetitive inhibitor of P-glycoprotein with Kd of 5.1 nM, reverses drug resistance in MDR cell Lines.
CSN13177 Sinapine thiocyanate 7431-77-8 Sinapine, an alkaloid isolated and purified from the seeds of Raphanus sativus L., possess antioxidant and radio-protective activities, downregulats multi-drug resistance 1 (MDR1) expression.
CSN22057 Sinapine 18696-26-9 Sinapine is an alkaloid from seeds of the cruciferous species which shows antioxidant and radio-protective activities and decreases expression of P-glycoprotein in Caco-2 cells.
CSN19434 Schisandrin 7432-28-2 Schizandrin is a natural product possessing antioxidant and anti-inflammatory activities.
CSN16588 SC144 895158-95-9 SC144 showed its function through both exhibiting potent cytotoxicity, by itself or synergism with other compounds, against a panel of drug-sensitive and drug-resistant cancer cell lines, and targeting to gp130.
CSN18576 SC144 hydrochloride 917497-70-2 SC144 HCl is the first-in-class orally active small-molecule gp130 inhibitor (IC50 = 0.72 μM) which blocks cytokine-triggered gp130 signaling.
CSN25413 RCGD423 108237-91-8 RCGD423 is a gp130 modulator, which prevents articular cartilage degeneration and promotes repair.
CSN14118 Phyllanthin 10351-88-9 Phyllanthin, a natural product isolated and purified from the herb of Phyllanthus niruri L., is widely used as hepatoprotective and antigenotoxic and inhibit function of P-gp.
CSN13555 Isosinensetin 17290-70-9 Isosinensetin exhibits HIV-1 protease inhibiting and antioxidant activities. It is a natural product isolated and purified from the fruit of Citrus aurantium L..
CSN15743 Encequidar 849675-66-7 HM30181 is a potent and selective inhibitor of P-glycoprotein.
CSN23176 GP130 receptor agonist-1 339303-87-6 gp130-agonist-2 is a brain penetrant gp130 agonist which protects against NMDA-induced toxicity and increases STAT3 phosphorylation.
CSN14838 Epimedokoreanin B 161068-53-7 Epimedokoreanin B is a natural product isolated and purified from the herbs of Epimedium brevicornum.
CSN10894 Elacridar   143664-11-3 Elacridar is a P-glycoprotein inhibitor, and has been used both in vitro and in vivo as a tool inhibitor of P-glycoprotein (Pgp) to investigate the role of transporters in the disposition of various test molecules.
CSN13175 Elacridar hydrochloride 143851-98-3 Elacridar HCl is a P-glycoprotein (P-gp) inhibitor, and has been used both in vitro and in vivo as a tool inhibitor of P-gp to investigate the role of transporters in the disposition of various test molecules.
CSN17917 Dofequidar fumarate 153653-30-6 Dofequidar fumarate, an orally active quinoline compound, has been reported to overcome MDR by inhibiting ABCB1/P-gp, ABCC1/MDR-associated protein 1, or both.
CSN22768 CP-100356 hydrochloride 142715-48-8 CP 100356 HCl is a high affinity P-glycoprotein (P-gp) inhibitor with Kis of 58 and 94 nM for mouse Pgp1a and Pgp1b isoforms.
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