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PAD

货号 产品名 CAS号 信息
CSN23163 Thr-Asp-F-amidine 1345019-64-8 PAD4 inhibitor
CSN21368 GSK484 HCl 1652591-81-5 GSK484 is a reversible and selective inhibitor of PAD4 with IC50 of 50 nM. GSK484 blocks the citrullination of PAD4 target proteins in human neutrophils and inhibits the formation of neutrophil extracellular traps in both mouse and human neutrophils.
CSN37337 Cl-amidine HCl 1373232-26-8 Cl-amidine is an irreversible pan-peptidylarginine deiminase (PAD) inhibitor with IC50 values of with IC50 values of 5.9 ± 0.3 μM, 0.8 ± 0.3 μM, 6.2 ± 1.0 μM for PAD4, PAD1 and PAD3, respectively.
CSN25240 Cl-amidine TFA   1043444-18-3 Cl-amidine is a peptidylarginine deminase (PAD) inhibitor, with an IC50 5.9±0.3 μM for PAD4.
CSN22375 Cl-amidine 913723-61-2 Cl-amidine is a peptidylarginine deminase (PAD) inhibitor, with an IC50 5.9±0.3 μM for PAD4.
CSN23725 BB-Cl-Amidine 1802637-39-3 BB-Cl-amidine is a irreversible peptidylarginine deminase (PAD) inhibitor.
CSN67079 GSK121 1652591-80-4
CSN67081 GSK106 1652591-82-6
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