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CAS No.: 2095393-15-8
Synonyms: MK-1026;nemtabrutinib
ARQ-531 is a potent and orally active BTK inhibitor with potential antineoplastic activity.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT03162536 | Lymphoma, B-Cell ... more >> Small Lymphocytic Lymphoma Chronic Lymphocytic Leukemia Waldenstrom Macroglobulinemia Mantle Cell Lymphoma Diffuse Large B Cell Lymphoma Collapse << | Phase 1 | Recruiting | April 2019 | United States, Ohio ... more >> Wexner Medical Center at The Ohio State University Recruiting Columbus, Ohio, United States, 43210 Contact 781-994-0300 ClinicalTrials@arqule.com United States, Tennessee Sarah Cannon Research Institute Recruiting Nashville, Tennessee, United States, 37203 Contact 781-994-0300 ClinicalTrials@arqule.com United States, Utah University of Utah, Huntsman Cancer Institute Recruiting Salt Lake City, Utah, United States, 84112 Contact 781-994-0300 ClinicalTrials@arqule.com Collapse << |
实验方案
技术信息
CAS号 | 2095393-15-8 | 储存条件 |
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分子式 | C25H23ClN4O4 | 运输 | 蓝冰 | |||||||
分子量 | 478.93 | 别名 | MK-1026;nemtabrutinib | |||||||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT03162536 | Lymphoma, B-Cell ... more >> Small Lymphocytic Lymphoma Chronic Lymphocytic Leukemia Waldenstrom Macroglobulinemia Mantle Cell Lymphoma Diffuse Large B Cell Lymphoma Collapse << | Phase 1 | Recruiting | April 2019 | United States, Ohio ... more >> Wexner Medical Center at The Ohio State University Recruiting Columbus, Ohio, United States, 43210 Contact 781-994-0300 ClinicalTrials@arqule.com United States, Tennessee Sarah Cannon Research Institute Recruiting Nashville, Tennessee, United States, 37203 Contact 781-994-0300 ClinicalTrials@arqule.com United States, Utah University of Utah, Huntsman Cancer Institute Recruiting Salt Lake City, Utah, United States, 84112 Contact 781-994-0300 ClinicalTrials@arqule.com Collapse << |
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