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CAS No.: 141430-65-1

ABT-751 Catalog No. CSN16987

Synonyms: E7010

ABT-751 can inhibit microtubule polymerization through binding to β-tubulin on the colchine site.

规格 价格 促销价格 库存 数量
纯度 & 质量文件 批次:

靶点选择性

生物活性

  • 描述
  • 细胞研究
  • Cell Data
  • 更多
  • 动物研究
    剂量

    Rat: 3 mg/kg - 30 mg/kg[3] (i.v.) Mice: 75 mg/kg, 100 mg/kg[4] (p.o.)

    给药途径

    i.v., p.o.

  • 临床研究
  • NCT号适应症或疾病临床期招募状态预计完成时间地点
    NCT00297089Lung Cancer N... more >>SCLC Non-Small-Cell Lung Cancer Collapse <<Phase 1 Phase 2Completed--
    NCT00439296Recurrent Pediatric ALL ... more >> Relapsed Pediatric ALL Acute Lymphoblastic Leukemia Refractory Pediatric ALL Collapse <<Phase 1Terminated(The study was stopp... more >>ed due to poor accrual and lack of funding.) Collapse <<-United States, California ... more >> City of Hope Duarte, California, United States, 91010 Childrens Hospital Los Angeles Los Angeles, California, United States, 90027 Stanford University Medical Center Palo Alto, California, United States, 94304-1812 UCSF School of Medicine San Francisco, California, United States, 94143-0106 United States, Florida University of Miami Cancer Center Miami, Florida, United States, 33136 United States, Michigan C.S. Mott Children's Hospital Ann Arbor, Michigan, United States, 48109-0914 United States, Minnesota Childrens Hospital & Clinics of Minnesota Minneapolis, Minnesota, United States, 55404-4597 United States, New York New York University Medical Center New York, New York, United States, 10016 United States, Washington Seattle Children's Hospital Seattle, Washington, United States, 98105 Collapse <<
    NCT00036959Brain and Central Nervous Syst... more >>em Tumors Childhood Germ Cell Tumor Extragonadal Germ Cell Tumor Kidney Cancer Liver Cancer Neuroblastoma Ovarian Cancer Sarcoma Unspecified Childhood Solid Tumor, Protocol Specific Collapse <<Phase 1Completed-United States, Illinois ... more >> Children's Memorial Hospital - Chicago Chicago, Illinois, United States, 60614 United States, Maryland Warren Grant Magnuson Clinical Center - NCI Clinical Trials Referral Office Bethesda, Maryland, United States, 20892-1182 United States, Pennsylvania Children's Hospital of Philadelphia Philadelphia, Pennsylvania, United States, 19104-4318 Collapse <<
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  • 参考文献

实验方案

技术信息

CAS号 141430-65-1 储存条件
分子式 C18H17N3O4S 运输 蓝冰
分子量 371.41 别名 E7010
溶解度
DMSO210.0 mg/mL (565.4 mM)
Waterinsoluble
动物实验配方
IP2% DMSO+2% Tween80+30% PEG300+water4.2 mg/mLclear
PO0.5% CMC-Na34 mg/mLsuspension

大规格询价

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