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CAS No.: 552325-73-2
Synonyms: A-674563
A-674563 is a potent selective Akt1 inhibitor with an IC50 of 14 nM. It also shows inhibitory activity against PKA and CDK2 with IC50 of 16 and 46 nM, respectively.
生物活性
实验方案
技术信息
CAS号 | 552325-73-2 | 储存条件 |
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分子式 | C22H22N4O | 运输 | 蓝冰 | |
分子量 | 358.44 | 别名 | A-674563 |
Cell Lines | Concentration | Assay Type | Time | Activity Description | Data Sources |
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MIA PaCa cells | - | Cytotoxic assay | - | Cytotoxicity against human MIA PaCa cells by MTT assay, EC50=0.64 μM | 17523610 |
MiaPaCa2 cell | - | Proliferation assay | - | Antiproliferative activity against human MiaPaCa2 cell line, EC50=0.4 μM | 16678413 |
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