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CAS No.: 90357-06-5

Bicalutamide/比卡鲁胺 Catalog No. CSN12437

Synonyms: ICI-176334;ZD 176334;Abbreviation: CDX. US brand name: Casodex. Foreign brand name: Cosudex

Bicalutamide is non-steroidal androgen receptor antagonist with IC50 value of 190 nM.

规格 价格 促销价格 库存 数量
纯度 & 质量文件 批次:

靶点选择性

生物活性

  • 靶点Androgen Receptor

    IC50:0.16μM
  • 描述
  • 细胞研究
  • Cell Data
  • 更多
  • 动物研究
    剂量

    Rat: 10 mg/kg, 20 mg/kg[3] (p.o.); 1 mg/kg - 250 mg/kg[4] (p.o.) Nude mice: 150 mg/kg[5] (p.o.), 50 mg/kg - 100 mg/kg[6] (p.o.) Dog: 0.1 mg/kg - 100 mg/kg[4] (p.o.); 0.25 mg/kg, 2.5 mg/kg[4] (i.v.)

    给药途径

    p.o.

    动物药代数据
    AnimalRats[4]Dogs[4]
    Dose50 mg/kg (male)2.5 mg/kg
    Administrationp.o.p.o. or i.v.
    F0.35766.5 ± 4.0% (p.o.)
    Tmax12 h16.6 ± 12.7 h (p.o.)
    t1/2λ18.6 h5.49 ± 0.53 days (p.o.)
    7.47 ± 0.90 days (i.v.)
    CL54.6 ± 9.2 μl/min/kg (i.v.)
    Cmax15.4 μg/ml2.44 ± 0.27 μg/ml (p.o.)
    Vλ0.852 ± 0.194 L/kg (i.v.)
    AUC379 μg·h/ml519 ± 34 μg·h/ml (p.o.)
    796 ± 148 μg·h/ml (i.v.)
  • 临床研究
  • NCT号适应症或疾病临床期招募状态预计完成时间地点
    NCT00298155Cancer Prosta... more >>te Neoplasms Collapse <<Phase 2Completed-United States, Washington ... more >> Veterans' Administration Puget Sound Health Care System (VAPSHCS) Seattle, Washington, United States, 98108-1532 University of Washington Seattle, Washington, United States, 98195-6158 Collapse <<
    NCT00298155--Completed--
    NCT02064036Adenocarcinoma of the ProstateNot ApplicableRecruitingOctober 2018United States, California ... more >> UC Davis Sacramento Cancer Center Dept of Radiation Oncology Recruiting Sacramento, California, United States, 95817 Contact: Richard Valicenti, MD    916-724-8295    rkvalicenti@ucdavis.edu    Principal Investigator: Richard Valicenti, MD Collapse <<
  • 更多

实验方案

技术信息

CAS号 90357-06-5 储存条件
分子式 C18H14F4N2O4S 运输 蓝冰
分子量 430.37 别名 ICI-176334;ZD 176334;Abbreviation: CDX. US brand name: Casodex. Foreign brand name: Cosudex;比卡鲁胺
溶解度
DMSO135.0 mg/mL (313.7 mM)
Waterinsoluble
动物实验配方
IP2% DMSO+2% Tween80+40% PEG300+water2.2 mg/mLclear
PO0.5% CMC-Na26 mg/mLsuspension

大规格询价

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