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Phospholipase

Phospholipase

货号 产品名 CAS号 信息
CSN23873 VU0155069 1130067-06-9 VU-0155069 is a selective phospholipase D1 (PLD1) inhibitor with IC50 values of 46 and 933 nM for PLD1 and PLD2 respectively.
CSN12192 Varespladib 172732-68-2 Varespladib is a potent and selective human non-pancreatic secretory phospholipase A2 (sPLA) inhibitor with IC50 of 7 nM.
CSN26229 U-73343 142878-12-4 U-73343, an inhibitor of PLC (putative phospholipase C)-dependent processes, is an inactive structural analog of U-73122 and can be used as a negative control.
CSN12944 U-73122 112648-68-7 U-73122 is an inhibitor of phospholipase C, phospholipase A2, and 5-LO(5-lipoxygenase).
CSN27559 (E)-4-Phenylbut-3-en-2-one 1896-62-4 trans-Benzylideneacetone (trans-Benzalacetone), a metabolite of gram-negative entomopathogenic bacterium Xenorhabdus nematophila, is an enzyme inhibitor against phospholipase A2 (PLA2). trans-Benzylideneacetone is an immunosuppressant.
CSN17463 SPK-601 1096687-52-3 SPK-601 is a potent phosphatidylcholine-specific phospholipase C (PC-PLC) inhibitor and is a useful antimicrobial agent.
CSN23724 N-(p-amylcinnamoyl) Anthranilic Acid 110683-10-8 N-(p-amylcinnamoyl) Anthranilic Acid is a PLA2 inhibitor and TRP channel modulator.
CSN18844 ML348 899713-86-1 ML348 is a selective and reversible lysophospholipase 1 (LYPLA1) inhibitor (IC50 = 210 nM), Exhibits 14-fold selectivity for LYPLA1 over LYPLA2, Also selective over a panel of ~30 other serine hydrolases.
CSN25338 ML349 890819-86-0 ML 349 is a selective and reversible lysophospholipase 2 (LYPLA2) inhibitor with IC50 of 144 nM.
CSN23868 Quinacrine 83-89-6 Mepacrine is an acridine derivative formerly widely used as an anthelmintic and in the treatment of giardiasis and malignant effusions. It's also an inhibitor of phospholipase A2.
CSN11815 N4-(6-Chloro-2-methoxyacridin-9-yl)-N1,N1-diethylpentane-1,4-diamine dihydrochloride 69-05-6 Mepacrine 2HCl is an acridine-derived yellow dye, previously used in the therapy and prevention of malaria and later as an antiprotozoal and immunomodulatory agent. It's also an inhibitor of phospholipase A2.
CSN21819 Quinacrine HCl 6151-30-0 Mepacrine 2HCl 2H2O is an acridine derivative formerly widely used as an anthelmintic and in the treatment of giardiasis and malignant effusions. It's also an inhibitor of phospholipase A2.
CSN27210 m-3M3FBS 200933-14-8 m-3M3FBS is a novel phospholipase C activator. It can be developed as a novel anti-leukemic agent.
CSN16514 FIPI 939055-18-2 FIPI is a derivative of halopemide which potently inhibits both PLD1 (IC50 = 25 nM) and PLD2 (IC50 = 20 nM) preventing PLD regulation of F-actin cytoskeleton reorganization, cell spreading, and chemotaxis.
CSN15706 Darapladib 356057-34-6 Darapladib is a reversible lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor with IC50 of 0.25 nM.
CSN10738 D609 83373-60-8 D609 is a selective competitive phosphatidyl choline-specific phospholipase C (PC-PLC) inhibitor (Ki = 6.4 μM) and antiviral and antitumor agent.
CSN17598 CAY10650 1233706-88-1 CAY10650 is a highly potent cytosolic phospholipase A2α (cPLA2α) inhibitor with an IC50 value of 12 nM.
CSN27739 CAY10594 1130067-34-3 CAY10594 is a selective PLD2 inhibitor with IC50 values of 140nM and 5.1μM for PLD2 and PLD1, respectively. It strongly inhibits the invasive migration of breast cancer cells in transwell assays.
CSN27249 7,7-Dimethyleicosadienoic Acid 89560-01-0 7,7-Dimethyleicosadienoic Acid is a selective secretory type phospholipase A2 (PLA2) inhibitor with IC50 value of 250μM in the presence of Epo.
CSN21980 1-Linoleoyl Glycerol 2277-28-3 1-Linoleoyl Glycerol is a fatty acid glycerol that has been isolated from S. chinensis roots and exhibits Lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitory activities with IC50 values of 45.0 μM for (R)-1-Linoleoyl Glycerol and 52.0 μM for (S)-1-Linoleoyl Glycerol, respectively.
CSN29448 (R)-Edelfosine 77286-66-9 Selective PI-PLC inhibitor, also PAF receptor agonist
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