Pim
货号 | 产品名 | CAS号 | 信息 |
---|---|---|---|
CSN16821 | TCS-PIM-1-4a | 327033-36-3 | TCS-PIM-1-4a is a Pim inhibitor that blocks mTORC1 activity via activation of AMPK and kills a wide range of both myeloid and lymphoid cell lines (with IC50 values ranging from 0.8 to 40 μM). |
CSN15804 | SMI-4a | 438190-29-5 | SMI-4a is a potent inhibitor of Pim1 with IC50 of 17 nM, modestly potent to Pim-2, does not significantly inhibit any other serine/threonine- or tyrosine-kinases. |
CSN20347 | SMI-16a | 587852-28-6 | SMI-16a, the PIM1/2 Kinase inhibitor VI, controls the biological activity of PIM1/2. This small molecular inhibitor is primarily used for Phosphorylation & Dephosphorylation applications |
CSN19180 | CX-6258 HCl | 1353859-00-3 | CX-6258 HCl is a potent, orally efficacious pan-Pim kinase inhibitor with IC50 of 5 nM, 25 nM and 16 nM for Pim1, Pim2, and Pim3, respectively. |