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CAS No.: 1633350-06-7
Synonyms: (±)-BGB-3111;BGB-3111 (Recemate)
BGB-3111 is a potent, selective and orally available Bruton's tyrosine kinase (Btk) inhibitor.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT03432884 | Healthy Volunteers | Phase 1 | Completed | - | United States, New Jersey ... more >> Frontage Clinical Services, Inc. Secaucus, New Jersey, United States, 07094 Collapse << |
NCT03561298 | Healthy Subjects | Phase 1 | Completed | - | United States, Florida ... more >> Covance Clinical Research Unit Daytona Beach, Florida, United States, 32117 Collapse << |
NCT03465059 | Hepatic Insufficiency & Health... more >>y Subjects Collapse << | Phase 1 | Active, not recruiting | December 2018 | United States, Florida ... more >> University of Miami Miami, Florida, United States, 33124 Orlando Clinical Research Center Orlando, Florida, United States, 32809 Collapse << |
实验方案
技术信息
CAS号 | 1633350-06-7 | 储存条件 |
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分子式 | C27H29N5O3 | 运输 | 蓝冰 | |
分子量 | 471.55 | 别名 | (±)-BGB-3111;BGB-3111 (Recemate) |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT03432884 | Healthy Volunteers | Phase 1 | Completed | - | United States, New Jersey ... more >> Frontage Clinical Services, Inc. Secaucus, New Jersey, United States, 07094 Collapse << |
NCT03561298 | Healthy Subjects | Phase 1 | Completed | - | United States, Florida ... more >> Covance Clinical Research Unit Daytona Beach, Florida, United States, 32117 Collapse << |
NCT03465059 | Hepatic Insufficiency & Health... more >>y Subjects Collapse << | Phase 1 | Active, not recruiting | December 2018 | United States, Florida ... more >> University of Miami Miami, Florida, United States, 33124 Orlando Clinical Research Center Orlando, Florida, United States, 32809 Collapse << |
NCT03734016 | Chronic Lymphocytic Leukemia ... more >> Small Lymphocytic Lymphoma Collapse << | Phase 3 | Recruiting | October 2025 | United States, Nevada ... more >> Comprehensive Cancer Centers of Nevada - USOR Recruiting Las Vegas, Nevada, United States, 89169 Principal Investigator: Edwin Kingsley, MD United States, New Jersey Summit Medical Group Recruiting Florham Park, New Jersey, United States, 07932 Principal Investigator: Charles Farber, MD United States, New York Clinical Research Alliance Inc Recruiting Lake Success, New York, United States, 11042 Principal Investigator: Morton Coleman, MD United States, Washington Medical Oncology Associates Recruiting Spokane, Washington, United States, 99208 Principal Investigator: Arvind Chaudhry Collapse << |
NCT02569476 | B-cell Lymphoid Malignancies | Phase 1 | Active, not recruiting | February 2019 | United States, Florida ... more >> Florida Cancer Specialists Fort Myers, Florida, United States, 33916 Florida Cancer Specialists Saint Petersburg, Florida, United States, 33705 United States, Tennessee Tennessee Oncology, PLLC - Nashville Nashville, Tennessee, United States, 37203 Australia, New South Wales Border Medical Oncology Albury, New South Wales, Australia, 2640 St George Hospital Kogarah, New South Wales, Australia, 2217 Australia, Queensland Brisbane Clinic for Lymphoma, Myeloma and Leukaemia Greenslopes, Queensland, Australia, 4120 Australia, South Australia Ashford Cancer Centre Research Kurralta Park, South Australia, Australia, 5037 Australia, Victoria St Vincent's Hospital Melbourne East Melbourne, Victoria, Australia, 3002 University Hospital Geelong Geelong, Victoria, Australia, 3220 St Frances Xavier Cabrini Hospital Malvern, Victoria, Australia, 3144 The Alfred Hospital Melbourne, Victoria, Australia, 3181 Australia, Western Australia Royal Perth Hospital Perth, Western Australia, Australia, 6000 Korea, Republic of Severance Hospital, Yonsei University Seoul, Korea, Republic of, 03722 Asan Medical Center Seoul, Korea, Republic of, 05505 Samsung Medical Center Seoul, Korea, Republic of, 06351 Collapse << |
NCT02795182 | Lymphoma Leuk... more >>emia Collapse << | Phase 1 | Recruiting | December 2019 | Australia, New South Wales ... more >> Concord Hospital Recruiting Sydney, New South Wales, Australia, 2139 Australia, Victoria Monash Hospital Recruiting Clayton, Victoria, Australia, 3168 Peter MacCallum Cancer Centre Recruiting Melbourne, Victoria, Australia, 3002 Australia, Western Australia Sir Charles Gairdner Hospital Recruiting Nedlands, Western Australia, Australia, 6009 Collapse << |
NCT03145064 | Diffuse Large B Cell Lymphoma | Phase 2 | Active, not recruiting | August 24, 2019 | China, Beijing ... more >> Cancer Hospital Chinese Academy of Medical Sciences Beijing, Beijing, China Peking University Cancer Hospital Beijing, Beijing, China China, Chengdu West China Hospital, Sichuan University Chengdu, Chengdu, China China, Hangzhou Zhengjiang Cancer hospital Hangzhou, Hangzhou, China China, Hebei Fourth Hospital of HeBei Medical University Shijiazhuang, Hebei, China China, Helongjiang Haerbin Cancer Hospital Haerbin, Helongjiang, China China, Henan Henan province cancer hospital Zhengzhou, Henan, China China, Jilin Jilin University Affiliated Hospital Changchun, Jilin, China China, Shanghai Fudan University Shanghai Cancer Center Shanghai, Shanghai, China Ruijin Hospital, Shanghai Jiaotong University School of Medicine Shanghai, Shanghai, China China, Suzhou The first affiliated hospital of Soochow University Suzhou, Suzhou, China China, Tianjin Institute of Hematology & Blood Diseases Hospital Tianjin, Tianjin, China Tianjin Medical University Cancer Institute&Hospital Tianjin, Tianjin, China Collapse << |
NCT02343120 | Relapsed/Refractory B-cell Mal... more >>ignancies Collapse << | Phase 1 | Recruiting | December 2023 | United States, Texas ... more >> M.D. Anderson Cancer Center Recruiting Houston, Texas, United States, 77030 Australia, New South Wales Concord Repatriation General Hospital Recruiting Concord, New South Wales, Australia Westmead Hospital Recruiting Westmead, New South Wales, Australia Australia, Queensland Princess Alexandra Hospital Recruiting Brisbane, Queensland, Australia Australia, Victoria Monash Health Recruiting Clayton, Victoria, Australia Austin Health Recruiting Heidelberg, Victoria, Australia Peter MacCallum Cancer Centre, East Melbourne Recruiting Parkville, Victoria, Australia, 3050 Melbourne Health Recruiting Parkville, Victoria, Australia Australia, Western Australia Sir Charles Gairdner Hospital Recruiting Nedlands, Western Australia, Australia Australia St Vincent's Hospital Recruiting Melbourne, Australia Contact: Joseph Nguyen Korea, Republic of Dong-A University Medical Centre Recruiting Busan, Korea, Republic of Inje University Busan Paik Hospital Recruiting Busan, Korea, Republic of National Cancer Center Recruiting Goyang-si, Korea, Republic of Samsung Medical Center Recruiting Seoul, Korea, Republic of New Zealand North Shore Hospital Recruiting Auckland, New Zealand Collapse << |
NCT03332017 | Relapsed/Refractory Follicular... more >> Non-Hodgkin Lymphoma Collapse << | Phase 2 | Recruiting | October 2021 | - |
NCT03301181 | Healthy Volunteers: Asian, Non... more >>-Asian Collapse << | Phase 1 | Completed | - | United States, California ... more >> West Coast Clinical Trials (WCCT) Cypress, California, United States, 90630 Collapse << |
NCT03206970 | Relapsed or Refractory Mantle ... more >>Cell Lymphoma Collapse << | Phase 2 | Active, not recruiting | November 2020 | China, Beijing ... more >> Beijing Cancer Hospital Beijing, Beijing, China, 100142 Peking Union Medical College Hospital Beijing, Beijing, China Peking University People's Hospital Beijing, Beijing, China China, Fujian Fujian Medical University Union Hospital Fuzhou, Fujian, China China, Guangdong Nanfang Hospital Guangzhou, Guangdong, China China, Henan Henan Cancer Province Zhengzhou, Henan, China China, Hubei Tongji Hospital, Tongji Medical College Huazhong University of Science and Technology Wuhan, Hubei, China China, Jiangsu Jiangsu Province Hospital Nanjing, Jiangsu, China The First Affiliated Hospital of Soochow University Suzhou, Jiangsu, China China, Jinlin The First Affilliated Hospital of Jinlin University Changchun, Jinlin, China China, Shanghai Fudan University Shanghai Cancer Center Shanghai, Shanghai, China Rui Jin Hospital Shanghai Jiao Tong University Schlool of Medicine Shanghai, Shanghai, China China, Sichuan West China Hospital of Sichuan University Chengdu, Sichuan, China China, Tianjin Tianjin Hematonosis Hospital Tianjin, Tianjin, China Tianjin Medical University Cancer Institute and Hospital Tianjin, Tianjin, China China, Zhejiang The First affiliated Hospital, Zhejiang University Hangzhou, Zhejiang, China Zhejiang Cancer Hospital Hangzhou, Zhejiang, China Collapse << |
NCT03332173 | Waldenström's Macroglobulinemi... more >>a (WM) Collapse << | Phase 2 | Recruiting | November 2021 | China, Beijing ... more >> Peking Union Medical College Hospital Recruiting Beijing, Beijing, China Peking University Pepole's Hospital Not yet recruiting Beijing, Beijing, China China, Guangdong Guangdong General Hospital Not yet recruiting Guangzhou, Guangdong, China China, Henan Henan Cancer Hospital Not yet recruiting Zhengzhou, Henan, China China, Hubei Tongji Hospital, Tongji Medical College, Huazhong University of Science and Technology Recruiting Wuhan, Hubei, China China, Jiangsu Jiangsu Province Hospital Not yet recruiting Nanjing, Jiangsu, China The first affiliated hospital of Soochow University Not yet recruiting Suzhou, Jiangsu, China China, Shanghai Ruijin Hospital, Shanghai Jiaotong University School of Medicine Not yet recruiting Shanghai, Shanghai, China China, Sichuan West China Hospital, Sichuan University Not yet recruiting Chengdu, Sichuan, China China, Tianjin Institute of Hematology & Blood Diseases Hospital Recruiting Tianjin, Tianjin, China China, Zhejiang The First Affiliated Hospital of Zhejiang University Not yet recruiting Hangzhou, Zhejiang, China Collapse << |
NCT03520920 | Marginal Zone Lymphoma ... more >> Follicular Lymphoma Diffuse Large B-Cell Lymphoma Collapse << | Phase 2 | Recruiting | December 2020 | China, Heilongjiang ... more >> Harbin Medical University Cancer Hospital Recruiting Harbin, Heilongjiang, China Contact: Qingyuan Zhang China, Hubei ongji Hospital, Tongji Medical College of HUST Recruiting Wuhan, Hubei, China Contact: Jianfeng Zhou China, Jiangsu The Affiliated Hospital of Xuzhou Medical University Recruiting Xuzhou, Jiangsu, China Contact: Zhenyu Li China, Shanghai Xinhua Hospital affiliated to Shanghai Jiao Tong University School of Mdicine Not yet recruiting Shanghai, Shanghai, China Contact: Rong Tao Collapse << |
NCT03336333 | Chronic Lymphocytic Leukemia ... more >> Small Lymphocytic Lymphoma Collapse << | Phase 3 | Recruiting | October 2022 | - |
NCT03189524 | B-cell Lymphoma | Phase 1 | Recruiting | June 30, 2021 | China, Beijing ... more >> Beijing Cancer Hospital Recruiting Beijing, Beijing, China, 100142 China, Hubei Tongji Hospital, Tongji Medical College Huazhong Univ of Sci and Tch Recruiting Wuhan, Hubei, China China, Jiangsu Jiangsu Province Hospital Recruiting Nanjing, Jiangsu, China China, Tianjin Tianjin Hematonosis Hospital Recruiting Tianjin, Tianjin, China Collapse << |
NCT03206918 | Relapsed or Refractory Chronic... more >> Lymphocytic Leukemia Relapsed or Refractory Small Lymphocytic Lymphoma Collapse << | Phase 2 | Active, not recruiting | December 2020 | China, Beijing ... more >> Peking Union Medical College Hospital Beijing, Beijing, China Peking University People's Hospital Beijing, Beijing, China China, Fujian Fujian Medical University Union Hospital Fuzhou, Fujian, China China, Guangdong Guangdong General Hospital Guangzhou, Guangdong, China Nanfang Hospital Guangzhou, Guangdong, China China, Guangxi The First Affiliated Hospital of GuangXi Medical University Nanning, Guangxi, China China, Henan Henan Cancer Province Zhengzhou, Henan, China China, Hubei Tongji Hospital, Tongji Medical College Huazhong University of Science and Technology Wuhan, Hubei, China China, Jiangsu Jiangsu Province Hospital Nanjing, Jiangsu, China The First Affiliated Hospital of Soochow University Suzhou, Jiangsu, China China, Jinlin The First Affilliated Hospital of Jinlin University Changchun, Jinlin, China China, Shanghai Rui Jin Hospital Shanghai Jiao Tong University Schlool of Medicine Shanghai, Shanghai, China China, Shanxi The 1st Affiliated Hospital of Xi'An Jiaotong University Xi'an, Shanxi, China China, Sichuan West China Hospital of Sichuan University Chengdu, Sichuan, China China, Tianjin Tianjin Hematonosis Hospital Tianjin, Tianjin, China China, Zhejiang The First affiliated Hospital, Zhejiang University Hangzhou, Zhejiang, China Collapse << |
NCT03053440 | Waldenström's Macroglobulinemi... more >>a Collapse << | Phase 3 | Active, not recruiting | June 2021 | - |
NCT03740529 | Chronic Lymphocytic Leukemia ... more >> Waldenstrom's Macroglobulinemia Mantle Cell Lymphoma Marginal Zone Lymphoma B-cell Lymphoma Small Lymphocytic Lymphoma Collapse << | Phase 1 Phase 2 | Recruiting | April 2021 | United States, Tennessee ... more >> Sarah Cannon Research Institute at Tennessee Oncology Recruiting Nashville, Tennessee, United States, 37203 Contact: Ian W Flinn, MD, PhD Collapse << |
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