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CAS No.: 1554458-53-5
Synonyms: N/A
BAY1217389 is a potent, and selective inhibitor of the monopolar spindle 1 (MPS1) kinase with an IC50 value less than 10 nM.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT02366949 | Medical Oncology | Phase 1 | Active, not recruiting | June 28, 2019 | United States, California ... more >> Santa Monica, California, United States, 90403 United States, Colorado Denver, Colorado, United States, 80262 United States, Connecticut New Haven, Connecticut, United States, 06520 United States, New Jersey Hackensack, New Jersey, United States, 07601-1991 United States, Texas Houston, Texas, United States, 77030 San Antonio, Texas, United States, 78229-3307 Netherlands Rotterdam, Netherlands, 3075 EA Collapse << |
实验方案
技术信息
CAS号 | 1554458-53-5 | 储存条件 |
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分子式 | C27H24F5N5O3 | 运输 | 蓝冰 | |
分子量 | 561.50 | 别名 | N/A |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT02366949 | Medical Oncology | Phase 1 | Active, not recruiting | June 28, 2019 | United States, California ... more >> Santa Monica, California, United States, 90403 United States, Colorado Denver, Colorado, United States, 80262 United States, Connecticut New Haven, Connecticut, United States, 06520 United States, New Jersey Hackensack, New Jersey, United States, 07601-1991 United States, Texas Houston, Texas, United States, 77030 San Antonio, Texas, United States, 78229-3307 Netherlands Rotterdam, Netherlands, 3075 EA Collapse << |
靶点 | Description | IC50 |
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