CAS No.: 161814-49-9
Amprenavir/安瑞那韦 Catalog No. CSN16717
Synonyms: VX-478;141W94;KVX-478
Amprenavir is a protease inhibitor used to treat HIV infection which can form an inhibitor-enzyme complex with HIV protease.
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纯度 & 质量文件
批次:
靶点选择性
生物活性
靶点 HIV Protease
Ki:0.6nM- 描述
- 作用机制
- 临床研究
NCT号 适应症或疾病 临床期 招募状态 预计完成时间 地点 NCT00363142 HIV Infection ... more >> Infection, Human Immunodeficiency Virus Collapse << Phase 3 Completed - - NCT00363142 - - Completed - - NCT00450580 Infection, Human Immunodeficie... more >>ncy Virus I HIV-1 Infection Collapse << Phase 3 Completed - - - 更多
- 参考文献
- [1] Helsley RN, Sui Y, et al. Pregnane X receptor mediates dyslipidemia induced by the HIV protease inhibitor amprenavir in mice. Mol Pharmacol. 2013 Jun;83(6):1190-9.
- [2] Fung HB, Kirschenbaum HL, Hameed R. Amprenavir: a new human immunodeficiency virus type 1 protease inhibitor. Clin Ther. 2000 May;22(5):549-72.
- [3] Sadler BM, Stein DS. Clinical pharmacology and pharmacokinetics of amprenavir. Ann Pharmacother. 2002 Jan;36(1):102-18
- [4] Esposito V, Verdina A, Manente L, Spugnini EP, Viglietti R, Parrella R, Pagliano P, Parrella G, Galati R, De Luca A, Baldi A, Montesarchio V, Chirianni A. Amprenavir inhibits the migration in human hepatocarcinoma cell and the growth of xenografts. J Cell Physiol. 2013 Mar;228(3):640-5
实验方案
- 计算器
- 储存液制备
技术信息
| CAS号 | 161814-49-9 | 储存条件 |
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| 分子式 | C25H35N3O6S | 运输 | 蓝冰 | |||||||
| 分子量 | 505.63 | 别名 | VX-478;141W94;KVX-478;APV;Prozei;Agenerase;安瑞那韦 | |||||||
| 溶解度 |
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动物实验配方 |
| NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
|---|
| NCT00363142 | HIV Infection ... more >> Infection, Human Immunodeficiency Virus Collapse << | Phase 3 | Completed | - | - |
| NCT00363142 | - | - | Completed | - | - |
| NCT00450580 | Infection, Human Immunodeficie... more >>ncy Virus I HIV-1 Infection Collapse << | Phase 3 | Completed | - | - |
| NCT00002426 | HIV Infections | Not Applicable | Completed | - | - |
| NCT00259727 | - | - | Completed | - | United States, California ... more >> VA Medical Center, San Francisco San Francisco, California, United States, 94121 Collapse << |
| NCT00450580 | - | - | Completed | - | - |
| NCT00240552 | Infection, Human Immunodeficie... more >>ncy Virus Collapse << | Phase 4 | Completed | - | Switzerland ... more >> GSK Investigational Site Aarau, Switzerland, 5001 GSK Investigational Site Basel, Switzerland, 4031 GSK Investigational Site Bern, Switzerland, 3010 GSK Investigational Site Bruderholz, Switzerland, 4101 GSK Investigational Site La Chaux-de-Fonds, Switzerland, CH 2301 GSK Investigational Site Lausanne, Switzerland, 1011 GSK Investigational Site Lugano, Switzerland, 6900 GSK Investigational Site Luzern, Switzerland, 6000 GSK Investigational Site St Gallen, Switzerland, 9007 GSK Investigational Site Zurich, Switzerland, 8008 GSK Investigational Site Zurich, Switzerland, 8038 GSK Investigational Site Zurich, Switzerland, 8091 Collapse << |
| NCT01252940 | HIV-1 Infection | Phase 3 | Completed | - | - |
| NCT01077557 | - | - | Completed | - | - |
| NCT01252940 | - | - | Completed | - | - |
| NCT00039741 | - | - | Completed | - | - |
| NCT00039741 | HIV Infections | Phase 2 Phase 3 | Completed | - | - |
| NCT01209065 | Infections, Human Immunodefici... more >>ency Virus and Herpesviridae Collapse << | Phase 1 | Completed | - | United States, New York ... more >> GSK Investigational Site Buffalo, New York, United States, 14202 Collapse << |
| NCT00000919 | HIV Infections | Not Applicable | Completed | - | - |
| NCT00001119 | HIV Infections | Not Applicable | Completed | - | United States, California ... more >> San Francisco Dept of Hlth / AIDS Office San Francisco, California, United States, 94102 United States, Illinois Univ of Illinois Chicago / Howard Brown Hlth Ctr Chicago, Illinois, United States, 60612 United States, Massachusetts Fenway Community Health Ctr / HIVNET Boston, Massachusetts, United States, 02115 United States, Minnesota Univ of Minnesota Minneapolis, Minnesota, United States, 55455 United States, New York Bronx-Lebanon Hosp Ctr Bronx, New York, United States, 10453 New York Univ Med Ctr New York, New York, United States, 10016 United States, Ohio Univ of Cincinnati Cincinnati, Ohio, United States, 452670405 United States, Rhode Island Mem Hosp of Rhode Island Pawtucket, Rhode Island, United States, 02860 United States, Washington Seattle HIVNET Seattle, Washington, United States, 98104 Univ of Washington Seattle, Washington, United States, 98104 Fred Hutchinson Cancer Research Ctr Seattle, Washington, United States, 98109 Australia Saint Vincent's Hosp Med Centre Darlinghurst, Australia Collapse << |
| NCT00000918 | HIV Infections | Phase 2 | Completed | - | - |
| NCT00192660 | HIV-Associated Lipodystrophy S... more >>yndrome Cardiovascular Disease Collapse << | Phase 4 | Completed | - | Australia, New South Wales ... more >> St. Vincent's Hospital Sydney, New South Wales, Australia, 2010 Collapse << |
| NCT00040664 | HIV Infection | Phase 2 | Completed | - | - |
| NCT00002440 | HIV Infections | Phase 2 | Completed | - | United States, California ... more >> UCSD Treatment Ctr San Diego, California, United States, 921036329 United States, Connecticut Yale U / New Haven Med Ctr / AIDS Clinical Trials Unit New Haven, Connecticut, United States, 065102483 United States, Missouri Kansas City AIDS Research Consortium Kansas City, Missouri, United States, 64111 United States, New York NYU Med Ctr / Dept of Medicine / AIDS Clinical Trial New York, New York, United States, 10016 United States, North Carolina Carolinas Med Ctr Charlotte, North Carolina, United States, 28232 United States, Ohio Case Western Reserve Univ / AIDS Clinical Trials Unit Cleveland, Ohio, United States, 44106 United States, Pennsylvania Univ of Pittsburgh Med Ctr Pittsburgh, Pennsylvania, United States, 15213 United States, Tennessee Vanderbilt Univ Med Ctr Nashville, Tennessee, United States, 372321302 Collapse << |
| NCT00089583 | Infection, Human Immunodeficie... more >>ncy Virus I Collapse << | Phase 2 | Completed | - | - |
| NCT00307502 | HIV Infections | Phase 1 | Completed | - | Spain ... more >> Germans Trias i Pujol Hospital Badalona, Barcelona, Spain, 08916 Hospital de Figueres Figueras, Barcelona, Spain, 17600 Fundació Hospital-Asil de Granollers Granollers, Barcelona, Spain, 08400 Hospital de Vic Vic, Barcelona, Spain, 08500 Hospital Universitari Sant Joan de Reus Reus, Tarragona, Spain, 43201 Hospital de la Santa Creu i Sant Pau Barcelona, Spain, 08025 Collapse << |
| NCT00046033 | HIV Infections | Phase 2 | Completed | - | United States, Florida ... more >> Univ of Miami Miami, Florida, United States, 33136-1013 United States, Hawaii Univ of Hawaii Honolulu, Hawaii, United States, 96816-2396 United States, New York NYU/Bellevue New York, New York, United States, 10016 United States, Ohio Case Western Reserve Univ Cleveland, Ohio, United States, 44106 United States, Pennsylvania Univ of Pittsburgh Pittsburgh, Pennsylvania, United States, 15213-2582 United States, Texas Univ of Texas, Galveston Galveston, Texas, United States, 77555-0435 Collapse << |
| NCT00071760 | - | - | Active, not recruiting | - | - |
| NCT00006519 | HIV Infection | Phase 1 | Completed | - | United States, Maryland ... more >> National Cancer Institute (NCI) Bethesda, Maryland, United States, 20892 Collapse << |
| NCT00032669 | HIV Infections | Phase 1 | Completed | - | United States, Maryland ... more >> National Cancer Institute (NCI) Bethesda, Maryland, United States, 20892 Collapse << |
| NCT00071760 | Infection, Human Immunodeficie... more >>ncy Virus Collapse << | Phase 2 | Active, not recruiting | June 2021 | United States, Florida ... more >> GSK Investigational Site Jacksonville, Florida, United States, 32209 United States, North Carolina GSK Investigational Site Durham, North Carolina, United States, 27705 Argentina GSK Investigational Site Buenos Aires, Argentina, 1405 Mexico GSK Investigational Site Mexico, D.F., Mexico, 06720 GSK Investigational Site Mexico, Mexico, 6720 Portugal GSK Investigational Site Almada, Portugal, 2805-267 GSK Investigational Site Amadora, Portugal, 2700 GSK Investigational Site Lisboa, Portugal, 1649-035 Puerto Rico GSK Investigational Site San Juan, Puerto Rico, 00935 Russian Federation GSK Investigational Site Moscow, Russian Federation, 105275 GSK Investigational Site Moscow, Russian Federation, 129110 GSK Investigational Site St. Petersburg, Russian Federation, 196645 South Africa GSK Investigational Site Durban, KwaZulu- Natal, South Africa, 4013 GSK Investigational Site Parow Valley, Western Province, South Africa, 7505 GSK Investigational Site Soweto, South Africa, 2013 Collapse << |
| NCT00040664 | - | - | Completed | - | - |
| NCT02105987 | Infection, Human Immunodeficie... more >>ncy Virus Collapse << | Phase 3 | Completed | - | - |
| NCT00089583 | - | - | Completed | - | - |
| NCT01054638 | - | - | Completed | - | - |
| NCT00006578 | HIV Infections | Not Applicable | Withdrawn | - | United States, Colorado ... more >> Univ of Colorado Health Sciences Ctr Denver, Colorado, United States, 80262 United States, Florida Univ of Miami School of Medicine Miami, Florida, United States, 331361013 United States, Illinois Northwestern Univ Med School Chicago, Illinois, United States, 60611 Rush Presbyterian - Saint Luke's Med Ctr Chicago, Illinois, United States, 60612 United States, North Carolina Univ of North Carolina Chapel Hill, North Carolina, United States, 275997215 Collapse << |
| NCT02105987 | - | - | Completed | - | - |
| NCT01137981 | - | - | Recruiting | December 31, 2024 | United States, North Carolina ... more >> GSK Investigational Site Recruiting Wilmington, North Carolina, United States, 28405 Contact: US Clincal Trials Call Center 877-379-3718 Contact: EU Clinical Trials Call Center +44 (0) 20 8990 4466 Collapse << |
| NCT00296504 | Infection, Human Immunodeficie... more >>ncy Virus Collapse << | Phase 3 | Completed | - | United States, California ... more >> GSK Investigational Site Fountain Valley, California, United States, 92708 GSK Investigational Site San Francisco, California, United States, 94115-1931 United States, Colorado GSK Investigational Site Denver, Colorado, United States, 80262 United States, Florida GSK Investigational Site Fort Lauderdale, Florida, United States, 33145 GSK Investigational Site Orlando, Florida, United States, 32804 GSK Investigational Site Orlando, Florida, United States, 32806 GSK Investigational Site Sarasota, Florida, United States, 34239 GSK Investigational Site Tampa, Florida, United States, 33614 United States, New York GSK Investigational Site Manhasset, New York, United States, 11030 United States, Texas GSK Investigational Site Galveston, Texas, United States, 77555-1188 Brazil GSK Investigational Site Campinas, São Paulo, Brazil, 13083970 Chile GSK Investigational Site Santiago, Región Metro De Santiago, Chile France GSK Investigational Site Le Kremlin Bicêtre Cedex, France, 94275 GSK Investigational Site Marseille, France, 13005 GSK Investigational Site Paris Cedex 10, France, 75475 GSK Investigational Site Paris Cedex 20, France, 75970 GSK Investigational Site Vandoeuvre Les Nancy Cedex, France, 54511 GSK Investigational Site Villejuif Cedex, France, 94805 Italy GSK Investigational Site Genova, Liguria, Italy, 16128 Portugal GSK Investigational Site Coimbra, Portugal, 3000-075 Spain GSK Investigational Site Badajoz, Spain, 6080 GSK Investigational Site Barcelona, Spain, 08036 United Kingdom GSK Investigational Site London, United Kingdom, NW3 2QG GSK Investigational Site London, United Kingdom, SE1 7EH Collapse << |
| NCT00817765 | HIV Infection ... more >> Fungal Infection Collapse << | Phase 1 | Completed | - | Netherlands ... more >> Radboud University Nijmegen Medical Centre Nijmegen, Gelderland, Netherlands Collapse << |
| NCT00624195 | - | - | Completed | - | - |
| NCT00006152 | HIV Infections | Phase 2 | Completed | - | United States, Alabama ... more >> Univ of Alabama at Birmingham Birmingham, Alabama, United States, 35294 United States, California Univ of Southern California / LA County USC Med Ctr Los Angeles, California, United States, 900331079 Univ of California, San Diego San Diego, California, United States, 92103 United States, Colorado Univ of Colorado Health Sciences Ctr Denver, Colorado, United States, 80262 United States, Illinois Northwestern Univ Med School Chicago, Illinois, United States, 60611 The CORE Ctr Chicago, Illinois, United States, 60612 United States, Massachusetts Beth Israel Deaconess - West Campus Boston, Massachusetts, United States, 02215 United States, Missouri St Louis Regional Hosp / St Louis Regional Med Ctr St Louis, Missouri, United States, 63112 United States, New York Beth Israel Med Ctr New York, New York, United States, 10003 United States, North Carolina Univ of North Carolina Chapel Hill, North Carolina, United States, 275997215 Duke Univ Med Ctr Durham, North Carolina, United States, 27710 United States, South Carolina Julio Arroyo West Columbia, South Carolina, United States, 29169 United States, Texas Univ of Texas Galveston Galveston, Texas, United States, 775550435 Collapse << |
| NCT00624195 | HIV Infections | Phase 2 Phase 3 | Completed | - | United States, California ... more >> HIV Neurobehavioral Research Center, University of California San Diego San Diego, California, United States, 92103 University of California, San Francisco San Francisco, California, United States, 94110 United States, Maryland Johns Hopkins University- School of Medicine Baltimore, Maryland, United States, 21287 United States, Missouri Washington University St. Louis, Missouri, United States, 63110 United States, New York Mount Sinai Medical Center New York, New York, United States, 10024 Collapse << |
| NCT00296504 | - | - | Completed | - | - |
| NCT01290211 | Healthy | Phase 1 | Completed | - | Belgium ... more >> Pfizer Investigational Site Bruxelles, Belgium, B-1070 Collapse << |
| NCT00764465 | Healthy | Phase 2 | Completed | - | United States, New Jersey ... more >> Garden State Infectious Disease Associates,PA Voorhees, New Jersey, United States, 08043 Collapse << |
| NCT00481182 | Healthy Subjects | Phase 1 | Completed | - | United States, Maryland ... more >> GSK Investigational Site Baltimore, Maryland, United States, 21287-5554 United States, New York GSK Investigational Site Buffalo, New York, United States, 14215-1199 Collapse << |
| NCT00764465 | - | - | Completed | - | - |
| NCT00002216 | HIV Infections | Not Applicable | Completed | - | United States, Pennsylvania ... more >> Anderson Clinical Research Pittsburgh, Pennsylvania, United States, 15213 Collapse << |
| NCT00000940 | HIV Infections | Phase 2 | Completed | - | United States, California ... more >> USC CRS Los Angeles, California, United States, 90033 UCLA CARE Center CRS Los Angeles, California, United States, 90035 Ucsd, Avrc Crs San Diego, California, United States, 92103 Ucsf Aids Crs San Francisco, California, United States, 94110 United States, Colorado University of Colorado Hospital CRS Aurora, Colorado, United States, 80045 United States, Hawaii Univ. of Hawaii at Manoa, Leahi Hosp. Honolulu, Hawaii, United States, 96816 United States, Massachusetts Massachusetts General Hospital ACTG CRS Boston, Massachusetts, United States, 02114 SSTAR, Family Healthcare Ctr. Fall River, Massachusetts, United States, 02720 United States, Missouri Washington U CRS St. Louis, Missouri, United States, 63110 United States, New York Beth Israel Med. Ctr. ACTU New York, New York, United States, 10003 NY Univ. HIV/AIDS CRS New York, New York, United States, 10016 Columbia P&S CRS New York, New York, United States, 10032 AIDS Care CRS Rochester, New York, United States, 14607 McCree McCuller Wellness Ctr. at the Connection, Infectious Disease Unit Rochester, New York, United States, 14642 Univ. of Rochester ACTG CRS Rochester, New York, United States, 14642 United States, North Carolina Unc Aids Crs Chapel Hill, North Carolina, United States, 27514 United States, Pennsylvania Hosp. of the Univ. of Pennsylvania CRS Philadelphia, Pennsylvania, United States, 19104 United States, Rhode Island The Miriam Hosp. ACTG CRS Providence, Rhode Island, United States, 02906 Collapse << |
| NCT01140412 | Healthy | Phase 1 | Terminated(The trial premature... more >>ly terminated on November 1, 2010, due to healthy volunteer participants experiencing non-serious fosamprenavir-related skin rash.) Collapse << | - | Singapore ... more >> Pfizer Investigational Site Singapore, Singapore, 188770 Collapse << |
| NCT00335270 | HIV | Phase 4 | Completed | - | United States, Florida ... more >> University of Miami School of Medicine Miami, Florida, United States, 33136 Collapse << |
| NCT00614991 | - | - | Completed | - | - |
| NCT00614991 | Healthy | Not Applicable | Completed | - | - |
| NCT00802074 | Healthy | Not Applicable | Completed | - | United States, New Jersey ... more >> Garden State Infectious Disease Associates, PA Voorhees, New Jersey, United States, 08043 Collapse << |
| NCT00056641 | HIV Infections | Phase 2 | Completed | - | - |
| NCT00002233 | HIV Infections | Phase 2 | Completed | - | United States, New York ... more >> Aaron Diamond AIDS Rsch Ctr / Rockefeller Univ New York, New York, United States, 10021 United States, Rhode Island Miriam Hosp / Family Healthcare Ctr at SSTAR Providence, Rhode Island, United States, 02906 Collapse << |
| NCT00802074 | - | - | Completed | - | - |
| NCT00005017 | HIV Infections | Phase 4 | Unknown | - | United States, North Carolina ... more >> Jaime Hernandez Research Triangle Park, North Carolina, United States, 27709 Collapse << |
| NCT00148785 | HIV Infections | Phase 4 | Completed | - | United States, Georgia ... more >> Grady Infectious Diseases Program Atlanta, Georgia, United States, 30308 Collapse << |
| NCT00001968 | Acquired Immunodeficiency Synd... more >>rome HIV Infections Collapse << | Phase 1 | Completed | - | United States, Maryland ... more >> National Institute of Allergy and Infectious Diseases (NIAID) Bethesda, Maryland, United States, 20892 Collapse << |
| NCT00001133 | HIV Infections | Phase 1 | Completed | - | United States, Alabama ... more >> Alabama Therapeutics CRS Birmingham, Alabama, United States, 35294 United States, California USC CRS Los Angeles, California, United States, 900331079 Ucsf Aids Crs San Francisco, California, United States, 94110 United States, Maryland Johns Hopkins Adult AIDS CRS Baltimore, Maryland, United States, 21287 United States, New York NY Univ. HIV/AIDS CRS New York, New York, United States, 10016 United States, Ohio Univ. of Cincinnati CRS Cincinnati, Ohio, United States, 452670405 United States, Pennsylvania Pitt CRS Pittsburgh, Pennsylvania, United States, 15213 Collapse << |
| NCT00002423 | HIV Infections | Phase 2 | Completed | - | United States, California ... more >> Saint Francis Mem Hosp San Francisco, California, United States, 94109 United States, District of Columbia Georgetown Univ Med Ctr Washington, District of Columbia, United States, 20007 United States, Florida IDC Research Initiative Altamonte Springs, Florida, United States, 32701 United States, Maryland Natl Institute of Allergy and Infectious Diseases Bethesda, Maryland, United States, 20892 United States, Missouri Kansas City AIDS Research Consortium Kansas City, Missouri, United States, 64111 United States, New York Bentley-Salick Med Practice New York, New York, United States, 10011 United States, Oklahoma Associates in Med and Mental Health Tulsa, Oklahoma, United States, 74114 United States, Oregon Portland Veterans Adm Med Ctr / Rsch & Education Grp Portland, Oregon, United States, 972109951 Collapse << |
| NCT00002213 | HIV Infections | Phase 2 | Completed | - | United States, California ... more >> East Bay AIDS Ctr Berkeley, California, United States, 94705 Kraus Med Partners Los Angeles, California, United States, 90036 United States, Illinois Northwestern Univ Med School AIDS Treatment Unit Chicago, Illinois, United States, 60611 United States, Maryland Niaid / Nih Bethesda, Maryland, United States, 20892 United States, Massachusetts Beth Israel Deaconess Med Ctr Boston, Massachusetts, United States, 02215 United States, New York Saint Vincents Hosp / AIDS Ctr / 4th Floor New York, New York, United States, 10011 United States, North Carolina Univ of North Carolina Chapel Hill Chapel Hill, North Carolina, United States, 27499 United States, Ohio Univ Int Med Assoc Inc / Holmes Hosp / U of Cincinnati Cincinnati, Ohio, United States, 45267 United States, Rhode Island The Miriam Hosp Providence, Rhode Island, United States, 02906 Collapse << |
| NCT00002183 | HIV Infections | Phase 1 | Completed | - | United States, California ... more >> UCSD San Diego, California, United States, 92103 United States, Colorado Univ of Colorado Health Sciences Ctr Denver, Colorado, United States, 80262 United States, Georgia AIDS Research Consortium of Atlanta Atlanta, Georgia, United States, 30308 Collapse << |
| NCT00002372 | HIV Infections | Phase 1 | Completed | - | United States, California ... more >> Univ of California / San Diego Treatment Ctr San Diego, California, United States, 92103 ViRx Inc San Francisco, California, United States, 94109 United States, North Carolina Univ of North Carolina at Chapel Hill / Duke Univ Med Ctr Durham, North Carolina, United States, 27710 Collapse << |
| NCT00001766 | HIV Infection | Phase 1 | Completed | - | United States, Maryland ... more >> National Institute of Allergy and Infectious Diseases (NIAID) Bethesda, Maryland, United States, 20892 Collapse << |
| NCT00002195 | HIV Infections | Phase 3 | Completed | - | United States, California ... more >> Pacific Oaks Research Beverly Hills, California, United States, 90211 United States, District of Columbia Dr Bruce Rashbaum Washington, District of Columbia, United States, 20037 United States, Florida Community Research Initiative of South Florida Coral Gables, Florida, United States, 33146 Community Research Initiative of Central Florida Maitland, Florida, United States, 32751 Univ of Miami School of Medicine Miami, Florida, United States, 33136 United States, Illinois Chicago Ctr for Clinical Research Chicago, Illinois, United States, 60610 United States, Massachusetts Community Research Initiative of New England Brookline, Massachusetts, United States, 02445 United States, New York Saint Vincent's AIDS Ctr New York, New York, United States, 10011 United States, Tennessee Methodist Hosp Memphis, Tennessee, United States, 38104 Collapse << |
| NCT00002217 | HIV Infections | Not Applicable | Completed | - | United States, Pennsylvania ... more >> Anderson Clinical Research Pittsburgh, Pennsylvania, United States, 15213 Collapse << |
| NCT00006617 | HIV Infections | Not Applicable | Completed | - | United States, New York ... more >> Aaron Diamond AIDS Res Ctr New York, New York, United States, 10016 Collapse << |
| NCT00001085 | HIV Infections | Phase 2 | Completed | - | United States, Alabama ... more >> Alabama Therapeutics CRS Birmingham, Alabama, United States, 35294 United States, California USC CRS Los Angeles, California, United States, 900331079 United States, Colorado University of Colorado Hospital CRS Aurora, Colorado, United States, 80262 United States, Florida Univ. of Miami AIDS CRS Miami, Florida, United States, 331361013 United States, Georgia The Ponce de Leon Ctr. CRS Atlanta, Georgia, United States, 30308 United States, Illinois Northwestern University CRS Chicago, Illinois, United States, 60611 Cook County Hosp. CORE Ctr. Chicago, Illinois, United States, 60612 Rush Univ. Med. Ctr. ACTG CRS Chicago, Illinois, United States, 60612 United States, Massachusetts Bmc Actg Crs Boston, Massachusetts, United States, 02118 Beth Israel Deaconess Med. Ctr., ACTG CRS Boston, Massachusetts, United States, 02215 United States, Missouri St. Louis ConnectCare, Infectious Diseases Clinic St Louis, Missouri, United States, 63112 Washington U CRS St. Louis, Missouri, United States United States, New York NY Univ. HIV/AIDS CRS New York, New York, United States, 10016 United States, North Carolina Unc Aids Crs Chapel Hill, North Carolina, United States, 275997215 United States, Pennsylvania Hosp. of the Univ. of Pennsylvania CRS Philadelphia, Pennsylvania, United States, 19104 Collapse << |
| NCT00000912 | HIV Infections | Phase 2 | Completed | - | - |
| NCT00005762 | HIV Infections | Not Applicable | Completed | - | United States, California ... more >> Stanford CRS Palo Alto, California, United States, 943055107 United States, Colorado University of Colorado Hospital CRS Aurora, Colorado, United States, 80262 United States, Hawaii Univ. of Hawaii at Manoa, Leahi Hosp. Honolulu, Hawaii, United States, 96816 United States, Indiana Indiana Univ. School of Medicine, Infectious Disease Research Clinic Indianapolis, Indiana, United States, 462025250 United States, Maryland Johns Hopkins Adult AIDS CRS Baltimore, Maryland, United States United States, Ohio The Ohio State University Medical Center Columbus, Ohio, United States, 43210 United States, Tennessee Vanderbilt Univ. Med. Ctr., AIDS Clinical Trials Ctr. Nashville, Tennessee, United States, 37203 United States, Washington University of Washington AIDS CRS Seattle, Washington, United States, 98104 Collapse << |
| NCT00002202 | HIV Infections | Phase 3 | Completed | - | - |
| NCT00002419 | HIV Infections | Phase 2 | Completed | - | United States, California ... more >> Pacific Oaks Med Group Beverly Hills, California, United States, 90211 United States, Colorado Univ of Colorado / Health Science Ctr Denver, Colorado, United States, 80262 United States, Georgia AIDS Research Consortium of Atlanta Atlanta, Georgia, United States, 30308 United States, Rhode Island Brown Univ School of Medicine Providence, Rhode Island, United States, 02908 United States, Virginia Hampton Roads Med Specialists Hampton, Virginia, United States, 23666 Collapse << |
| NCT00002239 | HIV Infections | Phase 2 | Completed | - | United States, California ... more >> Pacific Oaks Research Beverly Hills, California, United States, 90211 UCLA Care Ctr Los Angeles, California, United States, 90095 ViRx Inc Palm Springs, California, United States, 92262 Donald Northfelt Palm Springs, California, United States, 92270 UCSD San Diego, California, United States, 92103 ViRx Inc San Francisco, California, United States, 94109 Quest Clinical Research San Francisco, California, United States, 94115 United States, District of Columbia Dupont Circle Physicians Group Washington, District of Columbia, United States, 200091104 United States, Florida IDC Research Initiative Altamonte Springs, Florida, United States, 32701 Gary Richmond MD Fort Lauderdale, Florida, United States, 33316 United States, Georgia AIDS Research Consortium of Atlanta Atlanta, Georgia, United States, 30308 United States, Maryland Johns Hopkins Hosp Baltimore, Maryland, United States, 21287 United States, Missouri Washington Univ School of Medicine St. Louis, Missouri, United States, 63110 United States, New York New York Univ Med Ctr New York, New York, United States, 10016 United States, North Carolina Trimeris Inc Durham, North Carolina, United States, 27707 United States, Oklahoma Associates of Med and Mental Health Tulsa, Oklahoma, United States, 74114 United States, Pennsylvania Pennsylvania Oncology and Hematology Associates Philadelphia, Pennsylvania, United States, 19106 Philadelphia FIGHT Philadelphia, Pennsylvania, United States, 19107 Univ of Pittsburgh Pittsburgh, Pennsylvania, United States, 15261 United States, Texas Central Texas Clinical Research Austin, Texas, United States, 78705 Collapse << |
| NCT00006591 | HIV Infections | Not Applicable | Unknown | - | United States, Texas ... more >> Gathe, Joseph, M.D. Houston, Texas, United States, 77004 Collapse << |
| NCT00038532 | HIV Infections | Phase 2 | Completed | - | - |
| NCT00001758 | HIV Infection | Phase 2 | Completed | - | United States, Maryland ... more >> National Institute of Allergy and Infectious Diseases (NIAID) Bethesda, Maryland, United States, 20892 Collapse << |
| NCT00002193 | HIV Infections | Phase 3 | Completed | - | United States, Florida ... more >> Children's Diagnostic Treatment Ctr Fort Lauderdale, Florida, United States, 33301 United States, Tennessee Saint Jude Children's Hosp / Dept of Infect Diseases Memphis, Tennessee, United States, 38105 Collapse << |
| NCT00001095 | HIV Infections | Phase 2 | Completed | - | United States, California ... more >> Univ of Southern California / LA County USC Med Ctr Los Angeles, California, United States, 900331079 United States, Colorado Univ of Colorado Health Sciences Ctr Denver, Colorado, United States, 80262 United States, Florida Univ of Miami School of Medicine Miami, Florida, United States, 331361013 United States, Georgia Emory Univ Atlanta, Georgia, United States, 30308 United States, Illinois Cook County Hosp Chicago, Illinois, United States, 60612 United States, Massachusetts Boston Med Ctr Boston, Massachusetts, United States, 02118 Beth Israel Deaconess - West Campus Boston, Massachusetts, United States, 02215 United States, Missouri St Louis Regional Hosp / St Louis Regional Med Ctr St Louis, Missouri, United States, 63112 United States, New York Bellevue Hosp / New York Univ Med Ctr New York, New York, United States, 10016 United States, North Carolina Univ of North Carolina Chapel Hill, North Carolina, United States, 275997215 United States, Pennsylvania Univ of Pennsylvania at Philadelphia Philadelphia, Pennsylvania, United States, 19104 United States, South Carolina Julio Arroyo West Columbia, South Carolina, United States, 29169 Collapse << |
| NCT00002205 | HIV Infections | Not Applicable | Completed | - | United States, North Carolina ... more >> Glaxo Wellcome Inc Research Triangle Park, North Carolina, United States, 277093398 Collapse << |
| NCT00196625 | HIV Infections | Phase 2 | Completed | - | - |
| NCT00002417 | HIV Infections | Not Applicable | Completed | - | United States, North Carolina ... more >> Glaxo Wellcome Inc Research Triangle Park, North Carolina, United States, 27709 Collapse << |
| NCT00038519 | HIV Infections | Phase 2 Phase 3 | Completed | - | - |
| NCT00002405 | HIV Infections | Not Applicable | Completed | - | United States, North Carolina ... more >> Glaxo Wellcome Inc Research Triangle Park, North Carolina, United States, 277093398 Collapse << |
| NCT00002245 | HIV Infections | Phase 3 | Completed | - | United States, California ... more >> LAC / USC Med Ctr / Infectious Diseases Los Angeles, California, United States, 90033 Collapse << |
| NCT02182765 | HIV Infections | Phase 1 | Terminated | - | - |
| 靶点 | Description | IC50 |
|---|---|---|
| HIV Protease | Ki:0.6nM |
