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P450

P450

货号 产品名 CAS号 信息
CSN21919 Uniconazole 83657-22-1 Uniconazole inhibits CK biosynthesis by suppressing CYP735A activity in Arabidopsis. Uniconazole inhibits the biosynthesis of gibberellin (GA), and brassinosteroid (BR) and the catabolism of abscisic acid (ABA).
CSN26275 Tetrahydropiperine 23434-88-0 Tetrahydropiperine is a cyclohexyl analogue of piperine that inhibits the cytochrome P450 (CYP) isoform CYP1A1/arylhydrocarbon hydroxylase (AHH; IC50=23 µM).
CSN23249 Stiripentol 49763-96-4 Stiripentol is an antiepileptic drug that can inhibit the synaptosomal uptake of GABA, increase the activation of GABAA receptors, it's also a microsomal cytochrome P450 (CYP) isoforms CYP3A4, CYP1A2, and CYP2C19 inhibitor.
CSN19933 Rhodionin 85571-15-9 Rhodionin can inhibit cytochrome P450 2D6 non-competitively with high specificity which could have implications for interactions with co-administered drugs.
CSN19400 Ramatroban 116649-85-5 Ramatroban is a thromboxane A(2) (TxA(2)) antagonist marketed for allergic rhinitis.
CSN26727 Ozagrel Sodium 189224-26-8 Ozagrel Sodium, also known as KCT-0809 and Cataclot, is a thromboxane A2 synthase inhibitor used to treat cerebrovascular diseases.
CSN25582 NVP-VID-400 174262-13-6 NVP-VID-400 is an inhibitor of both CYP51 and CYP24A1.
CSN29462 17-ODYA 34450-18-5 LTB ω-hydroxylase inhibitor.
CSN24909 Sparteine 492-08-0 Inhibition of human CYP2D6 expressed in Escherichia coli JM109
CSN26726 Gemfibrozil 1-O-β-glucuronide 91683-38-4 Gemfibrozil 1-O-β-Glucuronide, a metabolite of Gemfibrozil (CI-719; HY-B0258), is a potent and competitive P450 (CYP) isoform CYP2C8 inhibitor with an IC50 of 4.07 μM[1][2].
CSN22095 Furafylline 80288-49-9 Furafylline is a potent and selective inhibitor of human cytochrome P450IA2 with IC50 of 0.07 μM.
CSN29463 7-Ethoxyresorufin 5725-91-7 Fluorometric CYP450 substrate.
CSN29461 Methoxyresorufin 5725-89-3 Fluorometric CYP450 substrate.
CSN23291 Flavone 525-82-6 Flavone can effect CYP (P450) activity, it's a class of flavonoids with antioxidant, anti-proliferative, anti-tumor, anti-microbial, estrogenic, acetyl cholinesterase, anti-inflammatory activities and are also used in cancer, cardiovascular disease, neurodegenerative disorders etc.
CSN22890 DMU2139 1821143-80-9 DMU2139 is a selective inhibitor of CYP1B1 with IC50 of 9 nM.
CSN27199 DMU2105 1031063-36-1 DMU2105 is a potent CYP1B1 inhibitor with IC50 value of 10nM for human CYP1B1 enzyme bound to yeast-derived microsomes (Sacchrosomes™).
CSN25347 Dazoxiben HCl 74226-22-5 Dazoxiben hydrochloride is a potent, orally active thromboxane (TX) synthase inhibitor that reduces the formation of blood clots.
CSN17441 Dafadine-A 1065506-69-5 Dafadine-A, an analog of dafadine, is an inhibitor of DAF-9 cytochrome P450 in the nematode Caenorhabditis elegans and also inhibits the mammalian ortholog of DAF-9 (CYP27A1).
CSN13101 Chlorzoxazone 95-25-0 Chlorzoxazone, a potassium channel activator, is a centrally acting muscle relaxant used to treat muscle spasm and the resulting pain or discomfort. It is also a CYP2E1 inhibitor with IC50 value of 1.03μM.
CSN21322 CGS 15435 95853-92-2 CGS 15435, a potent thromboxane (TxA2) synthetase inhibitor with an IC50 of 1 nM, has a selectivity for Tx synthetase 100000-fold greater than that for cyclooxygenase, PGI2 synthetase and lipoxygenase enzymes.
CSN19045 CDD3506 197913-15-8 CDD3506 is used for elevating high density lipoprotein cholesterol (HDL) by inducing hepaticcytochrome P450IIIA (CYP3A)activity.
CSN19044 CDD3505 173865-33-3 CDD3505 is used for elevating high density lipoprotein cholesterol (HDL) by inducing hepaticcytochrome P450IIIA (CYP3A)activity.
CSN21515 Bergaptin 7380-40-7 Bergaptin is a competitive inhibitor of CYP1A1 with Ki of 10.7 nM.
CSN22313 ABT 1614-12-6 ABT is a non-specific cytochrome P450 (CYP) inhibitor.
CSN26155 6-Aminochrysene 2642-98-0 6-aminochrysene was a potent inducer of CYP1A1 in rat.
CSN19374 3-Cyano-7-Ethoxycoumarin 117620-77-6 3-Cyano-7-ethoxycoumarin is a fluorogenic cytochrome P-450 substrate that generates blue fluorescent product upon enzyme cleavage.
CSN19771 25R-Inokosterone 19682-38-3 25R-Inokosterone has a role on cytochrome P450 from a hormone-resistant cell line.
CSN22146 1-Ethynylnaphthalene 15727-65-8 1-Ethynylnaphthalene is a selective inhibitor of cytochrome P450 1B1.
CSN29472 (S)-Mephenytoin 70989-04-7 (S)-Mephenytoin is a substrate of the cytochrome P450 (CYP) isoform CYP2C19, also known as mephenytoin 4-hydroxylase.
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