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PDK is a kinase enzyme which acts to inactivate the enzyme pyruvate dehydrogenase by phosphorylating it using ATP.

PDK

货号 产品名 CAS号 信息
CSN17521 PS48 1180676-32-7 PS48 is a phosphoinositide-dependent protein kinase-1 (PDK1) activator with Kd value of 10.3 μM and binds exclusively to the PIF-binding pocket of PDK1, distinct from the ATP binding site.
CSN25617 PDK-4 Inhibitor compound 8c HCl 2310262-11-2 PDK-4 Inhibitor compound 8c HCl is an allosteric PDK-4 inhibitor with IC50 value of 84nM.
CSN27211 JX06   729-46-4 JX06 is a selective covalent PDK1 inhibitor with IC50 values of 49, 101 and 313nM for PDK-1, PDK-2 and PDK-3, respectively.
CSN17589 GSK2334470 1227911-45-6 GSK2334470 is a PDK1 inhibitor with IC50 of ~10 nM, with no activity at other close related AGC-kinases.
CSN19146 BX517 850717-64-5 BX517 is a potent and selective inhibitor of PDK1 with IC50 of 6 nM.
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