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CAS No.: 14003-96-4
Synonyms: IRE1 Inhibitor III;4mu8C;4u8C
4μ8C is a potent and selective IRE1 Rnase inhibitor with IC50 of 76 nM.
生物活性
实验方案
技术信息
CAS号 | 14003-96-4 | 储存条件 |
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分子式 | C11H8O4 | 运输 | 蓝冰 | |||||||||
分子量 | 204.18 | 别名 | IRE1 Inhibitor III;4mu8C;4u8C | |||||||||
溶解度 |
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动物实验配方 |
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Cell Lines | Concentration | Assay Type | Time | Activity Description | Data Sources |
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human Jeko cells | - | Function assay | 24 h | Inhibition of XBP-1s expression in human Jeko cells after 24 hrs by immunoblotting analysis, IC50=1.57 μM | 24749861 |
human Mino cells | - | Function assay | 24 h | Inhibition of XBP-1s expression in human Mino cells after 24 hrs by immunoblotting analysis, IC50=1.62 μM | 24749861 |
SF21 cells | - | Function assay | 30 mins | Inhibition of human recombinant puritin-His-tagged IRE-1 RNase expressed in SF21 cells using XBP-1 RNA stem loop as substrate incubated for 30 mins prior to substrate addition measured after 2 hrs by FRET-suppression assay, IC50=0.206 μM | 24749861 |
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